RU2153494C2 - 1-n-алкил-n-арилпиримидинамины, способ лечения заболеваний, фармацевтическая композиция - Google Patents
1-n-алкил-n-арилпиримидинамины, способ лечения заболеваний, фармацевтическая композиция Download PDFInfo
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- RU2153494C2 RU2153494C2 RU96109047/04A RU96109047A RU2153494C2 RU 2153494 C2 RU2153494 C2 RU 2153494C2 RU 96109047/04 A RU96109047/04 A RU 96109047/04A RU 96109047 A RU96109047 A RU 96109047A RU 2153494 C2 RU2153494 C2 RU 2153494C2
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- ethyl
- phenyl
- bromo
- alkyl
- pyrimidinamine
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13420993A | 1993-10-12 | 1993-10-12 | |
| US29727494A | 1994-08-26 | 1994-08-26 | |
| US08/297,274 | 1994-08-26 | ||
| US08/134,209 | 1994-08-26 | ||
| US08/315,660 | 1994-09-29 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU96109047A RU96109047A (ru) | 1998-08-20 |
| RU2153494C2 true RU2153494C2 (ru) | 2000-07-27 |
Family
ID=26832075
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU96109047/04A RU2153494C2 (ru) | 1993-10-12 | 1994-10-06 | 1-n-алкил-n-арилпиримидинамины, способ лечения заболеваний, фармацевтическая композиция |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JP3398152B2 (en:Method) |
| CN (1) | CN1142817A (en:Method) |
| FI (1) | FI961599A7 (en:Method) |
| RU (1) | RU2153494C2 (en:Method) |
| TW (1) | TW286316B (en:Method) |
| WO (1) | WO1995010506A1 (en:Method) |
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2305110C2 (ru) * | 2002-01-16 | 2007-08-27 | Дзе Проктер Энд Гэмбл Компани | Агонисты рецептора кортикотропин-рилизинг фактора 2 и их применение |
| RU2308455C2 (ru) * | 2001-11-07 | 2007-10-20 | Ф.Хоффманн-Ля Рош Аг | Аминопиримидины и пиридины |
| RU2325387C2 (ru) * | 2001-12-21 | 2008-05-27 | Анормед Инк. | Гетероциклические соединения с повышенной эффективностью, связывающиеся с рецептором хемокина |
| RU2377241C2 (ru) * | 2003-11-24 | 2009-12-27 | Ф.Хоффманн-Ля Рош Аг | Производные пиразоло-имидазопиримидина, обладающие антагонистической активностью в отношении кортикотропин-рилизинг фактора (crf) |
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1994
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- 1994-10-06 RU RU96109047/04A patent/RU2153494C2/ru active
- 1994-10-06 WO PCT/US1994/011050 patent/WO1995010506A1/en not_active Ceased
- 1994-10-06 CN CN94194465A patent/CN1142817A/zh active Pending
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1996
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| RU2308455C2 (ru) * | 2001-11-07 | 2007-10-20 | Ф.Хоффманн-Ля Рош Аг | Аминопиримидины и пиридины |
| RU2325387C2 (ru) * | 2001-12-21 | 2008-05-27 | Анормед Инк. | Гетероциклические соединения с повышенной эффективностью, связывающиеся с рецептором хемокина |
| RU2305110C2 (ru) * | 2002-01-16 | 2007-08-27 | Дзе Проктер Энд Гэмбл Компани | Агонисты рецептора кортикотропин-рилизинг фактора 2 и их применение |
| RU2377241C2 (ru) * | 2003-11-24 | 2009-12-27 | Ф.Хоффманн-Ля Рош Аг | Производные пиразоло-имидазопиримидина, обладающие антагонистической активностью в отношении кортикотропин-рилизинг фактора (crf) |
| RU2382033C2 (ru) * | 2004-03-02 | 2010-02-20 | Ф.Хоффманн-Ля Рош Аг | Производные 4-(сульфанилпиримидин-4-илметил)морфолина в качестве лигандов gaba-рецептора для лечения тревожности, депрессии и эпилепсии |
| RU2592703C9 (ru) * | 2005-11-15 | 2016-10-20 | Эррей Байофарма Инк. | ИНГИБИТОРЫ ТИПА ErbB |
| RU2592703C2 (ru) * | 2005-11-15 | 2016-07-27 | Эррей Байофарма Инк. | ИНГИБИТОРЫ ТИПА ErbB |
| RU2428421C2 (ru) * | 2005-11-15 | 2011-09-10 | Эррей Байофарма Инк. | Производные n4-фенилхиназолин-4-амина и родственные соединения в качестве ингибиторов рецепторной тирозинкиназы типа erbb для лечения гиперпролиферативных заболеваний |
| RU2436778C2 (ru) * | 2006-07-13 | 2011-12-20 | Байер Кропсайенс Аг | Фунгицидные гидроксимоилтетразольные производные |
| RU2469032C2 (ru) * | 2006-12-13 | 2012-12-10 | Ф.Хоффманн-Ля Рош Аг | Производные 2-(пиперидин-4-ил)-4-фенокси- или фениламинопиримидина в качестве ненуклеозидных ингибиторов обратной транскриптазы |
| RU2481334C2 (ru) * | 2007-08-10 | 2013-05-10 | Альмираль, С.А. | Производные азабифениламинобензойной кислоты в качестве ингибиторов dhodh |
| RU2490015C2 (ru) * | 2008-02-22 | 2013-08-20 | Райджел Фармасьютикалз, Инк. | Применение 2,4-пиримидиндиаминов для лечения атеросклероза |
| RU2393158C1 (ru) * | 2008-10-06 | 2010-06-27 | Андрей Александрович Иващенко | ЗАМЕЩЕННЫЕ 3-АРИЛСУЛЬФОНИЛ-ПИРАЗОЛО[1,5-а]ПИРИМИДИНЫ, АНТАГОНИСТЫ СЕРОТОНИНОВЫХ 5-HT6 РЕЦЕПТОРОВ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ |
| RU2393157C1 (ru) * | 2008-10-06 | 2010-06-27 | Андрей Александрович Иващенко | 2-АЛКИЛАМИНО-3-АРИЛСУЛЬФОНИЛ-ПИРАЗОЛО[1,5-а]ПИРИМИДИНЫ, АНТАГОНИСТЫ СЕРОТОНИНОВЫХ 5-HT6 РЕЦЕПТОРОВ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ |
Also Published As
| Publication number | Publication date |
|---|---|
| TW286316B (en:Method) | 1996-09-21 |
| CN1142817A (zh) | 1997-02-12 |
| FI961599A7 (fi) | 1996-06-07 |
| FI961599A0 (fi) | 1996-04-11 |
| JP3398152B2 (ja) | 2003-04-21 |
| WO1995010506A1 (en) | 1995-04-20 |
| JPH09504520A (ja) | 1997-05-06 |
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