SG10201407453TA - Kinase inhibitors - Google Patents

Kinase inhibitors

Info

Publication number
SG10201407453TA
SG10201407453TA SG10201407453TA SG10201407453TA SG10201407453TA SG 10201407453T A SG10201407453T A SG 10201407453TA SG 10201407453T A SG10201407453T A SG 10201407453TA SG 10201407453T A SG10201407453T A SG 10201407453TA SG 10201407453T A SG10201407453T A SG 10201407453TA
Authority
SG
Singapore
Prior art keywords
provides
protein kinase
present
kinase inhibitors
pyrropyrimidine
Prior art date
Application number
SG10201407453TA
Other languages
English (en)
Inventor
Jaekyoo Lee
Ho-Juhn Song
Jong Sung Koh
Hee Kyu Lee
Youngsam Kim
Hong Woo Kim
Sunhwa Chang
Sun-Hee Lim
Jang-Sik Choi
Jung-Ho Kim
Se-Won Kim
Original Assignee
Genosco
Oscotec Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genosco, Oscotec Inc filed Critical Genosco
Publication of SG10201407453TA publication Critical patent/SG10201407453TA/en

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

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  • Neurology (AREA)
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SG10201407453TA 2009-11-13 2010-11-12 Kinase inhibitors SG10201407453TA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US26110009P 2009-11-13 2009-11-13

Publications (1)

Publication Number Publication Date
SG10201407453TA true SG10201407453TA (en) 2014-12-30

Family

ID=43992073

Family Applications (1)

Application Number Title Priority Date Filing Date
SG10201407453TA SG10201407453TA (en) 2009-11-13 2010-11-12 Kinase inhibitors

Country Status (17)

Country Link
US (1) US8629132B2 (es)
EP (1) EP2498607B1 (es)
JP (1) JP5740409B2 (es)
KR (1) KR101663637B1 (es)
CN (1) CN102811619B (es)
BR (1) BR112012011287B1 (es)
CA (1) CA2780892C (es)
CL (1) CL2012001221A1 (es)
EA (1) EA024729B1 (es)
HK (1) HK1179477A1 (es)
IL (1) IL219726A (es)
MX (1) MX2012005332A (es)
MY (1) MY160820A (es)
NZ (1) NZ599041A (es)
SG (1) SG10201407453TA (es)
WO (1) WO2011060295A1 (es)
ZA (1) ZA201204246B (es)

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