ZA78630B - 2,5-dihydro-1,2-thiazino(5,6-b)indol-3-carboxamides-1,1-dioxides,processes for their preparation and pharmaceutical compositions thereof - Google Patents

2,5-dihydro-1,2-thiazino(5,6-b)indol-3-carboxamides-1,1-dioxides,processes for their preparation and pharmaceutical compositions thereof

Info

Publication number
ZA78630B
ZA78630B ZA00780630A ZA78630A ZA78630B ZA 78630 B ZA78630 B ZA 78630B ZA 00780630 A ZA00780630 A ZA 00780630A ZA 78630 A ZA78630 A ZA 78630A ZA 78630 B ZA78630 B ZA 78630B
Authority
ZA
South Africa
Prior art keywords
thiazino
dioxides
carboxamides
indol
dihydro
Prior art date
Application number
ZA00780630A
Other languages
English (en)
Inventor
W Haarmann
G Engelhardt
G Trummlitz
W Engel
E Seeger
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of ZA78630B publication Critical patent/ZA78630B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ZA00780630A 1977-02-03 1978-02-02 2,5-dihydro-1,2-thiazino(5,6-b)indol-3-carboxamides-1,1-dioxides,processes for their preparation and pharmaceutical compositions thereof ZA78630B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772704485 DE2704485A1 (de) 1977-02-03 1977-02-03 Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
ZA78630B true ZA78630B (en) 1979-10-31

Family

ID=6000267

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00780630A ZA78630B (en) 1977-02-03 1978-02-02 2,5-dihydro-1,2-thiazino(5,6-b)indol-3-carboxamides-1,1-dioxides,processes for their preparation and pharmaceutical compositions thereof

Country Status (35)

Country Link
US (1) US4137313A (ru)
JP (1) JPS5398998A (ru)
AT (3) AT355585B (ru)
AU (1) AU516178B2 (ru)
BE (1) BE863588A (ru)
BG (1) BG36499A3 (ru)
CA (1) CA1088064A (ru)
CH (1) CH639389A5 (ru)
CS (1) CS194195B2 (ru)
DD (1) DD134767A5 (ru)
DE (1) DE2704485A1 (ru)
DK (1) DK150517C (ru)
ES (5) ES466555A1 (ru)
FI (1) FI62097C (ru)
FR (1) FR2379542A1 (ru)
GB (1) GB1569238A (ru)
GR (1) GR64418B (ru)
HK (1) HK71383A (ru)
HU (1) HU175550B (ru)
IE (1) IE46185B1 (ru)
IL (1) IL53948A (ru)
IT (1) IT1105151B (ru)
LU (1) LU78974A1 (ru)
MY (1) MY8400283A (ru)
NL (1) NL7801183A (ru)
NO (1) NO148490C (ru)
NZ (1) NZ186374A (ru)
PH (1) PH13882A (ru)
PL (1) PL109705B1 (ru)
PT (1) PT67607B (ru)
SE (1) SE436749B (ru)
SG (1) SG48083G (ru)
SU (1) SU654173A3 (ru)
YU (1) YU24478A (ru)
ZA (1) ZA78630B (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2838377A1 (de) * 1978-09-02 1980-03-20 Thomae Gmbh Dr K Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung
AU5811280A (en) 1979-06-13 1980-12-18 F. Hoffmann-La Roche Ag Thiazine derivatives
GR80576B (en) * 1983-10-17 1984-11-29 Fujisawa Pharmaceutical Co Thiazine derivatives, process for preparation thereof and pharmaceutical composition comprising the same
US4683306A (en) * 1984-07-13 1987-07-28 Yuhan Corporation Co., Ltd. Process for the preparation of 3,4-dihydro-2-substituted-2H-1,2-thiazine-carboxylic acid 1,1-dioxide derivatives
US6407124B1 (en) 1998-06-18 2002-06-18 Bristol-Myers Squibb Company Carbon substituted aminothiazole inhibitors of cyclin dependent kinases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH588693A5 (ru) * 1973-12-10 1977-06-15 Image Analysing Computers Ltd
IL47877A (en) * 1974-08-26 1978-10-31 Sparamedica Ag Thienothiazine carboxamide derivatives,their manufacture and pharmaceutical compositions containing them
AT345847B (de) * 1974-11-08 1978-10-10 Thomae Gmbh Dr K Verfahren zur herstellung neuer 4-hydroxy-2h- naphtho- (2,1-e)-1,2-thiazin-3-carboxamid-1,1-dioxid und deren salze

Also Published As

Publication number Publication date
ES469111A1 (es) 1978-11-16
PL204401A1 (pl) 1979-04-09
DD134767A5 (de) 1979-03-21
NO148490B (no) 1983-07-11
AU516178B2 (en) 1981-05-21
SE436749B (sv) 1985-01-21
JPS5398998A (en) 1978-08-29
DK150517B (da) 1987-03-16
IE780246L (en) 1978-08-03
FR2379542A1 (fr) 1978-09-01
MY8400283A (en) 1984-12-31
HK71383A (en) 1983-12-30
US4137313A (en) 1979-01-30
DE2704485A1 (de) 1978-08-10
IL53948A (en) 1980-10-26
ES469112A1 (es) 1978-11-16
NO780370L (no) 1978-08-04
PH13882A (en) 1980-10-27
SE7714833L (sv) 1978-08-04
AU3293178A (en) 1979-08-09
PT67607B (de) 1980-03-03
PT67607A (de) 1978-03-01
ES466555A1 (es) 1978-10-01
YU24478A (en) 1982-10-31
GB1569238A (en) 1980-06-11
CS194195B2 (en) 1979-11-30
NL7801183A (nl) 1978-08-07
GR64418B (en) 1980-03-21
AT355590B (de) 1980-03-10
CH639389A5 (de) 1983-11-15
JPS6111235B2 (ru) 1986-04-01
HU175550B (hu) 1980-08-28
IT7847828A0 (it) 1978-01-27
NO148490C (no) 1983-10-19
ATA269679A (de) 1979-08-15
AT355585B (de) 1980-03-10
IL53948A0 (en) 1978-04-30
SU654173A3 (ru) 1979-03-25
FI62097C (fi) 1982-11-10
NZ186374A (en) 1980-03-05
SG48083G (en) 1984-07-27
BG36499A3 (en) 1984-11-15
LU78974A1 (de) 1979-05-25
IT1105151B (it) 1985-10-28
DK48478A (da) 1978-08-04
ATA269579A (de) 1979-08-15
BE863588A (fr) 1978-08-02
FI780324A (fi) 1978-08-04
PL109705B1 (en) 1980-06-30
FI62097B (fi) 1982-07-30
DK150517C (da) 1987-10-19
ES469110A1 (es) 1978-11-16
CA1088064A (en) 1980-10-21
AT355591B (de) 1980-03-10
ES469113A1 (es) 1978-11-16
FR2379542B1 (ru) 1982-12-03
IE46185B1 (en) 1983-03-23
ATA11178A (de) 1979-08-15

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