RU95105419A - Производные боро-пептидов, их получение и содержащие их медикамент и фармацевтический состав - Google Patents

Производные боро-пептидов, их получение и содержащие их медикамент и фармацевтический состав

Info

Publication number
RU95105419A
RU95105419A RU95105419/04A RU95105419A RU95105419A RU 95105419 A RU95105419 A RU 95105419A RU 95105419/04 A RU95105419/04 A RU 95105419/04A RU 95105419 A RU95105419 A RU 95105419A RU 95105419 A RU95105419 A RU 95105419A
Authority
RU
Russia
Prior art keywords
alkyl group
ris
branched
linear
hydrogen atom
Prior art date
Application number
RU95105419/04A
Other languages
English (en)
Inventor
Сержио Маллар
Fr]
Жильбер Лассаль
Тома Андре Пурселль
Жан Клод Мюлле
Original Assignee
Синтелябо (FR)
Синтелябо
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Синтелябо (FR), Синтелябо filed Critical Синтелябо (FR)
Publication of RU95105419A publication Critical patent/RU95105419A/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Соединения, отвечающие формуле I, приведенной в описании, в форме оптических или геометрических изомеров, представленных в чистой форме или в форме смесей, а также солей, образующихся при добавлении к ним фармацевтически приемлемых кислот и оснований. Терапевтическое применение.

Claims (1)

  1. Соединения, отвечающие формуле I, приведенной в описании, в форме оптических или геометрических изомеров, представленных в чистой форме или в форме смесей, а также солей, образующихся при добавлении к ним фармацевтически приемлемых кислот и оснований. Терапевтическое применение.
RU95105419/04A 1994-04-12 1995-04-11 Производные боро-пептидов, их получение и содержащие их медикамент и фармацевтический состав RU95105419A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9404288A FR2718451B1 (fr) 1994-04-12 1994-04-12 Dérivés de peptides boroniques, leur préparation et leur application en thérapeutique.
FR9404288 1994-04-12

Publications (1)

Publication Number Publication Date
RU95105419A true RU95105419A (ru) 1997-01-10

Family

ID=9461981

Family Applications (1)

Application Number Title Priority Date Filing Date
RU95105419/04A RU95105419A (ru) 1994-04-12 1995-04-11 Производные боро-пептидов, их получение и содержащие их медикамент и фармацевтический состав

Country Status (17)

Country Link
EP (1) EP0677531A1 (ru)
JP (1) JPH07285990A (ru)
KR (1) KR950032225A (ru)
CN (1) CN1113493A (ru)
AU (1) AU1638095A (ru)
CA (1) CA2146833A1 (ru)
CZ (1) CZ92295A3 (ru)
FI (1) FI951726A (ru)
FR (1) FR2718451B1 (ru)
HU (1) HUT71617A (ru)
IL (1) IL113332A0 (ru)
NO (1) NO951418L (ru)
NZ (1) NZ270913A (ru)
PL (1) PL308074A1 (ru)
RU (1) RU95105419A (ru)
SK (1) SK47695A3 (ru)
ZA (1) ZA952983B (ru)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA951618B (en) * 1994-03-04 1996-08-27 Lilly Co Eli Antithrombotic agents
US5726159A (en) * 1994-03-04 1998-03-10 Eli Lilly And Company Antithrombotic agents
US5705487A (en) * 1994-03-04 1998-01-06 Eli Lilly And Company Antithrombotic agents
US5707966A (en) * 1994-03-04 1998-01-13 Eli Lilly And Company Antithrombotic agents
CA2143533A1 (en) * 1994-03-04 1995-09-05 Kenneth D. Kurz Antithrombotic agents
US5602101A (en) * 1994-03-04 1997-02-11 Eli Lilly And Company Antithrombotic agents
US5885967A (en) * 1994-03-04 1999-03-23 Eli Lilly And Company Antithrombotic agents
US5710130A (en) * 1995-02-27 1998-01-20 Eli Lilly And Company Antithrombotic agents
US5914319A (en) * 1995-02-27 1999-06-22 Eli Lilly And Company Antithrombotic agents
US5639739A (en) * 1995-03-24 1997-06-17 The Dupont Merck Pharmaceutical Company Imidazole containing aminoboronic acids
FR2739858B1 (fr) * 1995-10-11 1997-11-14 Synthelabo Derives de n-sulfonyl- et n-sulfamoylpeptidylprolinamide, leur preparation et leur application en therapeutique
US5811402A (en) * 1996-03-22 1998-09-22 Eli Lilly And Company Antithrombotic diamides
FR2758329B1 (fr) * 1997-01-16 1999-02-12 Synthelabo Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US5187157A (en) * 1987-06-05 1993-02-16 Du Pont Merck Pharmaceutical Company Peptide boronic acid inhibitors of trypsin-like proteases
EP0315574A3 (de) * 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin-Inhibitoren

Also Published As

Publication number Publication date
HU9501041D0 (en) 1995-06-28
NO951418L (no) 1995-10-13
CN1113493A (zh) 1995-12-20
FR2718451A1 (fr) 1995-10-13
FR2718451B1 (fr) 1996-05-10
ZA952983B (en) 1996-01-11
NZ270913A (en) 1996-05-28
AU1638095A (en) 1995-10-19
PL308074A1 (en) 1995-10-16
HUT71617A (en) 1996-01-29
IL113332A0 (en) 1995-07-31
KR950032225A (ko) 1995-12-20
FI951726A0 (fi) 1995-04-11
SK47695A3 (en) 1995-12-06
CZ92295A3 (en) 1995-11-15
JPH07285990A (ja) 1995-10-31
EP0677531A1 (fr) 1995-10-18
CA2146833A1 (fr) 1995-10-13
FI951726A (fi) 1995-10-13
NO951418D0 (no) 1995-04-11

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