RU2010139315A - Кристаллические формы 5-[3-(2,5-дихлор-4,6-диметил-1-окси-пиридин-3-ил)[1,2,4]оксадиазол-5-ил]-3-нитробензол-1,2-диола - Google Patents

Кристаллические формы 5-[3-(2,5-дихлор-4,6-диметил-1-окси-пиридин-3-ил)[1,2,4]оксадиазол-5-ил]-3-нитробензол-1,2-диола Download PDF

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Publication number
RU2010139315A
RU2010139315A RU2010139315/04A RU2010139315A RU2010139315A RU 2010139315 A RU2010139315 A RU 2010139315A RU 2010139315/04 A RU2010139315/04 A RU 2010139315/04A RU 2010139315 A RU2010139315 A RU 2010139315A RU 2010139315 A RU2010139315 A RU 2010139315A
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Russia
Prior art keywords
further characterized
crystalline modification
peaks
exhibits
modification according
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RU2010139315/04A
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English (en)
Russian (ru)
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Дэвид Александр ЛИРМОНТ (PT)
Дэвид Александр ЛИРМОНТ
Кейт ЛОРИМЕР (US)
Кейт ЛОРИМЕР
Кевин Уэйн МЕЙЕР (US)
Кевин Уэйн МЕЙЕР
Тибор ЭСЕНЬИ (HU)
Тибор ЭСЕНЬИ
Альмошне КОВАЧ (HU)
Альмошне КОВАЧ
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Биал - Портела Энд Ка., С.А. (Pt)
Биал - Портела Энд Ка., С.А.
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Application filed by Биал - Портела Энд Ка., С.А. (Pt), Биал - Портела Энд Ка., С.А. filed Critical Биал - Портела Энд Ка., С.А. (Pt)
Publication of RU2010139315A publication Critical patent/RU2010139315A/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
RU2010139315/04A 2008-03-17 2009-03-16 Кристаллические формы 5-[3-(2,5-дихлор-4,6-диметил-1-окси-пиридин-3-ил)[1,2,4]оксадиазол-5-ил]-3-нитробензол-1,2-диола RU2010139315A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6972108P 2008-03-17 2008-03-17
US61/069,721 2008-03-17

Publications (1)

Publication Number Publication Date
RU2010139315A true RU2010139315A (ru) 2012-04-27

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Family Applications (1)

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RU2010139315/04A RU2010139315A (ru) 2008-03-17 2009-03-16 Кристаллические формы 5-[3-(2,5-дихлор-4,6-диметил-1-окси-пиридин-3-ил)[1,2,4]оксадиазол-5-ил]-3-нитробензол-1,2-диола

Country Status (16)

Country Link
US (2) US8975410B2 (https=)
EP (1) EP2276758B1 (https=)
JP (2) JP2011514380A (https=)
KR (1) KR20110002462A (https=)
CN (1) CN102015696A (https=)
AR (1) AR070907A1 (https=)
AU (1) AU2009226221A1 (https=)
BR (1) BRPI0908731A2 (https=)
CA (1) CA2718772C (https=)
CL (1) CL2009000628A1 (https=)
ES (1) ES2565080T3 (https=)
IL (1) IL207854A0 (https=)
MX (1) MX2010009610A (https=)
RU (1) RU2010139315A (https=)
TW (1) TW200942531A (https=)
WO (1) WO2009116882A1 (https=)

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Publication number Publication date
AR070907A1 (es) 2010-05-12
MX2010009610A (es) 2010-09-30
CA2718772C (en) 2017-05-02
JP2011514380A (ja) 2011-05-06
CA2718772A1 (en) 2009-09-24
US9845316B2 (en) 2017-12-19
TW200942531A (en) 2009-10-16
ES2565080T3 (es) 2016-03-31
KR20110002462A (ko) 2011-01-07
CL2009000628A1 (es) 2010-04-09
JP2015044837A (ja) 2015-03-12
WO2009116882A1 (en) 2009-09-24
EP2276758B1 (en) 2016-01-06
CN102015696A (zh) 2011-04-13
IL207854A0 (en) 2010-12-30
AU2009226221A1 (en) 2009-09-24
EP2276758A1 (en) 2011-01-26
US20150166519A1 (en) 2015-06-18
US8975410B2 (en) 2015-03-10
BRPI0908731A2 (pt) 2017-05-16
US20110112301A1 (en) 2011-05-12

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