SE444315B - Forfarande for framstellning av bensimidazolderivat - Google Patents
Forfarande for framstellning av bensimidazolderivatInfo
- Publication number
- SE444315B SE444315B SE7804057A SE7804057A SE444315B SE 444315 B SE444315 B SE 444315B SE 7804057 A SE7804057 A SE 7804057A SE 7804057 A SE7804057 A SE 7804057A SE 444315 B SE444315 B SE 444315B
- Authority
- SE
- Sweden
- Prior art keywords
- group
- carbon atoms
- formula
- denotes
- halogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU77120A LU77120A1 (es) | 1977-04-12 | 1977-04-12 | |
LU79232A LU79232A1 (de) | 1978-03-15 | 1978-03-15 | Verfahren zur herstellung von anthelmintika |
Publications (2)
Publication Number | Publication Date |
---|---|
SE7804057L SE7804057L (sv) | 1978-10-13 |
SE444315B true SE444315B (sv) | 1986-04-07 |
Family
ID=26640224
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE7804057A SE444315B (sv) | 1977-04-12 | 1978-04-11 | Forfarande for framstellning av bensimidazolderivat |
Country Status (27)
Country | Link |
---|---|
US (1) | US4197307A (es) |
JP (1) | JPS6019753B2 (es) |
AR (1) | AR230270A1 (es) |
AT (1) | AT363078B (es) |
AU (1) | AU520836B2 (es) |
BE (1) | BE865870A (es) |
CA (1) | CA1105034A (es) |
CH (1) | CH634306A5 (es) |
CS (1) | CS209450B2 (es) |
DE (1) | DE2815621A1 (es) |
DK (1) | DK155603C (es) |
FR (1) | FR2387220A1 (es) |
GB (1) | GB1599970A (es) |
IE (1) | IE46718B1 (es) |
IL (1) | IL54474A (es) |
IT (1) | IT1113128B (es) |
KE (1) | KE3345A (es) |
MX (1) | MX5951E (es) |
MY (1) | MY8500089A (es) |
NL (1) | NL187808C (es) |
NZ (1) | NZ186936A (es) |
PH (1) | PH18234A (es) |
PL (2) | PL117396B1 (es) |
SE (1) | SE444315B (es) |
SU (1) | SU1097196A3 (es) |
YU (1) | YU41309B (es) |
ZA (1) | ZA782086B (es) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3132167A1 (de) * | 1981-08-14 | 1983-03-03 | Hoechst Ag, 6000 Frankfurt | "5(6)-phenylsulfonyloxy-benzimidazolderivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung gegen leberegel" |
MA19678A1 (fr) * | 1982-01-13 | 1983-10-01 | Ciba Geigy Ag | Agents anti-helmintiques. |
GB2124904B (en) * | 1982-08-13 | 1986-01-15 | Ciba Geigy Ag | Synergistic anthelmintic compositions |
US4472419A (en) * | 1984-01-25 | 1984-09-18 | American Cyanamid Company | Method of controlling plant nematodes |
GB8426367D0 (en) * | 1984-10-18 | 1984-11-21 | Shell Int Research | Heteroaromatic ether herbicides |
US4781920A (en) * | 1984-11-13 | 1988-11-01 | American Cyanamid Company | Anthelmintic paste compositions containing resinates of d1-6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole |
DE3508665A1 (de) * | 1985-03-12 | 1986-09-18 | Hoechst Ag, 6230 Frankfurt | Heterocyclische sulfide und ihre anwendung als immunmodulatoren |
GB8519920D0 (en) * | 1985-08-08 | 1985-09-18 | Fbc Ltd | Fungicides |
JPS62246587A (ja) * | 1986-03-17 | 1987-10-27 | ピ−ピ−ジ− インダストリイズ,インコ−ポレイテツド | 除草活性を有する置換ベンゾオキサゾロン(またはベンゾチアゾロン)化合物 |
DE3719783A1 (de) * | 1987-06-13 | 1988-12-22 | Hoechst Ag | Verfahren zur herstellung von 5-phenylsulfinyl-1h-2-(methoxycarbonylamino)- benzimidazol |
NZ335166A (en) | 1999-04-14 | 2001-11-30 | Ashmont Holdings Ltd | Anthelmintic composition containing triclabendazole in at least one solvent |
AU2003236405B2 (en) * | 1999-04-14 | 2007-10-25 | Merial Ltd | Anthelmintic Composition |
US5538989A (en) * | 1993-11-10 | 1996-07-23 | Hoechst-Roussel Agri-Vet Company | Fenbendazole formulations |
US20060205681A1 (en) * | 2002-06-21 | 2006-09-14 | Maryam Moaddeb | Homogenous paste formulations |
US7001889B2 (en) * | 2002-06-21 | 2006-02-21 | Merial Limited | Anthelmintic oral homogeneous veterinary pastes |
KR20050108373A (ko) | 2003-03-03 | 2005-11-16 | 마이코솔 인코포레이티드 | 피리디늄 염 화합물 및 이용 방법 |
WO2005074914A1 (en) * | 2004-02-03 | 2005-08-18 | Wyeth | Anthelmintic composition |
TWI387592B (zh) * | 2005-08-30 | 2013-03-01 | Novartis Ag | 經取代之苯并咪唑及其作為與腫瘤形成相關激酶之抑制劑之方法 |
US20080027011A1 (en) * | 2005-12-20 | 2008-01-31 | Hassan Nached | Homogeneous paste and gel formulations |
WO2010042395A1 (en) * | 2008-10-08 | 2010-04-15 | Wyeth Llc | Benzimidazole anthelmintic compositions |
CN101555231B (zh) * | 2009-05-04 | 2011-03-23 | 扬州天和药业有限公司 | 一种制备三氯苯达唑的方法 |
WO2012070068A2 (en) * | 2010-11-24 | 2012-05-31 | Sequent Scientific Limited | Process for preparation of triclabendazole |
PT2895465T (pt) * | 2012-04-20 | 2019-01-16 | Boehringer Ingelheim Animal Health Usa Inc | Composições parasiticidas compreendendo derivados de benzimidazoles, os seus métodos e as suas utilizações |
CN103319416B (zh) * | 2013-06-24 | 2015-02-25 | 常州佳灵药业有限公司 | 新型兽药三氯苯达唑亚砜及其制备方法 |
EP3235815A1 (de) | 2016-04-19 | 2017-10-25 | Philipps-Universität Marburg | Wirkstoffe gegen parasitäre helminthen |
RU2640482C2 (ru) * | 2016-04-22 | 2018-01-09 | ФАНО России Федеральное государственное бюджетное научное учреждение Всероссийский научно-исследовательский институт фундаментальной и прикладной паразитологии животных и растений им. К.И. Скрябина (ФГБНУ "ВНИИП им. К.И. Скрябина") | Супрамолекулярный комплекс триклабендазола для лечения животных при фасциолёзе |
US20220202835A1 (en) | 2019-03-01 | 2022-06-30 | Boehringer Ingelheim Animal Health USA Inc. | Injectable clorsulon compositions, methods and uses thereof |
BR112023017612A2 (pt) * | 2021-03-03 | 2023-12-05 | Terns Pharmaceuticals Inc | Compostos agonistas do receptor beta do hormônio da tireoide |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2666764A (en) * | 1951-07-14 | 1954-01-19 | Ciba Pharm Prod Inc | Process of splitting aralkylheterocyclic thioethers with aluminum bromide |
FR1476558A (fr) * | 1965-07-26 | 1967-04-14 | Chimetron Sarl | Thiazolylthiobenzimidazoles et thiazolylsulfinylbenzimidazoles |
US3506767A (en) * | 1965-08-06 | 1970-04-14 | Geigy Chem Corp | Benzimidazole compositions and methods of use |
CH443777A (de) * | 1965-08-06 | 1968-02-15 | Agripat Sa | Verfahren zum Schützen textiler Keratinfasern vor Insektenfrass und Mittel zur Durchführung dieses Verfahrens |
FR1509192A (fr) * | 1966-12-01 | 1968-01-12 | Benzylthio-2 benzimidazoles | |
US3480643A (en) * | 1967-05-09 | 1969-11-25 | American Cyanamid Co | Alkylsulfonylbenzimidazoles |
NL7013343A (es) * | 1969-09-26 | 1971-03-30 | ||
BE754874A (fr) * | 1969-10-30 | 1971-01-18 | Buckman Labor Inc | Composes s-chloromethyliques de 2-mercapto-benzothiazole, de 2-mercaptobenzoxazole et de 2-mercaptobenzimidazole |
DE2041324A1 (de) * | 1970-08-20 | 1972-02-24 | Agfa Gevaert Ag | Neue Benzimidazolderivate,sowie ein Verfahren zu ihrer Herstellung |
US3933841A (en) * | 1971-05-24 | 1976-01-20 | Ciba-Geigy Corporation | 2-Phenoxy, -phenylthio-, and -phenyl-amino-benzoxazoles having an isothiocyano substituent |
US3840550A (en) * | 1971-05-24 | 1974-10-08 | Ciba Geigy Corp | Certain 6-isothiocyanobenzothiazoles |
BE792402A (fr) * | 1971-12-07 | 1973-06-07 | Ciba Geigy | Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent |
-
1978
- 1978-04-10 CH CH382678A patent/CH634306A5/de not_active IP Right Cessation
- 1978-04-10 US US05/894,973 patent/US4197307A/en not_active Expired - Lifetime
- 1978-04-10 IL IL54474A patent/IL54474A/xx unknown
- 1978-04-11 MX MX787013U patent/MX5951E/es unknown
- 1978-04-11 IT IT22189/78A patent/IT1113128B/it active
- 1978-04-11 AT AT0253478A patent/AT363078B/de active
- 1978-04-11 BE BE186705A patent/BE865870A/xx not_active IP Right Cessation
- 1978-04-11 SU SU782601448A patent/SU1097196A3/ru active
- 1978-04-11 NZ NZ186936A patent/NZ186936A/xx unknown
- 1978-04-11 CS CS782366A patent/CS209450B2/cs unknown
- 1978-04-11 DK DK159478A patent/DK155603C/da not_active IP Right Cessation
- 1978-04-11 GB GB14183/78A patent/GB1599970A/en not_active Expired
- 1978-04-11 IE IE704/78A patent/IE46718B1/en not_active IP Right Cessation
- 1978-04-11 ZA ZA00782086A patent/ZA782086B/xx unknown
- 1978-04-11 YU YU857/78A patent/YU41309B/xx unknown
- 1978-04-11 SE SE7804057A patent/SE444315B/sv not_active IP Right Cessation
- 1978-04-11 DE DE19782815621 patent/DE2815621A1/de active Granted
- 1978-04-12 AU AU35022/78A patent/AU520836B2/en not_active Expired
- 1978-04-12 FR FR7810731A patent/FR2387220A1/fr active Granted
- 1978-04-12 JP JP53043058A patent/JPS6019753B2/ja not_active Expired
- 1978-04-12 CA CA300,973A patent/CA1105034A/en not_active Expired
- 1978-04-12 NL NLAANVRAGE7803886,A patent/NL187808C/xx not_active IP Right Cessation
- 1978-04-12 PL PL1978221071A patent/PL117396B1/pl unknown
- 1978-04-12 PL PL1978206019A patent/PL115361B1/pl unknown
- 1978-04-12 PH PH20998A patent/PH18234A/en unknown
-
1979
- 1979-06-28 AR AR277106A patent/AR230270A1/es active
-
1983
- 1983-11-16 KE KE3345A patent/KE3345A/xx unknown
-
1985
- 1985-12-30 MY MY89/85A patent/MY8500089A/xx unknown
Also Published As
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