RU2729518C2 - Мета-азациклические производные аминобензойной кислоты в качестве антагонистов пан-интегрина - Google Patents

Мета-азациклические производные аминобензойной кислоты в качестве антагонистов пан-интегрина Download PDF

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RU2729518C2
RU2729518C2 RU2018120935A RU2018120935A RU2729518C2 RU 2729518 C2 RU2729518 C2 RU 2729518C2 RU 2018120935 A RU2018120935 A RU 2018120935A RU 2018120935 A RU2018120935 A RU 2018120935A RU 2729518 C2 RU2729518 C2 RU 2729518C2
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amino
hydroxy
disease
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Питер Г. РУМИНСКИ
Дэвид В. ГРИГГС
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Сент-Луис Юниверсити
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RU2018120935A 2015-12-30 2016-12-30 Мета-азациклические производные аминобензойной кислоты в качестве антагонистов пан-интегрина RU2729518C2 (ru)

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US201562273246P 2015-12-30 2015-12-30
US62/273,246 2015-12-30
PCT/US2016/069511 WO2017117538A1 (en) 2015-12-30 2016-12-30 Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists

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RU2018120935A RU2018120935A (ru) 2020-01-30
RU2018120935A3 RU2018120935A3 (enExample) 2020-03-20
RU2729518C2 true RU2729518C2 (ru) 2020-08-07

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US (3) US10035778B2 (enExample)
EP (2) EP3738953A1 (enExample)
JP (1) JP2019500355A (enExample)
KR (1) KR20180107121A (enExample)
CN (1) CN108779077A (enExample)
AU (1) AU2016381336A1 (enExample)
BR (1) BR112018012981A2 (enExample)
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CA3008023A1 (en) * 2015-12-30 2017-07-06 Saint Louis University Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists
EP3589285A4 (en) 2017-02-28 2020-08-12 Morphic Therapeutic, Inc. INHIBITORS OF INTEGRIN (ALPHA-V) (BETA-6)
MA47697A (fr) 2017-02-28 2020-01-08 Morphic Therapeutic Inc Inhibiteurs de l'(alpha-v)(bêta-6) intégrine
JP7416700B2 (ja) * 2017-11-14 2024-01-17 ザ スキーペンズ アイ リサーチ インスティチュート インコーポレイテッド 増殖性硝子体網膜症および上皮間葉転換と関連付けられる状態の治療のためのｒｕｎｘ１阻害の方法
EP3617206A1 (en) 2018-08-29 2020-03-04 Morphic Therapeutic, Inc. Integrin inhibitors
EP4034236A1 (en) 2019-09-26 2022-08-03 Abionyx Pharma SA Compounds useful for treating liver diseases
IL293894A (en) * 2019-12-20 2022-08-01 Novartis Ag Combination treatment of liver diseases using integrin inhibitors
BR112022023058A2 (pt) * 2020-05-14 2022-12-20 Ube Corp Derivado de 1,4,5,6-tetrahidropirimidin-2-amina
WO2022189856A1 (en) 2021-03-08 2022-09-15 Abionyx Pharma Sa Compounds useful for treating liver diseases
JPWO2023085396A1 (enExample) 2021-11-12 2023-05-19
WO2024262620A1 (ja) * 2023-06-22 2024-12-26 株式会社抗体医学研究所 インテグリン阻害低分子化合物

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WO2014015054A1 (en) * 2012-07-18 2014-01-23 Saint Louis University Beta amino acid derivatives as integrin antagonists
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