SG176055A1 - Compositions and methods for drug delivery - Google Patents

Compositions and methods for drug delivery Download PDF

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Publication number
SG176055A1
SG176055A1 SG2011083789A SG2011083789A SG176055A1 SG 176055 A1 SG176055 A1 SG 176055A1 SG 2011083789 A SG2011083789 A SG 2011083789A SG 2011083789 A SG2011083789 A SG 2011083789A SG 176055 A1 SG176055 A1 SG 176055A1
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SG
Singapore
Prior art keywords
particle
cis
disease
particles
group
Prior art date
Application number
SG2011083789A
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English (en)
Inventor
Barrett Rabinow
Shawn F Bairstow
Mahesh V Chaubal
Sarah Lee
Jane Werling
Original Assignee
Baxter Int
Baxter Healthcare Sa
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Application filed by Baxter Int, Baxter Healthcare Sa filed Critical Baxter Int
Publication of SG176055A1 publication Critical patent/SG176055A1/en

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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SG2011083789A 2009-05-15 2010-05-13 Compositions and methods for drug delivery SG176055A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12/467,230 US10952965B2 (en) 2009-05-15 2009-05-15 Compositions and methods for drug delivery
PCT/US2010/034711 WO2010132664A1 (en) 2009-05-15 2010-05-13 Compositions and methods for drug delivery

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SG176055A1 true SG176055A1 (en) 2011-12-29

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US (2) US10952965B2 (https=)
EP (1) EP2429493B1 (https=)
JP (1) JP5668055B2 (https=)
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