AU2016381336A1 - Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists - Google Patents

Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists Download PDF

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Publication number
AU2016381336A1
AU2016381336A1 AU2016381336A AU2016381336A AU2016381336A1 AU 2016381336 A1 AU2016381336 A1 AU 2016381336A1 AU 2016381336 A AU2016381336 A AU 2016381336A AU 2016381336 A AU2016381336 A AU 2016381336A AU 2016381336 A1 AU2016381336 A1 AU 2016381336A1
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disease
compound
amino
disorder
pct
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AU2016381336A
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David W. Griggs
Peter G. Ruminski
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St Louis University
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St Louis University
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
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  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
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  • Communicable Diseases (AREA)
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  • Gastroenterology & Hepatology (AREA)
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  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2016381336A 2015-12-30 2016-12-30 Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists Abandoned AU2016381336A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562273246P 2015-12-30 2015-12-30
US62/273,246 2015-12-30
PCT/US2016/069511 WO2017117538A1 (en) 2015-12-30 2016-12-30 Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists

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AU2016381336A1 true AU2016381336A1 (en) 2018-06-28

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AU2016381336A Abandoned AU2016381336A1 (en) 2015-12-30 2016-12-30 Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists

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US (3) US10035778B2 (enExample)
EP (2) EP3294716B1 (enExample)
JP (1) JP2019500355A (enExample)
KR (1) KR20180107121A (enExample)
CN (1) CN108779077A (enExample)
AU (1) AU2016381336A1 (enExample)
BR (1) BR112018012981A2 (enExample)
CA (1) CA3008023A1 (enExample)
CO (1) CO2018007278A2 (enExample)
ES (1) ES2806276T3 (enExample)
HK (1) HK1244806A1 (enExample)
IL (1) IL259951A (enExample)
PH (1) PH12018501362A1 (enExample)
RU (1) RU2729518C2 (enExample)
SG (1) SG11201805387RA (enExample)
WO (1) WO2017117538A1 (enExample)

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BR112022023058A2 (pt) * 2020-05-14 2022-12-20 Ube Corp Derivado de 1,4,5,6-tetrahidropirimidin-2-amina
WO2022189856A1 (en) 2021-03-08 2022-09-15 Abionyx Pharma Sa Compounds useful for treating liver diseases
EP4431098A4 (en) * 2021-11-12 2025-10-08 Ube Corp PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OR PREVENTION OF ALPORT SYNDROME
EP4733297A1 (en) 2023-06-22 2026-04-29 Antibody Therapeutics, Inc. Integrin-inhibiting small molecule compound

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