RU2756273C2 - Полиморфные модификации n-[(3-фтор-4-метоксипиридин-2-ил)метил]-3-(метоксиметил)-1-({ 4-[(2-оксопиридин-1-ил)метил]фенил} метил)пиразол-4-карбоксамида и их соли - Google Patents

Полиморфные модификации n-[(3-фтор-4-метоксипиридин-2-ил)метил]-3-(метоксиметил)-1-({ 4-[(2-оксопиридин-1-ил)метил]фенил} метил)пиразол-4-карбоксамида и их соли Download PDF

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RU2756273C2
RU2756273C2 RU2018139276A RU2018139276A RU2756273C2 RU 2756273 C2 RU2756273 C2 RU 2756273C2 RU 2018139276 A RU2018139276 A RU 2018139276A RU 2018139276 A RU2018139276 A RU 2018139276A RU 2756273 C2 RU2756273 C2 RU 2756273C2
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methyl
fluoro
methoxymethyl
pyrazole
carboxamide
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Хейдн БИТОН
Дэвид Малкольм Кроу
Ханнах Джой ЭДВАРДС
Николас Джеймс ГРИФФИТС-ХЕЙНС
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Калвиста Фармасьютикалз Лимитед
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RU2018139276A 2016-06-01 2017-06-01 Полиморфные модификации n-[(3-фтор-4-метоксипиридин-2-ил)метил]-3-(метоксиметил)-1-({ 4-[(2-оксопиридин-1-ил)метил]фенил} метил)пиразол-4-карбоксамида и их соли RU2756273C2 (ru)

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US201662344059P 2016-06-01 2016-06-01
GBGB1609607.5A GB201609607D0 (en) 2016-06-01 2016-06-01 Polymorphs of N-(3-Fluoro-4-methoxypyridin-2-yl)methyl)-3-(methoxymethyl)-1-({4-((2-oxopy ridin-1-yl)methyl)phenyl}methyl)pyrazole-4-carboxamide and salts
US62/344,059 2016-06-01
GB1609607.5 2016-06-01
PCT/GB2017/051579 WO2017208005A1 (en) 2016-06-01 2017-06-01 Polymorphs of n-[(3-fluoro-4-methoxypyridin-2-yl)methyl]-3-(methoxymethyl)-1 -({4-[2-oxopyridin-1 -yl)methyl]phenyl} methyl) pyrazole -4-carboxamide as kallikrein inhibitors

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RU2018139276A RU2018139276A (ru) 2020-07-10
RU2018139276A3 RU2018139276A3 (enExample) 2020-10-07
RU2756273C2 true RU2756273C2 (ru) 2021-09-29

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