RU2159614C2 - Высушенные замораживанием композиции ондансетрона и способ лечения млекопитающих - Google Patents
Высушенные замораживанием композиции ондансетрона и способ лечения млекопитающих Download PDFInfo
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- RU2159614C2 RU2159614C2 RU97110065/14A RU97110065A RU2159614C2 RU 2159614 C2 RU2159614 C2 RU 2159614C2 RU 97110065/14 A RU97110065/14 A RU 97110065/14A RU 97110065 A RU97110065 A RU 97110065A RU 2159614 C2 RU2159614 C2 RU 2159614C2
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Nutrition Science (AREA)
- Engineering & Computer Science (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Physiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Zoology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Detergent Compositions (AREA)
- Orthopedics, Nursing, And Contraception (AREA)
- Fertilizers (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9423511.6 | 1994-11-22 | ||
| GB9423511A GB9423511D0 (en) | 1994-11-22 | 1994-11-22 | Compositions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU97110065A RU97110065A (ru) | 1999-06-10 |
| RU2159614C2 true RU2159614C2 (ru) | 2000-11-27 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU97110065/14A RU2159614C2 (ru) | 1994-11-22 | 1995-11-20 | Высушенные замораживанием композиции ондансетрона и способ лечения млекопитающих |
Country Status (30)
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|---|---|
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| EP (1) | EP0793495B1 (OSRAM) |
| JP (1) | JP3001264B2 (OSRAM) |
| KR (1) | KR970706814A (OSRAM) |
| CN (1) | CN1080118C (OSRAM) |
| AT (1) | ATE193444T1 (OSRAM) |
| AU (1) | AU704160B2 (OSRAM) |
| BE (1) | BE1010250A3 (OSRAM) |
| BR (1) | BR9509808A (OSRAM) |
| CY (1) | CY2166B1 (OSRAM) |
| CZ (1) | CZ285250B6 (OSRAM) |
| DE (1) | DE69517332T2 (OSRAM) |
| DK (1) | DK0793495T3 (OSRAM) |
| ES (1) | ES2147309T3 (OSRAM) |
| FI (1) | FI119355B (OSRAM) |
| FR (1) | FR2727016B1 (OSRAM) |
| GB (2) | GB9423511D0 (OSRAM) |
| GR (1) | GR3033937T3 (OSRAM) |
| HU (1) | HU226891B1 (OSRAM) |
| IL (1) | IL116084A (OSRAM) |
| IT (1) | IT1282352B1 (OSRAM) |
| MX (1) | MX9703735A (OSRAM) |
| NO (1) | NO306893B1 (OSRAM) |
| NZ (1) | NZ296982A (OSRAM) |
| PL (1) | PL181179B1 (OSRAM) |
| PT (1) | PT793495E (OSRAM) |
| RU (1) | RU2159614C2 (OSRAM) |
| TW (1) | TW398976B (OSRAM) |
| WO (1) | WO1996015785A1 (OSRAM) |
| ZA (1) | ZA959821B (OSRAM) |
Families Citing this family (45)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5976577A (en) * | 1997-07-11 | 1999-11-02 | Rp Scherer Corporation | Process for preparing fast dispersing solid oral dosage form |
| US7632517B2 (en) | 1997-10-01 | 2009-12-15 | Novadel Pharma Inc. | Buccal, polar and non-polar spray containing zolpidem |
| EP2042161A1 (en) * | 1997-10-01 | 2009-04-01 | Novadel Pharma Inc. | Propellant-free spray composition comprising anti-emetic agent |
| US20040136914A1 (en) | 1997-10-01 | 2004-07-15 | Dugger Harry A. | Buccal, polar and non-polar spray containing ondansetron |
| US6630006B2 (en) * | 1999-06-18 | 2003-10-07 | The Regents Of The University Of California | Method for screening microcrystallizations for crystal formation |
| ATE311227T1 (de) * | 1999-12-01 | 2005-12-15 | Natco Pharma Ltd | Schnell-wirkende, gefrier-trocknete, orale, pharmazeutische formulierung für die behandlung von migräne |
| RU2162847C1 (ru) * | 2000-07-14 | 2001-02-10 | ООО с иностранными инвестициями "Редди-Биомед лимитед" | Способ получения ондансетрона и его фармацевтически приемлемых солей |
| JP2004525083A (ja) * | 2000-10-30 | 2004-08-19 | テバ ファーマシューティカル インダストリーズ リミティド | 塩酸オンダンセトロンの新規結晶及び溶媒和物形態並びにその製法 |
| US20020115707A1 (en) * | 2001-01-11 | 2002-08-22 | Rami Lidor-Hadas | Process for preparing pure ondansetron hydrochloride dihydrate |
| MXPA04010846A (es) * | 2002-04-29 | 2005-01-25 | Biogal Gyogyszergyar | Proceso para preparar 1, 2, 3, 9-tetrahidro -9- metil-3 -[(2-metil -1h-imidazol -1-il) metil]- 4h- carbazol -4- ona. |
| US20050131045A1 (en) * | 2002-04-30 | 2005-06-16 | Judith Aronhime | Novel crystal forms of ondansetron, processes for their preparation, pharmaceutical, compositions containing the novel forms and methods for treating nausea using them |
| CA2483532A1 (en) * | 2002-04-30 | 2003-11-13 | Biogal Gyogyszergyar Rt. | Novel crystal forms of ondansetron, processes for their preparation, pharmaceutical compositions containing the novel forms and methods for treating nausea using them |
| AU2003302072A1 (en) * | 2002-11-15 | 2004-06-15 | Helsinn Healthcare Sa | Palonosetron for the treatment of chemotherapy-induced emesis |
| JO2735B1 (en) * | 2003-01-30 | 2013-09-15 | هيلسين هيلث كير أس ايه. | Liquid pharmaceutical formations of balloonosterone |
| US8598219B2 (en) | 2003-01-30 | 2013-12-03 | Helsinn Healthcare Sa | Liquid pharmaceutical formulations of palonosetron |
| MY143789A (en) * | 2003-02-18 | 2011-07-15 | Helsinn Healthcare Sa | Use of palonosetron treating post- operative nausea and vomiting |
| US7390503B1 (en) | 2003-08-22 | 2008-06-24 | Barr Laboratories, Inc. | Ondansetron orally disintegrating tablets |
| WO2005040123A1 (en) | 2003-10-10 | 2005-05-06 | Synhton B. V. | Solid-state montelukast |
| DE602005027308D1 (de) * | 2004-01-27 | 2011-05-19 | Synthon Bv | Stabile salze von olanzapin |
| US20050272720A1 (en) * | 2004-01-27 | 2005-12-08 | Rolf Keltjens | Process for making olanzapine Form I |
| US20060167072A1 (en) * | 2004-01-30 | 2006-07-27 | Helsinn Healthcare Sa | Liquid pharmaceutical formulations of palonosetron |
| US7501517B2 (en) * | 2004-04-30 | 2009-03-10 | Synthon Ip, Inc. | Process for making montelukast and intermediates therefor |
| US7829716B2 (en) * | 2004-04-30 | 2010-11-09 | Synthon Pharmaceuticals, Inc. | Process for making montelukast and intermediates therefor |
| DE602005016402D1 (de) * | 2004-05-24 | 2009-10-15 | Genvault Corp | Stabile lagerung von protein und stabile lagerung von nukleinsäure in wiedergewinnbarer form |
| US20060068010A1 (en) * | 2004-09-30 | 2006-03-30 | Stephen Turner | Method for improving the bioavailability of orally delivered therapeutics |
| GB0516604D0 (en) * | 2005-08-12 | 2005-09-21 | Sandoz Ag | Rapidly dispersing/disintegrating compositions |
| EP1919923A1 (en) * | 2005-08-17 | 2008-05-14 | Synthon B.V. | A process for making olanzapine form i |
| AR056815A1 (es) * | 2005-11-18 | 2007-10-24 | Synthon Bv | PROCESO PARA PREPARAR MONTELUKAST, INTERMEDIARIOS DEL MISMO Y SUS SALES DE ADICIoN Y PROCEDIMIENTO DE PURIFICACIoN DE ÉSTOS Y DE MONTELUKAST |
| US8158152B2 (en) * | 2005-11-18 | 2012-04-17 | Scidose Llc | Lyophilization process and products obtained thereby |
| CN101432267A (zh) * | 2006-03-17 | 2009-05-13 | 斯索恩有限公司 | 孟鲁司特金刚烷胺盐 |
| US20070293479A1 (en) * | 2006-05-18 | 2007-12-20 | Osinga Niels J | Olanzapine pharmaceutical composition |
| TWI343262B (en) * | 2006-09-26 | 2011-06-11 | Schering Corp | Rapidly disintegrating lyophilized oral formulations of a thrombin receptor antagonist |
| AR063043A1 (es) * | 2006-09-29 | 2008-12-23 | Synthon Bv | Composicion farmaceutica de olanzapina |
| SI2124556T1 (sl) | 2006-10-09 | 2015-01-30 | Charleston Laboratories, Inc. | Farmacevtske sestave |
| HRP20090341T1 (hr) * | 2006-10-24 | 2009-07-31 | Helsinn Healthcare S.A. | Mekane kapsule koje sadrže palonosetron hidroksiklorid s poboljšanom stabilnosti i bioraspoloživosti |
| US20080260823A1 (en) * | 2007-04-20 | 2008-10-23 | Sciele Pharma, Inc. | Orally disintegrating tablet comprising glycopyrrolate for treating sialorrhea |
| RU2363463C1 (ru) * | 2007-11-14 | 2009-08-10 | Федеральное государственное унитарное предприятие Научно-производственный центр "Фармзащита" Федерального медико-биологического агентства | Лекарственное средство |
| JP5714910B2 (ja) | 2008-01-09 | 2015-05-07 | チャールストン ラボラトリーズ，インコーポレイテッド | 薬学的組成物 |
| EP2276739A1 (en) * | 2008-04-25 | 2011-01-26 | Synthon B.V. | Process for making montelukast intermediates |
| ES2432618T3 (es) * | 2009-05-20 | 2013-12-04 | Inserm (Institut National De La Santé Et De La Recherche Medicale) | Antagonistas del receptor 5-HT3 de serotonina para usar en el tratamiento o prevención de una patología del oído interno con déficit vestibular |
| KR101779991B1 (ko) * | 2009-05-20 | 2017-09-19 | 인쎄름 (엥스띠뛰 나씨오날 드 라 쌍떼 에 드 라 흐쉐르슈 메디깔) | 병소성 전정 질환을 치료하기 위한 세로토닌 5-ｈｔ3 수용체 길항제의 용도 |
| WO2011006012A1 (en) | 2009-07-08 | 2011-01-13 | Charleston Laboratories Inc. | Pharmaceutical compositions |
| US10172833B2 (en) | 2015-08-11 | 2019-01-08 | Insys Development Company, Inc. | Sublingual ondansetron spray |
| WO2017152130A1 (en) | 2016-03-04 | 2017-09-08 | Charleston Laboratories, Inc. | Pharmaceutical compositions |
| ES2975016T3 (es) | 2016-04-14 | 2024-07-02 | Sensorion | (+)-Azasetrón para uso en el tratamiento de trastornos del oído |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| EP0450757A2 (en) * | 1990-02-22 | 1991-10-09 | Glaxo Group Limited | Use of 5-hydroxytryptamine-antagonists in the treatment of mental disorders originating in childhood |
| RU2002745C1 (ru) * | 1989-06-28 | 1993-11-15 | Глэксо Груп Лимитед (Gв) | Способ получени кристаллов дигидрата гидрохлорида ондансетрона уменьшенного размера |
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| EP0084705B1 (en) * | 1981-12-11 | 1987-01-14 | JOHN WYETH & BROTHER LIMITED | Process for preparing solid shaped articles |
| US5288497A (en) * | 1985-05-01 | 1994-02-22 | The University Of Utah | Compositions of oral dissolvable medicaments |
| US5785989A (en) * | 1985-05-01 | 1998-07-28 | University Utah Research Foundation | Compositions and methods of manufacturing of oral dissolvable medicaments |
| GB8516083D0 (en) * | 1985-06-25 | 1985-07-31 | Glaxo Group Ltd | Heterocyclic compounds |
| GB8917556D0 (en) * | 1989-08-01 | 1989-09-13 | Glaxo Group Ltd | Medicaments |
| US5188825A (en) * | 1989-12-28 | 1993-02-23 | Iles Martin C | Freeze-dried dosage forms and methods for preparing the same |
| US5046618A (en) * | 1990-11-19 | 1991-09-10 | R. P. Scherer Corporation | Child-resistant blister pack |
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1994
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1995
- 1995-11-20 HU HU9702135A patent/HU226891B1/hu unknown
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- 1995-11-20 CZ CZ971549A patent/CZ285250B6/cs not_active IP Right Cessation
- 1995-11-20 AU AU41739/96A patent/AU704160B2/en not_active Expired
- 1995-11-20 CN CN95197226A patent/CN1080118C/zh not_active Expired - Lifetime
- 1995-11-20 PT PT95940208T patent/PT793495E/pt unknown
- 1995-11-20 JP JP8516560A patent/JP3001264B2/ja not_active Expired - Lifetime
- 1995-11-20 FR FR9513723A patent/FR2727016B1/fr not_active Expired - Lifetime
- 1995-11-20 DE DE69517332T patent/DE69517332T2/de not_active Expired - Lifetime
- 1995-11-20 IT IT95RM000762A patent/IT1282352B1/it active IP Right Grant
- 1995-11-20 GB GB9523667A patent/GB2295318B/en not_active Expired - Lifetime
- 1995-11-20 KR KR1019970703399A patent/KR970706814A/ko not_active Expired - Lifetime
- 1995-11-20 DK DK95940208T patent/DK0793495T3/da active
- 1995-11-20 RU RU97110065/14A patent/RU2159614C2/ru active
- 1995-11-20 WO PCT/EP1995/004550 patent/WO1996015785A1/en not_active Ceased
- 1995-11-20 ZA ZA959821A patent/ZA959821B/xx unknown
- 1995-11-20 EP EP95940208A patent/EP0793495B1/en not_active Expired - Lifetime
- 1995-11-20 AT AT95940208T patent/ATE193444T1/de active
- 1995-11-20 ES ES95940208T patent/ES2147309T3/es not_active Expired - Lifetime
- 1995-11-20 BR BR9509808A patent/BR9509808A/pt active IP Right Grant
- 1995-11-20 NZ NZ296982A patent/NZ296982A/en not_active IP Right Cessation
- 1995-11-21 BE BE9500955A patent/BE1010250A3/fr active
- 1995-11-21 IL IL11608495A patent/IL116084A/xx not_active IP Right Cessation
- 1995-11-30 TW TW084112791A patent/TW398976B/zh not_active IP Right Cessation
-
1997
- 1997-05-21 MX MX9703735A patent/MX9703735A/es unknown
- 1997-05-21 NO NO972325A patent/NO306893B1/no not_active IP Right Cessation
- 1997-05-21 FI FI972167A patent/FI119355B/fi not_active IP Right Cessation
-
1998
- 1998-04-28 US US09/066,762 patent/US5955488A/en not_active Expired - Lifetime
-
1999
- 1999-01-28 US US09/238,165 patent/US6063802A/en not_active Expired - Lifetime
-
2000
- 2000-05-02 CY CY0000011A patent/CY2166B1/xx unknown
- 2000-07-12 GR GR20000401622T patent/GR3033937T3/el unknown
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2002745C1 (ru) * | 1989-06-28 | 1993-11-15 | Глэксо Груп Лимитед (Gв) | Способ получени кристаллов дигидрата гидрохлорида ондансетрона уменьшенного размера |
| EP0450757A2 (en) * | 1990-02-22 | 1991-10-09 | Glaxo Group Limited | Use of 5-hydroxytryptamine-antagonists in the treatment of mental disorders originating in childhood |
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| Date | Code | Title | Description |
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| PC43 | Official registration of the transfer of the exclusive right without contract for inventions |
Effective date: 20150529 |