ES469111A1 - Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos. - Google Patents

Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.

Info

Publication number
ES469111A1
ES469111A1 ES469111A ES469111A ES469111A1 ES 469111 A1 ES469111 A1 ES 469111A1 ES 469111 A ES469111 A ES 469111A ES 469111 A ES469111 A ES 469111A ES 469111 A1 ES469111 A1 ES 469111A1
Authority
ES
Spain
Prior art keywords
methyl
ethyl
substituent attached
salts
pyridyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES469111A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Publication of ES469111A1 publication Critical patent/ES469111A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES469111A 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos. Expired ES469111A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772704485 DE2704485A1 (de) 1977-02-03 1977-02-03 Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
ES469111A1 true ES469111A1 (es) 1978-11-16

Family

ID=6000267

Family Applications (5)

Application Number Title Priority Date Filing Date
ES466555A Expired ES466555A1 (es) 1977-02-03 1978-02-02 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.
ES469112A Expired ES469112A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.
ES469113A Expired ES469113A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.
ES469111A Expired ES469111A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.
ES469110A Expired ES469110A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.

Family Applications Before (3)

Application Number Title Priority Date Filing Date
ES466555A Expired ES466555A1 (es) 1977-02-03 1978-02-02 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.
ES469112A Expired ES469112A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.
ES469113A Expired ES469113A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES469110A Expired ES469110A1 (es) 1977-02-03 1978-04-25 Procedimiento para la preparacion de nuevos 2,5-dihidro-1,2-tiazino (5,6-b)indol-3-carboxamido-1,1-dioxidos.

Country Status (35)

Country Link
US (1) US4137313A (es)
JP (1) JPS5398998A (es)
AT (3) AT355585B (es)
AU (1) AU516178B2 (es)
BE (1) BE863588A (es)
BG (1) BG36499A3 (es)
CA (1) CA1088064A (es)
CH (1) CH639389A5 (es)
CS (1) CS194195B2 (es)
DD (1) DD134767A5 (es)
DE (1) DE2704485A1 (es)
DK (1) DK150517C (es)
ES (5) ES466555A1 (es)
FI (1) FI62097C (es)
FR (1) FR2379542A1 (es)
GB (1) GB1569238A (es)
GR (1) GR64418B (es)
HK (1) HK71383A (es)
HU (1) HU175550B (es)
IE (1) IE46185B1 (es)
IL (1) IL53948A (es)
IT (1) IT1105151B (es)
LU (1) LU78974A1 (es)
MY (1) MY8400283A (es)
NL (1) NL7801183A (es)
NO (1) NO148490C (es)
NZ (1) NZ186374A (es)
PH (1) PH13882A (es)
PL (1) PL109705B1 (es)
PT (1) PT67607B (es)
SE (1) SE436749B (es)
SG (1) SG48083G (es)
SU (1) SU654173A3 (es)
YU (1) YU24478A (es)
ZA (1) ZA78630B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2838377A1 (de) * 1978-09-02 1980-03-20 Thomae Gmbh Dr K Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung
AU5811280A (en) 1979-06-13 1980-12-18 F. Hoffmann-La Roche Ag Thiazine derivatives
GR80576B (en) * 1983-10-17 1984-11-29 Fujisawa Pharmaceutical Co Thiazine derivatives, process for preparation thereof and pharmaceutical composition comprising the same
US4683306A (en) * 1984-07-13 1987-07-28 Yuhan Corporation Co., Ltd. Process for the preparation of 3,4-dihydro-2-substituted-2H-1,2-thiazine-carboxylic acid 1,1-dioxide derivatives
US6407124B1 (en) 1998-06-18 2002-06-18 Bristol-Myers Squibb Company Carbon substituted aminothiazole inhibitors of cyclin dependent kinases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH588693A5 (es) * 1973-12-10 1977-06-15 Image Analysing Computers Ltd
IL47877A (en) * 1974-08-26 1978-10-31 Sparamedica Ag Thienothiazine carboxamide derivatives,their manufacture and pharmaceutical compositions containing them
AT345847B (de) * 1974-11-08 1978-10-10 Thomae Gmbh Dr K Verfahren zur herstellung neuer 4-hydroxy-2h- naphtho- (2,1-e)-1,2-thiazin-3-carboxamid-1,1-dioxid und deren salze

Also Published As

Publication number Publication date
PL204401A1 (pl) 1979-04-09
DD134767A5 (de) 1979-03-21
NO148490B (no) 1983-07-11
AU516178B2 (en) 1981-05-21
SE436749B (sv) 1985-01-21
JPS5398998A (en) 1978-08-29
DK150517B (da) 1987-03-16
IE780246L (en) 1978-08-03
FR2379542A1 (fr) 1978-09-01
MY8400283A (en) 1984-12-31
HK71383A (en) 1983-12-30
US4137313A (en) 1979-01-30
DE2704485A1 (de) 1978-08-10
IL53948A (en) 1980-10-26
ES469112A1 (es) 1978-11-16
NO780370L (no) 1978-08-04
PH13882A (en) 1980-10-27
SE7714833L (sv) 1978-08-04
AU3293178A (en) 1979-08-09
PT67607B (de) 1980-03-03
PT67607A (de) 1978-03-01
ES466555A1 (es) 1978-10-01
YU24478A (en) 1982-10-31
GB1569238A (en) 1980-06-11
CS194195B2 (en) 1979-11-30
NL7801183A (nl) 1978-08-07
GR64418B (en) 1980-03-21
AT355590B (de) 1980-03-10
CH639389A5 (de) 1983-11-15
JPS6111235B2 (es) 1986-04-01
HU175550B (hu) 1980-08-28
IT7847828A0 (it) 1978-01-27
NO148490C (no) 1983-10-19
ATA269679A (de) 1979-08-15
AT355585B (de) 1980-03-10
IL53948A0 (en) 1978-04-30
SU654173A3 (ru) 1979-03-25
FI62097C (fi) 1982-11-10
NZ186374A (en) 1980-03-05
SG48083G (en) 1984-07-27
BG36499A3 (en) 1984-11-15
LU78974A1 (de) 1979-05-25
IT1105151B (it) 1985-10-28
ZA78630B (en) 1979-10-31
DK48478A (da) 1978-08-04
ATA269579A (de) 1979-08-15
BE863588A (fr) 1978-08-02
FI780324A (fi) 1978-08-04
PL109705B1 (en) 1980-06-30
FI62097B (fi) 1982-07-30
DK150517C (da) 1987-10-19
ES469110A1 (es) 1978-11-16
CA1088064A (en) 1980-10-21
AT355591B (de) 1980-03-10
ES469113A1 (es) 1978-11-16
FR2379542B1 (es) 1982-12-03
IE46185B1 (en) 1983-03-23
ATA11178A (de) 1979-08-15

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19981103