SE415839B - Sett att framstella delta?7215-steroider - Google Patents

Sett att framstella delta?7215-steroider

Info

Publication number
SE415839B
SE415839B SE7611145A SE7611145A SE415839B SE 415839 B SE415839 B SE 415839B SE 7611145 A SE7611145 A SE 7611145A SE 7611145 A SE7611145 A SE 7611145A SE 415839 B SE415839 B SE 415839B
Authority
SE
Sweden
Prior art keywords
steroids
acyl
hydrogen atom
delta
image
Prior art date
Application number
SE7611145A
Other languages
English (en)
Swedish (sv)
Other versions
SE7611145L (sv
Inventor
H Hofmeister
R Wiechert
K Annen
H Laurent
H Steinbeck
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19752546062 external-priority patent/DE2546062A1/de
Priority claimed from DE19762636405 external-priority patent/DE2636405C2/de
Priority claimed from DE19762636407 external-priority patent/DE2636407A1/de
Priority claimed from DE19762636404 external-priority patent/DE2636404C2/de
Application filed by Schering Ag filed Critical Schering Ag
Publication of SE7611145L publication Critical patent/SE7611145L/xx
Publication of SE415839B publication Critical patent/SE415839B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0016—Oximes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE7611145A 1975-10-10 1976-10-07 Sett att framstella delta?7215-steroider SE415839B (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19752546062 DE2546062A1 (de) 1975-10-10 1975-10-10 Delta hoch 15 -steroide
DE19762636405 DE2636405C2 (de) 1976-08-12 1976-08-12 Δ↑1↑↑5↑-17α-Chloräthinyl- und -Propinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate
DE19762636407 DE2636407A1 (de) 1976-08-12 1976-08-12 Delta hoch 15 -steroide
DE19762636404 DE2636404C2 (de) 1976-08-12 1976-08-12 Δ↑1↑↑5↑-17α-Äthinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate

Publications (2)

Publication Number Publication Date
SE7611145L SE7611145L (sv) 1977-04-11
SE415839B true SE415839B (sv) 1980-11-03

Family

ID=27432034

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7611145A SE415839B (sv) 1975-10-10 1976-10-07 Sett att framstella delta?7215-steroider
SE7907224A SE428929B (sv) 1975-10-10 1979-08-30 Delta ?7215-stereoider till anvendning som antifertilitetsmedel

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE7907224A SE428929B (sv) 1975-10-10 1979-08-30 Delta ?7215-stereoider till anvendning som antifertilitetsmedel

Country Status (33)

Country Link
US (1) US4081537A (de)
JP (1) JPS5246060A (de)
AT (1) AT358199B (de)
AU (1) AU500942B2 (de)
BE (1) BE847090A (de)
BG (1) BG34187A3 (de)
CA (1) CA1069885A (de)
CH (2) CH630392A5 (de)
CY (1) CY1119A (de)
DD (1) DD126925B3 (de)
DK (2) DK138749C (de)
ES (1) ES452226A1 (de)
FI (1) FI56389C (de)
FR (1) FR2326927A1 (de)
GB (1) GB1569135A (de)
GR (1) GR60835B (de)
HK (1) HK41381A (de)
HU (1) HU176164B (de)
IE (1) IE43742B1 (de)
IT (1) IT1070580B (de)
KE (1) KE3153A (de)
LU (2) LU75961A1 (de)
MX (1) MX3847E (de)
MY (1) MY8200128A (de)
NL (2) NL187116C (de)
NO (2) NO144490C (de)
NZ (1) NZ182237A (de)
PH (1) PH12941A (de)
PL (1) PL103002B1 (de)
PT (1) PT65697B (de)
SE (2) SE415839B (de)
SU (1) SU671733A3 (de)
YU (1) YU39668B (de)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178784A (en) * 1963-03-27 1965-04-20 Krauthamer Charles Magnetic pocket pencil holder
DE3002746A1 (de) * 1980-01-23 1981-07-30 Schering Ag Berlin Und Bergkamen, 1000 Berlin 1-hydroxysteroide, verfahren zu ihrer herstellung und pharmazeutische praeparate, die diese verbindungen enthalten
DE3005374A1 (de) * 1980-02-11 1981-08-20 Schering Ag Berlin Und Bergkamen, 1000 Berlin 3-desoxy-delta hoch 15 -steroide, verfahren zu ihrer herstellung sowie diese enthaltende pharmazeutische praeparate
DE3042529A1 (de) * 1980-11-07 1982-06-24 Schering Ag, 1000 Berlin Und 4619 Bergkamen 11-methylen- (delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch) -steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3214690A1 (de) * 1982-04-16 1983-10-27 Schering AG, 1000 Berlin und 4709 Bergkamen 11ss-chlor-(delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch)-steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
CN1008820B (zh) * 1985-05-10 1990-07-18 施林工业产权保护股份公司 17α-乙炔基-17β-羟基-18-甲基-4，15-雌甾二烯-3-酮的制备方法
CA1317283C (en) * 1986-11-05 1993-05-04 Douglas Alan Livingston Steroidal 17–-silyl ethers and process to corticoids and progesterones
DE3710728A1 (de) * 1987-03-31 1988-10-13 Schering Ag Verfahren zur herstellung von 17(alpha)-ethinyl-17ss-hydroxy-18-methyl-4,15-estradien-3-on und die neuen zwischenprodukte fuer dieses verfahren
US5512292A (en) * 1990-10-29 1996-04-30 Alza Corporation Transdermal contraceptive formulations methods and devices
EP0555360A1 (de) * 1990-10-29 1993-08-18 Alza Corporation Transdermale verhütungsmittelformulierung, verfahren und vorrichtung
CA2100514C (en) * 1992-07-29 2005-03-29 Johannes A. M. Hamersma 17-spiromethylene steroids
DE4329242A1 (de) * 1993-08-26 1995-03-02 Schering Ag Mittel zur transdermalen Applikation enthaltend Gestodenester
US5567830A (en) * 1994-02-14 1996-10-22 Cocensys, Inc. Process for synthesis of acetylenic carbinols
IT1271004B (it) 1994-09-09 1997-05-26 Ind Chimica Srl Processo per la preparazione del gestodene
JP2004522754A (ja) * 2001-02-02 2004-07-29 ファルマシア・コーポレーション 月経困難症の治療および予防のための組み合わせ治療としてシクロオキシゲナーゼ‐２阻害剤および性ステロイドを使用する方法
UA89766C2 (en) 2003-12-12 2010-03-10 Байер Шеринг Фарма Акциенгезельшафт Transdermal delivery system of gestodene
EP2354150A1 (de) 2010-02-09 2011-08-10 Laboratoire Theramex Verfahren zur Herstellung von Gestoden
PT2613772T (pt) 2010-09-06 2017-03-06 Bayer Ip Gmbh Emplastros transdérmicos de dose baixa com alta libertação de fármaco
CN105237605B (zh) * 2014-07-11 2019-01-25 上海迪赛诺生物医药有限公司 一种用于合成孕二烯酮的中间体及其制备方法和应用
CN115850359B (zh) * 2022-12-14 2024-06-11 梯尔希（南京）药物研发有限公司 一种孕二烯酮杂质i的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3475463A (en) * 1966-07-11 1969-10-28 Sterling Drug Inc 15,16-unsaturated 19-norsteroids and their preparation
US3433785A (en) * 1966-07-11 1969-03-18 Sterling Drug Inc 15,16-disubstituted aromatic steroids,intermediates and processes
DE2439082A1 (de) * 1974-08-12 1976-02-26 Schering Ag 17 alpha-hydroxy-1,3,5(10),15-oestratetraene und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
PL103002B1 (pl) 1979-05-31
NL930071I1 (nl) 1993-09-01
FI56389B (fi) 1979-09-28
FR2326927A1 (fr) 1977-05-06
LU88290I2 (de) 1994-05-04
NO144967C (no) 1981-12-16
IE43742L (en) 1977-04-10
HK41381A (en) 1981-08-28
DK77678A (da) 1978-02-21
NO801013L (no) 1977-04-13
DD126925A5 (de) 1977-08-24
GR60835B (en) 1978-08-31
YU245276A (en) 1982-08-31
ES452226A1 (es) 1977-11-01
CH626636A5 (en) 1981-11-30
FI56389C (fi) 1980-01-10
IT1070580B (it) 1985-03-29
DK143604B (da) 1981-09-14
AT358199B (de) 1980-08-25
AU500942B2 (en) 1979-06-07
KE3153A (en) 1981-09-18
CH630392A5 (de) 1982-06-15
NZ182237A (en) 1978-09-20
HU176164B (en) 1980-12-28
SE428929B (sv) 1983-08-01
NL930071I2 (nl) 1994-02-16
NL7611073A (nl) 1977-04-13
JPS6119640B2 (de) 1986-05-17
IE43742B1 (en) 1981-05-20
NL187116C (nl) 1991-06-03
NL187116B (nl) 1991-01-02
DK138749C (da) 1979-04-02
NO144967B (no) 1981-09-07
FR2326927B1 (de) 1979-09-28
PT65697B (pt) 1978-04-17
CA1069885A (en) 1980-01-15
DD126925B3 (de) 1990-06-06
PH12941A (en) 1979-10-18
MX3847E (es) 1981-08-18
BG34187A3 (en) 1983-07-15
ATA748776A (de) 1980-01-15
BE847090A (fr) 1977-04-08
NO763434L (de) 1977-04-13
MY8200128A (en) 1982-12-31
DK454376A (da) 1977-04-11
JPS5246060A (en) 1977-04-12
FI762876A (de) 1977-04-11
GB1569135A (en) 1980-06-11
NO144490C (no) 1981-09-09
DK138749B (da) 1978-10-23
DK143604C (da) 1982-02-22
CY1119A (en) 1981-12-04
NO144490B (no) 1981-06-01
LU75961A1 (de) 1977-05-09
SE7907224L (sv) 1979-08-30
US4081537A (en) 1978-03-28
SU671733A3 (ru) 1979-06-30
AU1851076A (en) 1978-04-13
SE7611145L (sv) 1977-04-11
YU39668B (en) 1985-03-20
PT65697A (en) 1976-11-01

Similar Documents

Publication Publication Date Title
SE415839B (sv) Sett att framstella delta?7215-steroider
ES441783A1 (es) Procedimiento para la preparacion de 1-alfa-hidroxiesteroi- des.
ES8200648A2 (es) Procedimiento de preparacion de compuestos opacificantes para radiografia y similares
JPS5427578A (en) 1-carboxyalkylcarbamoyl-5-fluorouracil derivatives and their preparation
DK166089C (da) Analogifremgangsmaade til fremstilling af 11beta-chlor-delta15-steroider
ES458818A1 (es) Procedimiento para la produccion de derivados de benzofura- no.
JPS5283823A (en) Naphthohydroxamates
JPS5398974A (en) 1-carbamoyl-5-fluorouracils and process for their preparation
JPS52134634A (en) 3,10-dialkoxy-4-halogeno-13-cyanotriphenodioxazines
JPS53132534A (en) Vanillylacylamide and antioxidant containing the same
ES8204983A1 (es) Un procedimiento para la preparacion de derivados de amino- alcoholes
JPS545924A (en) Derivative of butylaldeyde and its preparation
JPS51131825A (en) Process for preparation of cystindialkylester-n,n'-disuccinate
ES443309A1 (es) Procedimiento para la obtencion de amidas de esteres de aci-dos s-(fenoximetil)-ditiofosforicos.
JPS5210220A (en) Preparation of novel alifatic alcohols possessing-son-ch-ch-linkages i n the carbon chains
JPS5234930A (en) Insecticids
JPS5283446A (en) Preparation of hydrocortisone derivatives
JPS5289651A (en) 5 -amino-3 , 5 -dideoxybutirosins and preparation thereof
JPS5282720A (en) Preparation of cataplasm
JPS52148084A (en) 1-carbamoyluracils and their preparation
JPS5253815A (en) Preparation of n-alkyl-beta-oxybutyramides
JPS5287139A (en) Cyanoaniline derivative

Legal Events

Date Code Title Description
NAL Patent in force

Ref document number: 7611145-9

Format of ref document f/p: F

NUG Patent has lapsed

Ref document number: 7611145-9

Format of ref document f/p: F