SG160438A1 - Process for preparing pyrido[2,3-d]pyrimidin-7-one and 3,4-dihydropyrimido[4,5- d]pyrimidin-2(1h)-one derivatives - Google Patents

Process for preparing pyrido[2,3-d]pyrimidin-7-one and 3,4-dihydropyrimido[4,5- d]pyrimidin-2(1h)-one derivatives

Info

Publication number
SG160438A1
SG160438A1 SG201002044-4A SG2010020444A SG160438A1 SG 160438 A1 SG160438 A1 SG 160438A1 SG 2010020444 A SG2010020444 A SG 2010020444A SG 160438 A1 SG160438 A1 SG 160438A1
Authority
SG
Singapore
Prior art keywords
pyrimidin
dihydropyrimido
derivatives
preparing pyrido
pyrido
Prior art date
Application number
SG201002044-4A
Other languages
English (en)
Inventor
James Francis Callahan
Jeffrey Boehm
Zehong Wan
Hongxing Yan
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of SG160438A1 publication Critical patent/SG160438A1/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SG201002044-4A 2005-03-25 2006-03-24 Process for preparing pyrido[2,3-d]pyrimidin-7-one and 3,4-dihydropyrimido[4,5- d]pyrimidin-2(1h)-one derivatives SG160438A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US66515405P 2005-03-25 2005-03-25

Publications (1)

Publication Number Publication Date
SG160438A1 true SG160438A1 (en) 2010-04-29

Family

ID=37053945

Family Applications (1)

Application Number Title Priority Date Filing Date
SG201002044-4A SG160438A1 (en) 2005-03-25 2006-03-24 Process for preparing pyrido[2,3-d]pyrimidin-7-one and 3,4-dihydropyrimido[4,5- d]pyrimidin-2(1h)-one derivatives

Country Status (18)

Country Link
US (3) US7479558B2 (ru)
EP (1) EP1865959A2 (ru)
JP (1) JP2008537937A (ru)
KR (1) KR20080002865A (ru)
CN (1) CN101495475A (ru)
AR (1) AR059937A1 (ru)
AU (1) AU2006229995A1 (ru)
CA (1) CA2603163A1 (ru)
EA (1) EA200702073A1 (ru)
IL (1) IL186422A0 (ru)
MA (1) MA29391B1 (ru)
MX (1) MX2007012951A (ru)
NO (1) NO20075232L (ru)
NZ (1) NZ562433A (ru)
SG (1) SG160438A1 (ru)
TW (1) TW200735876A (ru)
WO (1) WO2006104917A2 (ru)
ZA (1) ZA200708524B (ru)

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PE20100737A1 (es) * 2005-03-25 2010-11-27 Glaxo Group Ltd Nuevos compuestos
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WO2016014542A1 (en) 2014-07-21 2016-01-28 Dana-Farber Cancer Institute, Inc. Imidazolyl kinase inhibitors and uses thereof
EP3172213B1 (en) 2014-07-21 2021-09-22 Dana-Farber Cancer Institute, Inc. Macrocyclic kinase inhibitors and uses thereof
AU2015300782B2 (en) 2014-08-08 2020-04-16 Dana-Farber Cancer Institute, Inc. Uses of salt-inducible kinase (SIK) inhibitors
US20190060286A1 (en) 2016-02-29 2019-02-28 University Of Florida Research Foundation, Incorpo Chemotherapeutic Methods
KR20190075043A (ko) 2016-07-05 2019-06-28 더 브로드 인스티튜트, 인코퍼레이티드 비시클릭 우레아 키나제 억제제 및 그의 용도
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RU2019129727A (ru) 2017-02-28 2021-03-30 Зэ Дженерал Хоспитал Корпорэйшн Применения пиримидопиримидинонов в качестве ингибиторов sik
WO2019168874A1 (en) 2018-02-27 2019-09-06 The Research Foundation For The State University Of New York Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same
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WO2006104917A3 (en) 2009-04-16
ZA200708524B (en) 2009-08-26
AU2006229995A1 (en) 2006-10-05
NO20075232L (no) 2007-11-28
US20080096905A1 (en) 2008-04-24
WO2006104917A2 (en) 2006-10-05
CN101495475A (zh) 2009-07-29
US20060258687A1 (en) 2006-11-16
IL186422A0 (en) 2009-02-11
NZ562433A (en) 2010-12-24
AR059937A1 (es) 2008-05-14
EA200702073A1 (ru) 2008-12-30
CA2603163A1 (en) 2006-10-05
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MA29391B1 (fr) 2008-04-01

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