MX5951E - Procedimiento para la preparacion de derivados de benzoimidazol - Google Patents
Procedimiento para la preparacion de derivados de benzoimidazolInfo
- Publication number
- MX5951E MX5951E MX787013U MX701378U MX5951E MX 5951 E MX5951 E MX 5951E MX 787013 U MX787013 U MX 787013U MX 701378 U MX701378 U MX 701378U MX 5951 E MX5951 E MX 5951E
- Authority
- MX
- Mexico
- Prior art keywords
- procedure
- preparation
- benzoimidazole derivatives
- benzoimidazole
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU77120A LU77120A1 (es) | 1977-04-12 | 1977-04-12 | |
LU79232A LU79232A1 (de) | 1978-03-15 | 1978-03-15 | Verfahren zur herstellung von anthelmintika |
Publications (1)
Publication Number | Publication Date |
---|---|
MX5951E true MX5951E (es) | 1984-09-06 |
Family
ID=26640224
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX787013U MX5951E (es) | 1977-04-12 | 1978-04-11 | Procedimiento para la preparacion de derivados de benzoimidazol |
Country Status (27)
Country | Link |
---|---|
US (1) | US4197307A (es) |
JP (1) | JPS6019753B2 (es) |
AR (1) | AR230270A1 (es) |
AT (1) | AT363078B (es) |
AU (1) | AU520836B2 (es) |
BE (1) | BE865870A (es) |
CA (1) | CA1105034A (es) |
CH (1) | CH634306A5 (es) |
CS (1) | CS209450B2 (es) |
DE (1) | DE2815621A1 (es) |
DK (1) | DK155603C (es) |
FR (1) | FR2387220A1 (es) |
GB (1) | GB1599970A (es) |
IE (1) | IE46718B1 (es) |
IL (1) | IL54474A (es) |
IT (1) | IT1113128B (es) |
KE (1) | KE3345A (es) |
MX (1) | MX5951E (es) |
MY (1) | MY8500089A (es) |
NL (1) | NL187808C (es) |
NZ (1) | NZ186936A (es) |
PH (1) | PH18234A (es) |
PL (2) | PL117396B1 (es) |
SE (1) | SE444315B (es) |
SU (1) | SU1097196A3 (es) |
YU (1) | YU41309B (es) |
ZA (1) | ZA782086B (es) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3132167A1 (de) * | 1981-08-14 | 1983-03-03 | Hoechst Ag, 6000 Frankfurt | "5(6)-phenylsulfonyloxy-benzimidazolderivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung gegen leberegel" |
MA19678A1 (fr) * | 1982-01-13 | 1983-10-01 | Ciba Geigy Ag | Agents anti-helmintiques. |
GB2124904B (en) * | 1982-08-13 | 1986-01-15 | Ciba Geigy Ag | Synergistic anthelmintic compositions |
US4472419A (en) * | 1984-01-25 | 1984-09-18 | American Cyanamid Company | Method of controlling plant nematodes |
GB8426367D0 (en) * | 1984-10-18 | 1984-11-21 | Shell Int Research | Heteroaromatic ether herbicides |
US4781920A (en) * | 1984-11-13 | 1988-11-01 | American Cyanamid Company | Anthelmintic paste compositions containing resinates of d1-6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole |
DE3508665A1 (de) * | 1985-03-12 | 1986-09-18 | Hoechst Ag, 6230 Frankfurt | Heterocyclische sulfide und ihre anwendung als immunmodulatoren |
GB8519920D0 (en) * | 1985-08-08 | 1985-09-18 | Fbc Ltd | Fungicides |
JPS62246587A (ja) * | 1986-03-17 | 1987-10-27 | ピ−ピ−ジ− インダストリイズ,インコ−ポレイテツド | 除草活性を有する置換ベンゾオキサゾロン(またはベンゾチアゾロン)化合物 |
DE3719783A1 (de) * | 1987-06-13 | 1988-12-22 | Hoechst Ag | Verfahren zur herstellung von 5-phenylsulfinyl-1h-2-(methoxycarbonylamino)- benzimidazol |
AU2003236405B2 (en) * | 1999-04-14 | 2007-10-25 | Merial Ltd | Anthelmintic Composition |
NZ335166A (en) | 1999-04-14 | 2001-11-30 | Ashmont Holdings Ltd | Anthelmintic composition containing triclabendazole in at least one solvent |
US5538989A (en) * | 1993-11-10 | 1996-07-23 | Hoechst-Roussel Agri-Vet Company | Fenbendazole formulations |
US7001889B2 (en) * | 2002-06-21 | 2006-02-21 | Merial Limited | Anthelmintic oral homogeneous veterinary pastes |
US20060205681A1 (en) * | 2002-06-21 | 2006-09-14 | Maryam Moaddeb | Homogenous paste formulations |
JP4742028B2 (ja) * | 2003-03-03 | 2011-08-10 | マイコソル,インコーポレイテッド | ピリジニウム塩、化合物および使用法 |
ES2342668T3 (es) * | 2004-02-03 | 2010-07-12 | Wyeth Llc | Composicion antihelmintica. |
TW200804345A (en) * | 2005-08-30 | 2008-01-16 | Novartis Ag | Substituted benzimidazoles and methods of preparation |
US20080027011A1 (en) * | 2005-12-20 | 2008-01-31 | Hassan Nached | Homogeneous paste and gel formulations |
JP5547738B2 (ja) * | 2008-10-08 | 2014-07-16 | ゾエティス・ダブリュー・エルエルシー | ベンゾイミダゾール駆虫組成物 |
CN101555231B (zh) * | 2009-05-04 | 2011-03-23 | 扬州天和药业有限公司 | 一种制备三氯苯达唑的方法 |
WO2012070068A2 (en) * | 2010-11-24 | 2012-05-31 | Sequent Scientific Limited | Process for preparation of triclabendazole |
EP2895465B1 (en) * | 2012-04-20 | 2018-10-03 | Merial, Inc. | Parasiticidal compositions comprising benzimidazole derivatives, methods and uses thereof |
CN103319416B (zh) * | 2013-06-24 | 2015-02-25 | 常州佳灵药业有限公司 | 新型兽药三氯苯达唑亚砜及其制备方法 |
EP3235815A1 (de) | 2016-04-19 | 2017-10-25 | Philipps-Universität Marburg | Wirkstoffe gegen parasitäre helminthen |
RU2640482C2 (ru) * | 2016-04-22 | 2018-01-09 | ФАНО России Федеральное государственное бюджетное научное учреждение Всероссийский научно-исследовательский институт фундаментальной и прикладной паразитологии животных и растений им. К.И. Скрябина (ФГБНУ "ВНИИП им. К.И. Скрябина") | Супрамолекулярный комплекс триклабендазола для лечения животных при фасциолёзе |
CA3129329A1 (en) | 2019-03-01 | 2020-09-10 | Boehringer Ingelheim Animal Health USA Inc. | Injectable clorsulon compositions, methods and uses thereof |
CA3212130A1 (en) * | 2021-03-03 | 2022-09-09 | Terns Pharmaceuticals, Inc. | Thyroid hormone receptor beta agonist compounds |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2666764A (en) * | 1951-07-14 | 1954-01-19 | Ciba Pharm Prod Inc | Process of splitting aralkylheterocyclic thioethers with aluminum bromide |
FR1476558A (fr) * | 1965-07-26 | 1967-04-14 | Chimetron Sarl | Thiazolylthiobenzimidazoles et thiazolylsulfinylbenzimidazoles |
CH443777A (de) * | 1965-08-06 | 1968-02-15 | Agripat Sa | Verfahren zum Schützen textiler Keratinfasern vor Insektenfrass und Mittel zur Durchführung dieses Verfahrens |
US3506767A (en) * | 1965-08-06 | 1970-04-14 | Geigy Chem Corp | Benzimidazole compositions and methods of use |
FR1509192A (fr) * | 1966-12-01 | 1968-01-12 | Benzylthio-2 benzimidazoles | |
US3480643A (en) * | 1967-05-09 | 1969-11-25 | American Cyanamid Co | Alkylsulfonylbenzimidazoles |
NL7013343A (es) * | 1969-09-26 | 1971-03-30 | ||
BE754874A (fr) * | 1969-10-30 | 1971-01-18 | Buckman Labor Inc | Composes s-chloromethyliques de 2-mercapto-benzothiazole, de 2-mercaptobenzoxazole et de 2-mercaptobenzimidazole |
DE2041324A1 (de) * | 1970-08-20 | 1972-02-24 | Agfa Gevaert Ag | Neue Benzimidazolderivate,sowie ein Verfahren zu ihrer Herstellung |
US3840550A (en) * | 1971-05-24 | 1974-10-08 | Ciba Geigy Corp | Certain 6-isothiocyanobenzothiazoles |
US3933841A (en) * | 1971-05-24 | 1976-01-20 | Ciba-Geigy Corporation | 2-Phenoxy, -phenylthio-, and -phenyl-amino-benzoxazoles having an isothiocyano substituent |
BE792402A (fr) * | 1971-12-07 | 1973-06-07 | Ciba Geigy | Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent |
-
1978
- 1978-04-10 CH CH382678A patent/CH634306A5/de not_active IP Right Cessation
- 1978-04-10 IL IL54474A patent/IL54474A/xx unknown
- 1978-04-10 US US05/894,973 patent/US4197307A/en not_active Expired - Lifetime
- 1978-04-11 BE BE186705A patent/BE865870A/xx not_active IP Right Cessation
- 1978-04-11 GB GB14183/78A patent/GB1599970A/en not_active Expired
- 1978-04-11 DK DK159478A patent/DK155603C/da not_active IP Right Cessation
- 1978-04-11 AT AT0253478A patent/AT363078B/de active
- 1978-04-11 SE SE7804057A patent/SE444315B/sv not_active IP Right Cessation
- 1978-04-11 ZA ZA00782086A patent/ZA782086B/xx unknown
- 1978-04-11 IE IE704/78A patent/IE46718B1/en not_active IP Right Cessation
- 1978-04-11 CS CS782366A patent/CS209450B2/cs unknown
- 1978-04-11 SU SU782601448A patent/SU1097196A3/ru active
- 1978-04-11 YU YU857/78A patent/YU41309B/xx unknown
- 1978-04-11 NZ NZ186936A patent/NZ186936A/xx unknown
- 1978-04-11 IT IT22189/78A patent/IT1113128B/it active
- 1978-04-11 MX MX787013U patent/MX5951E/es unknown
- 1978-04-11 DE DE19782815621 patent/DE2815621A1/de active Granted
- 1978-04-12 PH PH20998A patent/PH18234A/en unknown
- 1978-04-12 JP JP53043058A patent/JPS6019753B2/ja not_active Expired
- 1978-04-12 NL NLAANVRAGE7803886,A patent/NL187808C/xx not_active IP Right Cessation
- 1978-04-12 AU AU35022/78A patent/AU520836B2/en not_active Expired
- 1978-04-12 CA CA300,973A patent/CA1105034A/en not_active Expired
- 1978-04-12 FR FR7810731A patent/FR2387220A1/fr active Granted
- 1978-04-12 PL PL1978221071A patent/PL117396B1/pl unknown
- 1978-04-12 PL PL1978206019A patent/PL115361B1/pl unknown
-
1979
- 1979-06-28 AR AR277106A patent/AR230270A1/es active
-
1983
- 1983-11-16 KE KE3345A patent/KE3345A/xx unknown
-
1985
- 1985-12-30 MY MY89/85A patent/MY8500089A/xx unknown
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