SE426485B - Forfarande att framstella meta-sulfonamido-bensamid-derivat innehallande en pyrrolidinrest - Google Patents

Forfarande att framstella meta-sulfonamido-bensamid-derivat innehallande en pyrrolidinrest

Info

Publication number
SE426485B
SE426485B SE7800982A SE7800982A SE426485B SE 426485 B SE426485 B SE 426485B SE 7800982 A SE7800982 A SE 7800982A SE 7800982 A SE7800982 A SE 7800982A SE 426485 B SE426485 B SE 426485B
Authority
SE
Sweden
Prior art keywords
group
methoxy
formula
ethyl
methylene chloride
Prior art date
Application number
SE7800982A
Other languages
English (en)
Swedish (sv)
Other versions
SE7800982L (sv
Inventor
M Ogata
H Matsumoto
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP52008443A external-priority patent/JPS5920667B2/ja
Priority claimed from JP52094884A external-priority patent/JPS5822110B2/ja
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of SE7800982L publication Critical patent/SE7800982L/xx
Publication of SE426485B publication Critical patent/SE426485B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14Nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/04Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D307/10Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/14Radicals substituted by nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SE7800982A 1977-01-27 1978-01-26 Forfarande att framstella meta-sulfonamido-bensamid-derivat innehallande en pyrrolidinrest SE426485B (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP52008443A JPS5920667B2 (ja) 1977-01-27 1977-01-27 スルホンアミド系ベンズアミド誘導体
JP52094884A JPS5822110B2 (ja) 1977-08-08 1977-08-08 ベンズアミド誘導体の合成法

Publications (2)

Publication Number Publication Date
SE7800982L SE7800982L (sv) 1978-07-28
SE426485B true SE426485B (sv) 1983-01-24

Family

ID=26342958

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7800982A SE426485B (sv) 1977-01-27 1978-01-26 Forfarande att framstella meta-sulfonamido-bensamid-derivat innehallande en pyrrolidinrest

Country Status (18)

Country Link
US (6) US4351770A (fr)
AR (1) AR225881A1 (fr)
AU (1) AU512057B2 (fr)
CA (1) CA1085411A (fr)
CH (1) CH642945A5 (fr)
DE (1) DE2803651A1 (fr)
DK (1) DK154137C (fr)
ES (1) ES466366A1 (fr)
FR (1) FR2378758A1 (fr)
GB (1) GB1557019A (fr)
GR (1) GR70058B (fr)
HU (1) HU176613B (fr)
IE (1) IE46497B1 (fr)
IL (1) IL53881A (fr)
NL (1) NL7801005A (fr)
NZ (1) NZ186175A (fr)
PH (1) PH12853A (fr)
SE (1) SE426485B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2440946A2 (fr) * 1978-01-20 1980-06-06 Ile De France Nouveaux benzamides heterocycliques substitues, leurs procedes de preparation et leur application comme modificateurs du comportement
FR2485526A1 (fr) * 1980-06-24 1981-12-31 Shionogi & Co Procede de preparation de derives de n-(diethylaminoethyl)-2 - alcoxybenzamide, nouveaux produits ainsi obtenus et leurs utilisations comme produits pharmaceutiques antiemetiques ou pour guerir les troubles gastriques
SE8101536L (sv) * 1981-03-11 1982-09-12 Astra Laekemedel Ab Bensamid-derivat
PT77219B (fr) * 1982-08-24 1986-02-04 May & Baker Ltd Procede de preparation des derives de la benzamide
SE8205135D0 (sv) * 1982-09-09 1982-09-09 Astra Laekemedel Ab Benzamido-derivatives
FR2550447B1 (fr) * 1983-08-10 1986-01-17 Ile De France Application du n-(ally-2-pyrrolidinylmethyl) 2-methoxy 4-amino 5-methylsulfamoyl benzamide comme antiagregant plaquettaire
FR2557110B1 (fr) * 1983-12-23 1989-11-24 Sandoz Sa Nouveaux derives d'amines cycliques, leur preparation et leur utilisation comme medicaments
AU567140B2 (en) * 1984-01-06 1987-11-12 Shionogi & Co., Ltd. Sulphonamido-benzamide derivatives
US4544654A (en) * 1984-03-20 1985-10-01 Schering A.G. Substituted sulfonamidobenzamides, antiarrhythmic agents and compositions thereof
CA2057324A1 (fr) * 1990-12-18 1992-06-19 Lora Louise Fitch Agents hypoglycemiques de type benzamide et sulfonamide
CA2350903A1 (fr) * 1998-11-20 2000-06-02 F. Hoffmann-La Roche Ag Antagonistes du recepteur de derives de pyrrolidine-ccr-3
CA2716949A1 (fr) 2008-02-29 2009-09-11 Array Biopharma Inc. Derives de n-(6-aminopyridin-3-yl)-3-(sulfonamido) benzamide comme inhibiteurs de b-raf pour le traitement du cancer
AU2009222144A1 (en) * 2008-02-29 2009-09-11 Array Biopharma Inc. Pyrazole [3, 4-b] pyridine Raf inhibitors
PE20091561A1 (es) 2008-02-29 2009-10-30 Array Biopharma Inc Compuestos inhibidores de raf y metodos para su uso
US20110003809A1 (en) * 2008-02-29 2011-01-06 Array Biopharma Inc. Imidazo [4,5-b] pyridine derivatives used as raf inhibitors

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2334186A (en) * 1938-12-20 1943-11-16 Du Pont Organic sulphonamides and their preparation
GB993584A (fr) * 1962-01-24
US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
US3210370A (en) * 1964-06-22 1965-10-05 Upjohn Co Process for preparing 2, 2'-methylene-bisareneimiazoles
FR5916M (fr) * 1966-01-21 1968-05-06
FR2313935A1 (fr) * 1975-06-10 1977-01-07 Ile De France Nouveaux benzamides substitues, leurs derives et leur procede de preparation
CH547797A (de) * 1971-08-20 1974-04-11 Fratmann Ag Verfahren zur herstellung von n - ((1-aethyl-pyrrolidinyl2)-methyl) -2-methoxy-5-sulfamoyl-benzamid.
US4021229A (en) * 1972-09-05 1977-05-03 Stauffer Chemical Company Sulfonamide herbicide antidote compositions and method of use
IL46696A (en) * 1974-03-05 1978-07-31 Ile De France Substituted n-(2-pyrrolidinylalkyl)benzamides, their preparation and pharmaceutical compositions containing them
CH605793A5 (fr) * 1974-03-05 1978-10-13 Ile De France
FR2294698A1 (fr) * 1974-12-18 1976-07-16 Synthelabo Nouveaux derives des methoxy-2 benzamides substitues, leurs sels, leur preparation et les medicaments qui en renferment

Also Published As

Publication number Publication date
DK154137C (da) 1989-04-10
US4328155A (en) 1982-05-04
IE780145L (en) 1978-07-27
SE7800982L (sv) 1978-07-28
FR2378758A1 (fr) 1978-08-25
AU512057B2 (en) 1980-09-18
AU3268778A (en) 1979-08-02
US4431663A (en) 1984-02-14
US4330472A (en) 1982-05-18
US4328344A (en) 1982-05-04
NZ186175A (en) 1980-03-05
DK154137B (da) 1988-10-17
IL53881A (en) 1981-05-20
GR70058B (fr) 1982-07-26
FR2378758B1 (fr) 1981-02-06
IE46497B1 (en) 1983-06-29
ES466366A1 (es) 1978-10-01
NL7801005A (nl) 1978-07-31
IL53881A0 (en) 1978-04-30
DE2803651A1 (de) 1978-08-03
DE2803651C2 (fr) 1988-10-20
PH12853A (en) 1979-09-12
US4351770A (en) 1982-09-28
US4350635A (en) 1982-09-21
HU176613B (en) 1981-03-28
CA1085411A (fr) 1980-09-09
GB1557019A (en) 1979-12-05
DK37278A (da) 1978-07-28
AR225881A1 (es) 1982-05-14
CH642945A5 (de) 1984-05-15

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