SE436749B - Forfarande for framstellning av 2,5-dihydro-1,2-tiazino/5,6-b/indol-3-karboxamid-1,1-dioxider - Google Patents
Forfarande for framstellning av 2,5-dihydro-1,2-tiazino/5,6-b/indol-3-karboxamid-1,1-dioxiderInfo
- Publication number
- SE436749B SE436749B SE7714833A SE7714833A SE436749B SE 436749 B SE436749 B SE 436749B SE 7714833 A SE7714833 A SE 7714833A SE 7714833 A SE7714833 A SE 7714833A SE 436749 B SE436749 B SE 436749B
- Authority
- SE
- Sweden
- Prior art keywords
- dihydro
- indole
- thiazino
- dioxide
- hydroxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Hematology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19772704485 DE2704485A1 (de) | 1977-02-03 | 1977-02-03 | Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE7714833L SE7714833L (sv) | 1978-08-04 |
| SE436749B true SE436749B (sv) | 1985-01-21 |
Family
ID=6000267
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7714833A SE436749B (sv) | 1977-02-03 | 1977-12-28 | Forfarande for framstellning av 2,5-dihydro-1,2-tiazino/5,6-b/indol-3-karboxamid-1,1-dioxider |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US4137313A (ru) |
| JP (1) | JPS5398998A (ru) |
| AT (3) | AT355585B (ru) |
| AU (1) | AU516178B2 (ru) |
| BE (1) | BE863588A (ru) |
| BG (1) | BG36499A3 (ru) |
| CA (1) | CA1088064A (ru) |
| CH (1) | CH639389A5 (ru) |
| CS (1) | CS194195B2 (ru) |
| DD (1) | DD134767A5 (ru) |
| DE (1) | DE2704485A1 (ru) |
| DK (1) | DK150517C (ru) |
| ES (5) | ES466555A1 (ru) |
| FI (1) | FI62097C (ru) |
| FR (1) | FR2379542A1 (ru) |
| GB (1) | GB1569238A (ru) |
| GR (1) | GR64418B (ru) |
| HK (1) | HK71383A (ru) |
| HU (1) | HU175550B (ru) |
| IE (1) | IE46185B1 (ru) |
| IL (1) | IL53948A (ru) |
| IT (1) | IT1105151B (ru) |
| LU (1) | LU78974A1 (ru) |
| MY (1) | MY8400283A (ru) |
| NL (1) | NL7801183A (ru) |
| NO (1) | NO148490C (ru) |
| NZ (1) | NZ186374A (ru) |
| PH (1) | PH13882A (ru) |
| PL (1) | PL109705B1 (ru) |
| PT (1) | PT67607B (ru) |
| SE (1) | SE436749B (ru) |
| SG (1) | SG48083G (ru) |
| SU (1) | SU654173A3 (ru) |
| YU (1) | YU24478A (ru) |
| ZA (1) | ZA78630B (ru) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2838377A1 (de) * | 1978-09-02 | 1980-03-20 | Thomae Gmbh Dr K | Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung |
| AU5811280A (en) | 1979-06-13 | 1980-12-18 | F. Hoffmann-La Roche Ag | Thiazine derivatives |
| GR80576B (en) * | 1983-10-17 | 1984-11-29 | Fujisawa Pharmaceutical Co | Thiazine derivatives, process for preparation thereof and pharmaceutical composition comprising the same |
| US4683306A (en) * | 1984-07-13 | 1987-07-28 | Yuhan Corporation Co., Ltd. | Process for the preparation of 3,4-dihydro-2-substituted-2H-1,2-thiazine-carboxylic acid 1,1-dioxide derivatives |
| US6407124B1 (en) | 1998-06-18 | 2002-06-18 | Bristol-Myers Squibb Company | Carbon substituted aminothiazole inhibitors of cyclin dependent kinases |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH588693A5 (ru) * | 1973-12-10 | 1977-06-15 | Image Analysing Computers Ltd | |
| IL47877A (en) * | 1974-08-26 | 1978-10-31 | Sparamedica Ag | Thienothiazine carboxamide derivatives,their manufacture and pharmaceutical compositions containing them |
| AT345847B (de) * | 1974-11-08 | 1978-10-10 | Thomae Gmbh Dr K | Verfahren zur herstellung neuer 4-hydroxy-2h- naphtho- (2,1-e)-1,2-thiazin-3-carboxamid-1,1-dioxid und deren salze |
-
1977
- 1977-02-03 DE DE19772704485 patent/DE2704485A1/de not_active Withdrawn
- 1977-12-28 SE SE7714833A patent/SE436749B/sv not_active IP Right Cessation
-
1978
- 1978-01-09 AT AT11178A patent/AT355585B/de active
- 1978-01-17 BG BG038411A patent/BG36499A3/xx unknown
- 1978-01-27 US US05/872,889 patent/US4137313A/en not_active Expired - Lifetime
- 1978-01-27 IT IT47828/78A patent/IT1105151B/it active
- 1978-01-30 SU SU782571747A patent/SU654173A3/ru active
- 1978-01-31 CS CS78650A patent/CS194195B2/cs unknown
- 1978-02-01 DD DD78203510A patent/DD134767A5/xx unknown
- 1978-02-01 PH PH20738A patent/PH13882A/en unknown
- 1978-02-01 IL IL53948A patent/IL53948A/xx unknown
- 1978-02-01 FI FI780324A patent/FI62097C/fi not_active IP Right Cessation
- 1978-02-01 GR GR55322A patent/GR64418B/el unknown
- 1978-02-01 LU LU78974A patent/LU78974A1/de unknown
- 1978-02-01 HU HU78TO1069A patent/HU175550B/hu unknown
- 1978-02-02 NL NL7801183A patent/NL7801183A/xx not_active Application Discontinuation
- 1978-02-02 ES ES466555A patent/ES466555A1/es not_active Expired
- 1978-02-02 CA CA296,063A patent/CA1088064A/en not_active Expired
- 1978-02-02 YU YU00244/78A patent/YU24478A/xx unknown
- 1978-02-02 BE BE184854A patent/BE863588A/xx not_active IP Right Cessation
- 1978-02-02 CH CH114778A patent/CH639389A5/de not_active IP Right Cessation
- 1978-02-02 AU AU32931/78A patent/AU516178B2/en not_active Expired
- 1978-02-02 PL PL1978204401A patent/PL109705B1/pl unknown
- 1978-02-02 PT PT67607A patent/PT67607B/pt unknown
- 1978-02-02 ZA ZA00780630A patent/ZA78630B/xx unknown
- 1978-02-02 NO NO780370A patent/NO148490C/no unknown
- 1978-02-02 NZ NZ186374A patent/NZ186374A/xx unknown
- 1978-02-02 DK DK048478A patent/DK150517C/da not_active IP Right Cessation
- 1978-02-02 GB GB4304/78A patent/GB1569238A/en not_active Expired
- 1978-02-02 JP JP1104478A patent/JPS5398998A/ja active Granted
- 1978-02-03 IE IE246/78A patent/IE46185B1/en unknown
- 1978-02-03 FR FR7803158A patent/FR2379542A1/fr active Granted
- 1978-04-25 ES ES469112A patent/ES469112A1/es not_active Expired
- 1978-04-25 ES ES469113A patent/ES469113A1/es not_active Expired
- 1978-04-25 ES ES469111A patent/ES469111A1/es not_active Expired
- 1978-04-25 ES ES469110A patent/ES469110A1/es not_active Expired
-
1979
- 1979-04-11 AT AT269679A patent/AT355591B/de not_active IP Right Cessation
- 1979-04-11 AT AT269579A patent/AT355590B/de not_active IP Right Cessation
-
1983
- 1983-08-10 SG SG48083A patent/SG48083G/en unknown
- 1983-12-20 HK HK713/83A patent/HK71383A/xx unknown
-
1984
- 1984-12-30 MY MY283/84A patent/MY8400283A/xx unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NUG | Patent has lapsed |
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