SG10202101389TA - Crystalline forms of a bruton’s tyrosine kinase inhibitor - Google Patents

Crystalline forms of a bruton’s tyrosine kinase inhibitor

Info

Publication number
SG10202101389TA
SG10202101389TA SG10202101389TA SG10202101389TA SG10202101389TA SG 10202101389T A SG10202101389T A SG 10202101389TA SG 10202101389T A SG10202101389T A SG 10202101389TA SG 10202101389T A SG10202101389T A SG 10202101389TA SG 10202101389T A SG10202101389T A SG 10202101389TA
Authority
SG
Singapore
Prior art keywords
bruton
tyrosine kinase
kinase inhibitor
crystalline forms
crystalline
Prior art date
Application number
SG10202101389TA
Other languages
English (en)
Inventor
Mark Smyth
Erick Goldman
David Wirth
Norbert Purro
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49712527&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10202101389T(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of SG10202101389TA publication Critical patent/SG10202101389TA/en

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    • C07—ORGANIC CHEMISTRY
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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  • Health & Medical Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
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  • Molecular Biology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
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  • Pain & Pain Management (AREA)
  • Mechanical Engineering (AREA)
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  • Inorganic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
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  • Ophthalmology & Optometry (AREA)
SG10202101389TA 2012-06-04 2013-06-03 Crystalline forms of a bruton’s tyrosine kinase inhibitor SG10202101389TA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261655381P 2012-06-04 2012-06-04

Publications (1)

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SG10202101389TA true SG10202101389TA (en) 2021-03-30

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SG11201408067YA SG11201408067YA (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor
SG10202101389TA SG10202101389TA (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton’s tyrosine kinase inhibitor

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US (25) US9296753B2 (he)
EP (1) EP2854859A4 (he)
JP (8) JP6236071B2 (he)
KR (7) KR20190040370A (he)
CN (2) CN104736178A (he)
AR (2) AR092844A1 (he)
AU (6) AU2013271918C1 (he)
BR (1) BR112014030424A8 (he)
CA (4) CA2991994C (he)
CL (3) CL2014003306A1 (he)
CO (1) CO7240408A2 (he)
CR (1) CR20140558A (he)
DO (3) DOP2014000274A (he)
EA (1) EA201492082A1 (he)
EC (2) ECSP14033163A (he)
GT (1) GT201400281A (he)
HK (1) HK1208803A1 (he)
IL (3) IL235894B (he)
JO (2) JO3754B1 (he)
MA (2) MA41654B2 (he)
MX (2) MX348290B (he)
MY (2) MY187999A (he)
NZ (4) NZ737725A (he)
PE (3) PE20150174A1 (he)
PH (2) PH12014502681A1 (he)
SG (2) SG11201408067YA (he)
TN (1) TN2014000492A1 (he)
TW (3) TWI662964B (he)
UA (2) UA114421C2 (he)
UY (2) UY39740A (he)
WO (1) WO2013184572A1 (he)
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Families Citing this family (119)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2201840B1 (en) 2006-09-22 2011-11-02 Pharmacyclics, Inc. Inhibitors of Bruton's Tyrosine Kinase
US20120101114A1 (en) 2007-03-28 2012-04-26 Pharmacyclics, Inc. Inhibitors of bruton's tyrosine kinase
EP2307025B1 (en) 2008-07-16 2017-09-20 Pharmacyclics LLC Inhibitors of bruton's tyrosine kinase for the treatment of solid tumors
US8491927B2 (en) * 2009-12-02 2013-07-23 Nimble Epitech, Llc Pharmaceutical composition containing a hypomethylating agent and a histone deacetylase inhibitor
CA3113343A1 (en) 2010-06-03 2011-12-08 Pharmacyclics Llc Use of inhibitors of bruton's tyrosine kinase (btk) in the treatment of follicular lymphoma
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