RU2010113997A - Тиролиберин для терапевтического применения - Google Patents
Тиролиберин для терапевтического применения Download PDFInfo
- Publication number
- RU2010113997A RU2010113997A RU2010113997/15A RU2010113997A RU2010113997A RU 2010113997 A RU2010113997 A RU 2010113997A RU 2010113997/15 A RU2010113997/15 A RU 2010113997/15A RU 2010113997 A RU2010113997 A RU 2010113997A RU 2010113997 A RU2010113997 A RU 2010113997A
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- Russia
- Prior art keywords
- diseases
- disease
- pharmaceutical composition
- peptide
- fibrosis
- Prior art date
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- XNSAINXGIQZQOO-SRVKXCTJSA-N protirelin Chemical compound NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H]1NC(=O)CC1)CC1=CN=CN1 XNSAINXGIQZQOO-SRVKXCTJSA-N 0.000 title claims abstract 5
- 102400000336 Thyrotropin-releasing hormone Human genes 0.000 title 1
- 101800004623 Thyrotropin-releasing hormone Proteins 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 claims abstract 10
- 108090000765 processed proteins & peptides Proteins 0.000 claims abstract 10
- 239000000203 mixture Substances 0.000 claims abstract 7
- 208000023275 Autoimmune disease Diseases 0.000 claims abstract 5
- 208000035473 Communicable disease Diseases 0.000 claims abstract 5
- 206010016654 Fibrosis Diseases 0.000 claims abstract 5
- 208000019693 Lung disease Diseases 0.000 claims abstract 5
- 201000011510 cancer Diseases 0.000 claims abstract 5
- 230000004761 fibrosis Effects 0.000 claims abstract 5
- 208000019622 heart disease Diseases 0.000 claims abstract 5
- 208000027866 inflammatory disease Diseases 0.000 claims abstract 5
- 230000030833 cell death Effects 0.000 claims abstract 4
- 239000007788 liquid Substances 0.000 claims abstract 4
- 238000011282 treatment Methods 0.000 claims abstract 3
- 208000019553 vascular disease Diseases 0.000 claims abstract 3
- 208000030507 AIDS Diseases 0.000 claims abstract 2
- 208000003918 Acute Kidney Tubular Necrosis Diseases 0.000 claims abstract 2
- 208000007788 Acute Liver Failure Diseases 0.000 claims abstract 2
- 206010000804 Acute hepatic failure Diseases 0.000 claims abstract 2
- 208000024827 Alzheimer disease Diseases 0.000 claims abstract 2
- 208000032467 Aplastic anaemia Diseases 0.000 claims abstract 2
- 208000026372 Congenital cystic kidney disease Diseases 0.000 claims abstract 2
- 206010025327 Lymphopenia Diseases 0.000 claims abstract 2
- 201000003793 Myelodysplastic syndrome Diseases 0.000 claims abstract 2
- 206010038540 Renal tubular necrosis Diseases 0.000 claims abstract 2
- 208000007014 Retinitis pigmentosa Diseases 0.000 claims abstract 2
- 241000193998 Streptococcus pneumoniae Species 0.000 claims abstract 2
- 208000006011 Stroke Diseases 0.000 claims abstract 2
- 210000001744 T-lymphocyte Anatomy 0.000 claims abstract 2
- 231100000836 acute liver failure Toxicity 0.000 claims abstract 2
- 206010002026 amyotrophic lateral sclerosis Diseases 0.000 claims abstract 2
- 210000004204 blood vessel Anatomy 0.000 claims abstract 2
- 239000000872 buffer Substances 0.000 claims abstract 2
- 239000007853 buffer solution Substances 0.000 claims abstract 2
- 239000002577 cryoprotective agent Substances 0.000 claims abstract 2
- 230000007812 deficiency Effects 0.000 claims abstract 2
- 239000003085 diluting agent Substances 0.000 claims abstract 2
- 239000003937 drug carrier Substances 0.000 claims abstract 2
- 206010015037 epilepsy Diseases 0.000 claims abstract 2
- 210000002919 epithelial cell Anatomy 0.000 claims abstract 2
- 102000010705 glucose-6-phosphate dehydrogenase activity proteins Human genes 0.000 claims abstract 2
- 108040005050 glucose-6-phosphate dehydrogenase activity proteins Proteins 0.000 claims abstract 2
- 208000015181 infectious disease Diseases 0.000 claims abstract 2
- 208000000509 infertility Diseases 0.000 claims abstract 2
- 230000036512 infertility Effects 0.000 claims abstract 2
- 231100000535 infertility Toxicity 0.000 claims abstract 2
- 238000001990 intravenous administration Methods 0.000 claims abstract 2
- 230000000302 ischemic effect Effects 0.000 claims abstract 2
- 210000003734 kidney Anatomy 0.000 claims abstract 2
- -1 lyoprotector Substances 0.000 claims abstract 2
- 238000004519 manufacturing process Methods 0.000 claims abstract 2
- 208000010125 myocardial infarction Diseases 0.000 claims abstract 2
- 239000000546 pharmaceutical excipient Substances 0.000 claims abstract 2
- 208000030761 polycystic kidney disease Diseases 0.000 claims abstract 2
- 238000011321 prophylaxis Methods 0.000 claims abstract 2
- 229940031000 streptococcus pneumoniae Drugs 0.000 claims abstract 2
- 241000712461 unidentified influenza virus Species 0.000 claims abstract 2
- 210000004251 human milk Anatomy 0.000 claims 2
- 235000020256 human milk Nutrition 0.000 claims 2
- 230000002265 prevention Effects 0.000 claims 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
-
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/095—Oxytocins; Vasopressins; Related peptides
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23C—DAIRY PRODUCTS, e.g. MILK, BUTTER OR CHEESE; MILK OR CHEESE SUBSTITUTES; MAKING THEREOF
- A23C9/00—Milk preparations; Milk powder or milk powder preparations
- A23C9/152—Milk preparations; Milk powder or milk powder preparations containing additives
- A23C9/1526—Amino acids; Peptides; Protein hydrolysates; Nucleic acids; Derivatives thereof
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- A23L—FOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
- A23L33/00—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
- A23L33/40—Complete food formulations for specific consumer groups or specific purposes, e.g. infant formula
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- A61K9/08—Solutions
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
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Abstract
1. Применение пептида Pyr-His-Pro-NH2 для получения фармацевтической композиции для лечения и/или профилактики злокачественной опухоли, аутоиммунных заболеваний, фиброзов, воспалительных заболеваний, инфекционных заболеваний, заболеваний легких, заболеваний сердца и сосудов. ! 2. Применение пептида по п.1, где злокачественная опухоль, аутоиммунное заболевание, фиброз, воспалительное заболевание, инфекционное заболевание, заболевание легких, заболевание сердца и сосудов выбраны из СПИДа, болезни Альцгеймера, бокового амиотрофического склероза, ишемического повреждения почки, пигментного ретинита, эпилепсии, апластической анемии, миелодиспластического синдрома, CD4+ T-клеточной лимфоцитопении, дефицита Г6ФДГ, инфаркта миокарда, инсульта, поликистозной почки, острой печеночной недостаточности, острого тубулярного некроза, бесплодия, индуцированной Streptococcus pneumoniae гибели эпителиальных клеток и индуцированной вирусом гриппа гибели клеток. ! 3. Применение пептида по п.1 или 2 для получения состава для перорального введения новорожденным, детям ясельного возраста и/или детям дошкольного возраста. ! 4. Применение пептида по п.1 или 2 для получения лиофилизированного состава или буферного жидкого состава. ! 5. Фармацевтическая композиция, содержащая пептид Pyr-His-Pro-NH2, по меньшей мере, совместно с одним фармацевтически приемлемым носителем, криопротектором, лиопротектором, эксципиентом и/или разбавителем. ! 6. Фармацевтическая композиция по п.5 в форме лиофилизата или жидкого буферного раствора. ! 7. Фармацевтическая композиция по п.5 или 6, пригодная для внутривенного введения, перорального введения или для введения посредство
Claims (9)
1. Применение пептида Pyr-His-Pro-NH2 для получения фармацевтической композиции для лечения и/или профилактики злокачественной опухоли, аутоиммунных заболеваний, фиброзов, воспалительных заболеваний, инфекционных заболеваний, заболеваний легких, заболеваний сердца и сосудов.
2. Применение пептида по п.1, где злокачественная опухоль, аутоиммунное заболевание, фиброз, воспалительное заболевание, инфекционное заболевание, заболевание легких, заболевание сердца и сосудов выбраны из СПИДа, болезни Альцгеймера, бокового амиотрофического склероза, ишемического повреждения почки, пигментного ретинита, эпилепсии, апластической анемии, миелодиспластического синдрома, CD4+ T-клеточной лимфоцитопении, дефицита Г6ФДГ, инфаркта миокарда, инсульта, поликистозной почки, острой печеночной недостаточности, острого тубулярного некроза, бесплодия, индуцированной Streptococcus pneumoniae гибели эпителиальных клеток и индуцированной вирусом гриппа гибели клеток.
3. Применение пептида по п.1 или 2 для получения состава для перорального введения новорожденным, детям ясельного возраста и/или детям дошкольного возраста.
4. Применение пептида по п.1 или 2 для получения лиофилизированного состава или буферного жидкого состава.
5. Фармацевтическая композиция, содержащая пептид Pyr-His-Pro-NH2, по меньшей мере, совместно с одним фармацевтически приемлемым носителем, криопротектором, лиопротектором, эксципиентом и/или разбавителем.
6. Фармацевтическая композиция по п.5 в форме лиофилизата или жидкого буферного раствора.
7. Фармацевтическая композиция по п.5 или 6, пригодная для внутривенного введения, перорального введения или для введения посредством ингаляции.
8. Фармацевтическая композиция по п.5 или 6 в форме состава искусственного материнского молока или заменителя материнского молока, пригодная для пероральной доставки новорожденным, детям ясельного возраста и/или детям дошкольного возраста.
9. Фармацевтическая композиция по п.5 или 6, пригодная для лечения и/или профилактики злокачественной опухоли, аутоиммунного заболевания, фиброза, воспалительного заболевания, инфекционного заболевания, заболевания легких, заболевания сердца и сосудов.
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RU2010114044/15A RU2010114044A (ru) | 2007-09-11 | 2008-09-09 | Применение белка полосы 3 (824-829) и/или фактора ингибирования высвобождения меланотропина в качестве терапевтического средства при лечении инфекции pseudomonas aeruginosa |
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