RU2010114001A - Применение пептида в качестве терапевтического средства - Google Patents

Применение пептида в качестве терапевтического средства Download PDF

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RU2010114001A
RU2010114001A RU2010114001/15A RU2010114001A RU2010114001A RU 2010114001 A RU2010114001 A RU 2010114001A RU 2010114001/15 A RU2010114001/15 A RU 2010114001/15A RU 2010114001 A RU2010114001 A RU 2010114001A RU 2010114001 A RU2010114001 A RU 2010114001A
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disease
diseases
pharmaceutical composition
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val
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Дориан БЕВЕК (DE)
Дориан БЕВЕК
Фабио КАВАЛЛИ (CH)
Фабио КАВАЛЛИ
Вера КАВАЛЛИ (CH)
Вера КАВАЛЛИ
Геральд БАХЕР (DE)
Геральд БАХЕР
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Мондобайотек Лабораториз Аг (Li)
Мондобайотек Лабораториз Аг
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Abstract

1. Применение пептида Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Gln-Phe-Lys-Val-Val-Thr-OH для получения фармацевтической композиции для лечения и/или профилактики злокачественной опухоли, аутоиммунных заболеваний, фиброзов, воспалительных заболеваний, нейродегенеративных заболеваний, инфекционных заболеваний, заболеваний легких, заболеваний сердца и сосудов и болезней обмена веществ. ! 2. Применение пептида по п.1, где злокачественная опухоль, аутоиммунное заболевание, фиброз, воспалительное заболевание, нейродегенеративное заболевание, инфекционное заболевание, заболевание легких, заболевание сердца и сосудов или болезнь обмена веществ выбраны из инфекции Streptococus pneumoniae, связанных с инфекцией Streptococus pneumoniae заболеваний, а именно гемолитического уремического синдрома, пневмонии, осложнения кистозного фиброза, заболеваний среднего уха, инфекций в кровотоке, инфекции синусов и ушей, острого синусита, отита среднего уха, остеомиелита, септического артрита, эндокардита, перитонита, перикардита и абсцесса головного мозга. ! 3. Применение пептида по п.1 или 2 для получения состава для перорального введения новорожденным, детям ясельного возраста и/или детям дошкольного возраста. ! 4. Применение пептида по п.1 или 2 для получения лиофилизированного состава или буферного жидкого состава. ! 5. Фармацевтическая композиция, содержащая пептид Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Gln-Phe-Lys-Val-Val-Thr-OH, по меньшей мере, совместно с одним фармацевтически приемлемым носителем, криопротектором, лиопротектором, эксципиентом и/или разбавителем. ! 6. Фармацевтическая композиция по п.5 в форме лиофилизата или жидкого буферного раствора. ! 7. Фармацевтическая композиция по п.5 или 6, пригодная для

Claims (9)

1. Применение пептида Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Gln-Phe-Lys-Val-Val-Thr-OH для получения фармацевтической композиции для лечения и/или профилактики злокачественной опухоли, аутоиммунных заболеваний, фиброзов, воспалительных заболеваний, нейродегенеративных заболеваний, инфекционных заболеваний, заболеваний легких, заболеваний сердца и сосудов и болезней обмена веществ.
2. Применение пептида по п.1, где злокачественная опухоль, аутоиммунное заболевание, фиброз, воспалительное заболевание, нейродегенеративное заболевание, инфекционное заболевание, заболевание легких, заболевание сердца и сосудов или болезнь обмена веществ выбраны из инфекции Streptococus pneumoniae, связанных с инфекцией Streptococus pneumoniae заболеваний, а именно гемолитического уремического синдрома, пневмонии, осложнения кистозного фиброза, заболеваний среднего уха, инфекций в кровотоке, инфекции синусов и ушей, острого синусита, отита среднего уха, остеомиелита, септического артрита, эндокардита, перитонита, перикардита и абсцесса головного мозга.
3. Применение пептида по п.1 или 2 для получения состава для перорального введения новорожденным, детям ясельного возраста и/или детям дошкольного возраста.
4. Применение пептида по п.1 или 2 для получения лиофилизированного состава или буферного жидкого состава.
5. Фармацевтическая композиция, содержащая пептид Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Gln-Phe-Lys-Val-Val-Thr-OH, по меньшей мере, совместно с одним фармацевтически приемлемым носителем, криопротектором, лиопротектором, эксципиентом и/или разбавителем.
6. Фармацевтическая композиция по п.5 в форме лиофилизата или жидкого буферного раствора.
7. Фармацевтическая композиция по п.5 или 6, пригодная для внутривенного введения, перорального введения или для введения посредством ингаляции.
8. Фармацевтическая композиция по п.5 или 6 в форме состава искусственного материнского молока или заменителя материнского молока, пригодная для пероральной доставки новорожденным, детям ясельного возраста и/или детям дошкольного возраста.
9. Фармацевтическая композиция по п.5 или 6, пригодная для лечения и/или профилактики злокачественной опухоли, аутоиммунного заболевания, фиброза, воспалительного заболевания, нейродегенеративного заболевания, инфекционного заболевания, заболевания легких, заболевания сердца и сосудов или болезней обмена веществ.
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2528094C2 (ru) * 2012-08-03 2014-09-10 Татьяна Георгиевна Емельянова Средство пептидной структуры, обладающее анальгетическим, противовоспалительным действием, и лекарственные формы на его основе

Families Citing this family (53)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1697035B1 (en) * 2003-12-22 2017-11-15 Warren H. Finlay Powder formation by atmospheric spray-freeze drying
EP3404102B1 (en) 2004-04-21 2021-08-11 Alexion Pharmaceuticals, Inc. Bone delivery conjugates and method of using same to target proteins to bone
WO2009033745A2 (en) * 2007-09-11 2009-03-19 Mondobiotech Laboratories Ag Use of a peptide as a therapeutic agent
WO2009083844A1 (en) 2007-12-20 2009-07-09 Koninklijke Philips Electronics N.V. Method and device for case-based decision support
KR101760758B1 (ko) 2008-05-14 2017-07-24 애그리컬쳐 빅토리아 서비스 피티와이 엘티디 질병 및 장애를 치료하기 위한 안지오게닌 또는 안지오게닌 아고니스트의 이용
AU2013204721B2 (en) * 2008-05-14 2016-08-18 Agriculture Victoria Services Pty Ltd Methods for treating cachexia
WO2011047287A1 (en) * 2009-10-15 2011-04-21 Immuneregen Biosciences, Inc. Methods of treating inflammatory and fibrotic lung diseases with substance p analogs
AU2011350066A1 (en) 2010-12-27 2013-07-11 Alexion Pharma International Sarl Compositions comprising natriuretic peptides and methods of use thereof
EP2476441A1 (en) 2011-01-13 2012-07-18 Universitat Autònoma De Barcelona Methods and reagents for efficient and targeted delivery of therapeutic molecules to CXCR4 cells
SG187271A1 (en) * 2011-07-07 2013-02-28 Agency Science Tech & Res Anti-amyloidogenic, alpha-helix breaking ultra-small peptide therapeutic
WO2013051767A1 (ko) * 2011-10-06 2013-04-11 중앙대학교 산학협력단 안지오제닌의 신규 용도
US10272133B2 (en) 2011-10-06 2019-04-30 Vanderbilt University Compositions and methods for treating and preventing hyperlipidemia, fatty liver, atherosclerosis and other disorders associated with metabolic syndrome
KR101327663B1 (ko) * 2011-10-07 2013-11-14 중앙대학교 산학협력단 안지오제닌의 신규 용도
WO2013052813A1 (en) 2011-10-06 2013-04-11 Vanderbilt University Compositions and methods for treating and preventing hyperlipidemia, fatty liver, atherosclerosis and other disorders associated with metabolic syndrome
CN102973926A (zh) * 2011-11-20 2013-03-20 上海市肺科医院 胸腺肽α1在制备治疗肺纤维化药物中的用途
CN108653715A (zh) * 2011-12-16 2018-10-16 卡乐斯治疗公司 用于治疗视网膜病症和疾病的anp、bnp以及cnp相关肽及其衍生物的方法和用途
JP6198715B2 (ja) 2012-03-06 2017-09-20 武田薬品工業株式会社 三環性化合物
RU2507212C3 (ru) * 2012-03-28 2022-05-04 Общество С Ограниченной Ответственностью "Айвикс" Способ получения рекомбинантного пептида и полученный пептид
AU2013204740C1 (en) * 2012-05-10 2015-10-01 Agriculture Victoria Services Pty Ltd Methods of treating cancer using angiogenin or an angiogenin agonist
US10052366B2 (en) 2012-05-21 2018-08-21 Alexion Pharmaceuticsl, Inc. Compositions comprising alkaline phosphatase and/or natriuretic peptide and methods of use thereof
WO2014007547A1 (en) * 2012-07-03 2014-01-09 Il Yang Pharm. Co.,Ltd. Novel peptides and use thereof
WO2014021942A1 (en) * 2012-08-01 2014-02-06 University Of Southern California Methods for limiting development of neurodegeneration
WO2014039504A1 (en) * 2012-09-04 2014-03-13 Lauren Sciences Llc Bolaamphiphilic compounds, compositions and uses thereof
CN105102485B (zh) 2013-02-05 2019-04-19 特普塞拉公司 磷酸胆碱缀合物及其用途
US10046021B2 (en) 2013-02-05 2018-08-14 Tpcera Ltd. Phosphorylcholine conjugates and uses thereof
US9492544B2 (en) * 2013-04-11 2016-11-15 Vanderbilt University Compositions and methods for targeting nuclear import shuttles and treating inflammatory disorders
US11571455B2 (en) * 2013-04-11 2023-02-07 Vanderbilt University Methods and compositions for treating alcoholic liver disease
CN104662034B (zh) * 2013-05-28 2021-05-11 "Ivix"有限公司 用于生产重组肽的方法及所得到的肽
CN103613643B (zh) * 2013-12-04 2015-04-22 南京晓庄学院 一种生物活性小肽、其合成方法及其作为畜禽饲料添加剂的用途
WO2015179490A1 (en) * 2014-05-21 2015-11-26 Stemnion, Inc. Treatment of diseases and conditions caused by increased vascular permeability
US10822596B2 (en) 2014-07-11 2020-11-03 Alexion Pharmaceuticals, Inc. Compositions and methods for treating craniosynostosis
BR112017011900A2 (pt) 2014-12-05 2018-02-27 Alexion Pharma Inc tratamento de ataques com fosfatase alcalina recombinante
DE102015201100B4 (de) * 2015-01-22 2018-05-17 Friedrich-Alexander-Universität Erlangen-Nürnberg Antivirale Mittel
JP6868561B2 (ja) 2015-01-28 2021-05-12 アレクシオン ファーマシューティカルズ, インコーポレイテッド アルカリホスファターゼ欠損を有する被験者を治療する方法
MX2018002121A (es) 2015-08-17 2018-06-18 Alexion Pharma Inc Elaboracion de fosfatasas alcalinas.
US11229686B2 (en) 2015-09-28 2022-01-25 Alexion Pharmaceuticals, Inc. Reduced frequency dosage regimens for tissue non-specific alkaline phosphatase (TNSALP)-enzyme replacement therapy of hypophosphatasia
WO2017074466A1 (en) 2015-10-30 2017-05-04 Alexion Pharmaceuticals, Inc. Methods for treating craniosynostosis in a patient
WO2017155569A1 (en) 2016-03-08 2017-09-14 Alexion Pharmaceuticals, Inc. Methods for treating hypophosphatasia in children
WO2017173413A1 (en) 2016-04-01 2017-10-05 Alexion Pharmaceuticals, Inc. Treating muscle weakness with alkaline phosphatases
US10898549B2 (en) 2016-04-01 2021-01-26 Alexion Pharmaceuticals, Inc. Methods for treating hypophosphatasia in adolescents and adults
WO2017214130A1 (en) 2016-06-06 2017-12-14 Alexion Pharmaceuticals, Inc. Metal impact on manufacturing of alkaline phosphatases
EP3500289A4 (en) 2016-08-18 2020-05-06 Alexion Pharmaceuticals, Inc. METHODS OF TREATING TRACHEOBRONCHOMALACIA
RU2626002C1 (ru) 2016-10-24 2017-07-21 Общество С Ограниченной Ответственностью "Айвикс" Новая группа пептидов для лечения женской сексуальной дисфункции
CA3051855A1 (en) * 2017-01-27 2018-08-02 Vanderbilt University Fused in sarcoma (fus) nuclear translocation inhibitors for preventing fibrosis
CN106860855B (zh) * 2017-03-01 2021-06-11 成都惠泰生物医药有限公司 多肽及多肽衍生物在预防和治疗纤维化疾病中的应用
AU2018243320A1 (en) 2017-03-31 2019-10-10 Alexion Pharmaceuticals, Inc. Methods for treating hypophosphatasia (HPP) in adults and adolescents
EP3717504A4 (en) * 2017-11-27 2021-10-20 The University of Hong Kong YEAT INHIBITORS AND THEIR METHODS OF USE
WO2019190752A1 (en) 2018-03-30 2019-10-03 Alexion Pharmaceuticals, Inc. Manufacturing of glycoproteins
EP3773497B1 (en) * 2018-04-09 2023-10-18 Elgan Pharma Ltd. Oxytocin compositions and methods of use
US20220072095A1 (en) * 2018-09-14 2022-03-10 Vanderbilt University Methods and compositions for treating skin diseases
KR20210095132A (ko) * 2018-10-04 2021-07-30 럿거스, 더 스테이트 유니버시티 오브 뉴 저지 뉴로메딘 펩티드를 이용하여 2형 사이토카인 매개 염증을 감소시키는 방법
CN112386678B (zh) * 2019-08-13 2023-07-07 成都惠泰生物医药有限公司 多肽或其衍生物的应用
WO2022149159A1 (en) * 2021-01-05 2022-07-14 Jaya Shukla Molecular imaging complex for positron emission tomography

Family Cites Families (105)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3778426A (en) * 1970-12-16 1973-12-11 Research Corp Therapeutically useful polypeptides
US4041155A (en) * 1974-10-29 1977-08-09 American Home Products Corporation Long acting somatostatin composition
US4100271A (en) 1976-02-26 1978-07-11 Cooper Laboratories, Inc. Clear, water-miscible, liquid pharmaceutical vehicles and compositions which gel at body temperature for drug delivery to mucous membranes
US4188373A (en) 1976-02-26 1980-02-12 Cooper Laboratories, Inc. Clear, water-miscible, liquid pharmaceutical vehicles and compositions which gel at body temperature for drug delivery to mucous membranes
US4235988A (en) 1976-12-13 1980-11-25 Imperial Chemical Industries Limited Delivery means for biologically active agents
US4125605A (en) * 1977-10-19 1978-11-14 The United States Government Method of employing oral TRH
JPS56138154A (en) * 1980-02-28 1981-10-28 Genentech Inc Desacetylthymosin-alpha-1 and manufacture
US4481139A (en) * 1983-04-13 1984-11-06 Board Of Regents, The University Of Texas System Peptide antagonists of substance P
US4478822A (en) 1983-05-16 1984-10-23 Merck & Co., Inc. Drug delivery system utilizing thermosetting gels
US4474753A (en) 1983-05-16 1984-10-02 Merck & Co., Inc. Topical drug delivery system utilizing thermosetting gels
US4474751A (en) 1983-05-16 1984-10-02 Merck & Co., Inc. Ophthalmic drug delivery system utilizing thermosetting gels
US4474752A (en) 1983-05-16 1984-10-02 Merck & Co., Inc. Drug delivery system utilizing thermosetting gels
US4705778A (en) * 1985-10-22 1987-11-10 Sri International Orally active LHRH analogs
US5691310A (en) * 1987-09-29 1997-11-25 Vesely; David L. Methods of treatment using proANF peptides
SE8803847A0 (sv) * 1988-10-27 1990-04-28 Kabigen Ab Neuromodulerande peptid
US5432176A (en) * 1988-11-29 1995-07-11 The John Hopkins University Method of retarding the progression of chronic renal failure
US5118670A (en) * 1988-12-14 1992-06-02 Massachusetts Institute Of Technology Process and composition for increasing brain dopamine release
US4874744A (en) * 1989-03-13 1989-10-17 University Of Cincinnati Method of using melanocyte stimulating hormone as dermatis treatment
US5217955A (en) * 1989-09-15 1993-06-08 Biomeasure, Inc. Treatment of cancer with peptide analog of bombesin, grp, litorin or neuromedin
US5256396A (en) 1990-01-24 1993-10-26 Colgate-Palmolive Company Topical composition
JP3130080B2 (ja) * 1990-12-27 2001-01-31 日清製粉株式会社 ペプチドおよびその製造方法
ES2110986T3 (es) 1991-08-12 1998-03-01 Nestle Sa Composicion alimenticia.
US5308833A (en) * 1992-02-06 1994-05-03 Sciclone Pharmaceuticals Method for treating hepatitis B carriers with minimal disease
AU5081193A (en) * 1992-08-31 1994-03-29 Magainin Pharmaceuticals, Inc. Treatment of gynecological malignancies with biologically active peptides
US6200952B1 (en) * 1993-06-02 2001-03-13 Sciclone Pharmaceuticals, Inc. Combination therapy method for treating chronic hepatitis B
WO1995008337A1 (en) * 1993-09-24 1995-03-30 The University Of Southern California Use of angiotensin iii and analogs thereof in tissue repair
US5449761A (en) * 1993-09-28 1995-09-12 Cytogen Corporation Metal-binding targeted polypeptide constructs
WO1995030418A1 (en) * 1994-05-09 1995-11-16 The Johns Hopkins University Method of slowing the progression of hiv infection
US7553929B2 (en) * 1994-06-13 2009-06-30 Vanderbilt University Cell permeable peptides for inhibition of inflammatory reactions and methods of use
US6495518B1 (en) * 1994-06-13 2002-12-17 Vanderbilt University Method for importing biologically active molecules into cells
CZ262698A3 (cs) 1996-02-19 1999-03-17 Nycomed Imaging A/S Kontrastní prostředek pro zobrazování ultrazvukem a způsob jeho výroby
JPH09227590A (ja) * 1996-02-27 1997-09-02 Nisshin Flour Milling Co Ltd ペプチド
US5691314A (en) * 1996-03-18 1997-11-25 The Medical College Of Hampton Roads Adjunctive therapy
TW360501B (en) 1996-06-27 1999-06-11 Nestle Sa Dietetically balanced milk product
US6492330B1 (en) * 1996-08-16 2002-12-10 National Institute Of Immunology Antiangiogenic drugs
DK0832565T3 (da) 1996-09-24 2000-11-20 Nestle Sa Mælkeerstatningsprodukt og fremgangsmåde til fremstilling deraf
US5830434A (en) * 1997-02-26 1998-11-03 Medical University Of South Carolina Foundation For Research Development Methods of treating non-insulin dependent diabetes mellitus with pancreatic polypeptide
SE9701162D0 (sv) * 1997-03-27 1997-03-27 Karolinska Innovations Ab New use II
WO1999003491A1 (en) * 1997-07-15 1999-01-28 Novo Nordisk A/S New use of nociceptin
WO1999040106A2 (en) * 1998-02-09 1999-08-12 University Of Southern California Use of angiotensin analogues for promoting erythropoiesis
SE9801571D0 (sv) * 1998-05-05 1998-05-05 Wapharm Ab Melanokortin-1-receptorselektiva föreningar
US6333313B1 (en) * 1998-10-29 2001-12-25 Board Of Regents, The University Of Texas System Clinical use of oxytocin alone or in combination to treat bone disorders
DE69919019T2 (de) 1998-11-24 2004-11-25 Société des Produits Nestlé S.A. Verfahren zur Herstellung einer Proteinzusammensetzung und einer diese enthaltenden Säuglingsnahrung
EP1144597A2 (en) * 1999-01-21 2001-10-17 Vitro Diagnostics, Inc. Immortalized cell lines and methods of making the same
US20040013641A1 (en) 1999-04-15 2004-01-22 Monash University Disease prevention by reactivation of the thymus
US6313370B1 (en) * 1999-04-29 2001-11-06 Morton Hyson Medicated wrap
US6849714B1 (en) * 1999-05-17 2005-02-01 Conjuchem, Inc. Protection of endogenous therapeutic peptides from peptidase activity through conjugation to blood components
CA2499211A1 (en) * 1999-05-17 2000-11-23 Conjuchem Inc. Modified peptides yy and conjugates thereof
JP2003501394A (ja) * 1999-06-04 2003-01-14 ノボ ノルディスク アクティーゼルスカブ 延長された重度の疾患の異化状態の処理のための組成物
US6894026B1 (en) * 2000-01-11 2005-05-17 Atossa Healthcare, Inc. Long-acting oxytocin analogues for the treatment and prevention of breast cancer and psychiatric disorders
SE0001440D0 (sv) * 2000-04-18 2000-04-18 Entretech Medical Ab A drug against climacteric disorders
AU2001257129A1 (en) * 2000-04-21 2001-11-07 Advanced Research And Technology Institute, Inc. Novel pharmacotherapeutic process and composition for central nervous system disorders
WO2001096527A2 (en) * 2000-06-14 2001-12-20 Chanda Zaveri Peptides with physiological activity
CA2412899C (en) 2000-07-05 2010-11-09 Takeda Chemical Industries, Ltd. Medicinal preparations for treating sex hormone-dependent diseases
EP1305338A2 (en) * 2000-08-02 2003-05-02 Theratechnologies Inc. Modified peptides with increased potency
CN1283314C (zh) * 2000-08-31 2006-11-08 盐野义制药株式会社 抗帕金森氏病药
AU2001297873A1 (en) * 2000-11-21 2003-01-02 New England Medical Center Novel antimicrobial compounds
US20020103131A1 (en) * 2001-01-26 2002-08-01 Jacobson Jill D. Prevention of diabetes by administration of GnRH antagonists
SE0100684D0 (sv) * 2001-02-28 2001-02-28 Kerstin Uvnaes Moberg New subject-matter
US7019109B2 (en) * 2001-03-16 2006-03-28 The Salk Institute For Bilogical Studies SSTR1-selective analogs
US6682753B2 (en) 2001-03-23 2004-01-27 Neuronz Limited Methods for promoting weight gain using GPE-related compounds
EP1389126B1 (en) * 2001-04-18 2016-12-21 The Regents of The University of California Retrocyclins: antiviral and antimicrobial peptides
IL156777A0 (en) * 2001-04-30 2004-02-08 Zentaris Gmbh Treatment of dementia and neurodegenerative diseases with intermediate doses of lhrh antagonists
AU2002316221A1 (en) * 2001-05-16 2002-11-25 Nicholas P. Plotnikoff Methods for inducing sustained immune response
WO2002096934A1 (en) * 2001-05-25 2002-12-05 Kemia, Inc. Non-natural galanin receptor ligands
GB0115515D0 (en) * 2001-06-25 2001-08-15 Ferring Bv Oxytocin agonisys
DE10137174A1 (de) * 2001-07-31 2003-02-13 Zentaris Ag Verwendung von LHRH-Antagonisten in nichtkastrierenden Dosen zur Verbesserung der T-Zellen-vermittelten Immunität
SE0102910D0 (sv) * 2001-08-31 2001-08-31 Moberg Kerstin Uvnaes New use
WO2003020223A2 (en) * 2001-09-05 2003-03-13 James Lipton A cancer treatment system
US6770625B2 (en) * 2001-09-07 2004-08-03 Nobex Corporation Pharmaceutical compositions of calcitonin drug-oligomer conjugates and methods of treating diseases therewith
ES2287065T3 (es) 2001-11-23 2007-12-16 Societe Des Produits Nestle S.A. Proceso para la preparacion de leche en polvo y productos lacteos concentrados.
CA2391118A1 (en) * 2002-06-21 2003-12-21 Universite Du Quebec A Montreal Oxytocin as cardiomyogenesis inducer and uses thereof
US7655772B2 (en) * 2002-09-06 2010-02-02 University Of South Florida Materials and methods for treatment of allergic diseases
IL152289A0 (en) * 2002-10-14 2003-05-29 Vectabiotics Ltd Method and composition for inhibiting h.pylori infection in a mammalian tissue
US20040152769A1 (en) * 2002-11-09 2004-08-05 Ekwuribe Nnochiri Nkem Modified carbamate-containing prodrugs and methods of synthesizing same
US8309117B2 (en) * 2002-12-19 2012-11-13 Novartis, Ag Method for making medical devices having antimicrobial coatings thereon
EP1608318A4 (en) * 2003-03-27 2009-07-29 Univ Emory CXCR4 ANTAGONISTS AND METHODS OF USE
EP1663282A4 (en) * 2003-09-24 2007-09-19 Vecta Ltd ORAL COMPOSITIONS FOR STIMULATING MAGNESIC ACID DETERRECTION WITH PENTAAGASTRINE
EP1687452A4 (en) * 2003-09-30 2008-08-06 Centocor Inc HUMAN HINGE-CORE MIMETICORPS, COMPOSITIONS, METHODS AND APPLICATIONS THEREOF
EP1522311A1 (fr) 2003-10-10 2005-04-13 Institut National De La Sante Et De La Recherche Medicale (Inserm) Utilisation de la somatostine ou d'un de ses analogues pour préparer un médicament destiné à réguler la réserve folliculaire ovarienne chez la femme non ménopausée
JP2007509169A (ja) * 2003-10-23 2007-04-12 ニューレン ファーマシューティカルズ リミテッド 静脈内注入後のGly−Pro−Gluの神経保護効果
US20070053954A1 (en) * 2003-10-24 2007-03-08 Rowe Stephen C Macromer-melt formulations
WO2005094420A2 (en) * 2004-02-17 2005-10-13 University Of South Florida Materials and methods for treatment of inflammatory and cell proliferation disorders
US7776815B2 (en) * 2004-02-24 2010-08-17 Wisconsin Alumni Research Foundation Use of neuropeptides for ligament healing
WO2005097158A1 (en) * 2004-03-29 2005-10-20 The Arizona Board Of Regents On Behalf Of The University Of Arizona Amphipathic glycopeptides
WO2005097161A2 (en) 2004-03-30 2005-10-20 Neuren Pharmaceuticals Limited Gpe and g-2mepe, caffeine and alkanol for treatment of cns injury
US7462595B2 (en) * 2004-09-17 2008-12-09 Prange Jr Arthur Jergen Methods for treating cancer-related fatigue
AU2005319578A1 (en) * 2004-11-24 2006-06-29 Neopro Labs, Llc Methods and compositions for treating conditions
WO2006063596A2 (en) * 2004-12-15 2006-06-22 Aditech Pharma Ab A composition comprising pp for the treatment of gastrointestinal disorders
WO2006085075A2 (en) * 2005-02-09 2006-08-17 Da Volterra Colonic delivery of active agents
US20060205642A1 (en) * 2005-03-08 2006-09-14 Vesely David L Oral methods of treatment using proANF peptides
WO2006119388A2 (en) 2005-05-03 2006-11-09 Novetide, Ltd. Methods for the production of peptide having a c-terminal amide
EP1888618A4 (en) 2005-05-23 2009-07-15 Neuren Pharmaceuticals Ltd GLYCYL-PROLYL-GLUTAMATE ANALOGS
JP5276982B2 (ja) * 2005-08-26 2013-08-28 ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティ オキシトシンの投与による頭痛の処置のための方法
US20090069233A1 (en) * 2005-09-13 2009-03-12 Abburi Ramaiah Agonist Peptides of Basic Fibroblast Growth Factor (bFGF) and the Method of Reduction of Wrinkles on Skin, Darkening of Hair and Acceleration of Wound Healing
US7601361B2 (en) * 2005-10-03 2009-10-13 E. I. Du Pont De Nemours And Company Process for providing antimicrobial surfaces
WO2007044998A1 (en) * 2005-10-12 2007-04-19 The Regents Of The University Of California Retrocyclins: antiviral and antimicrobial peptides
US20070197445A1 (en) * 2006-01-18 2007-08-23 University Of Cincinnati Compounds for control of appetite
MX2008009654A (es) * 2006-01-24 2009-01-15 Univ British Columbia Polimorfismos de vias de vasopresina como indicadores del resultado expuesto en sujetos criticamente enfermos.
KR101433962B1 (ko) 2006-03-10 2014-08-25 라보스위스 아게 물질의 용해, 분산 및 안정을 위한 방법, 상기 방법에 따라제조된 제품 및 상기 제품의 이용
EP2015765A4 (en) * 2006-03-28 2011-11-23 Neopro Labs Llc METHODS AND COMPOSITIONS FOR TREATING CONDITIONS
US20070238661A1 (en) * 2006-04-11 2007-10-11 Witten Mark L Substance P treatment for hepatitis C
WO2007134151A2 (en) * 2006-05-10 2007-11-22 Smithkline Beecham Corporation Composition and method for increasing cell permeability of a compound
WO2008052043A2 (en) * 2006-10-24 2008-05-02 Cogenesys, Inc. Opioid receptor agonist fusion proteins
CN101795675A (zh) * 2006-11-17 2010-08-04 达沃尔泰拉公司 使用具有Eudragit包衣的Zn/果胶珠粒进行的结肠递送

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2528094C2 (ru) * 2012-08-03 2014-09-10 Татьяна Георгиевна Емельянова Средство пептидной структуры, обладающее анальгетическим, противовоспалительным действием, и лекарственные формы на его основе

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