RS67304A - Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles - Google Patents

Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles

Info

Publication number
RS67304A
RS67304A YU67304A YUP67304A RS67304A RS 67304 A RS67304 A RS 67304A YU 67304 A YU67304 A YU 67304A YU P67304 A YUP67304 A YU P67304A RS 67304 A RS67304 A RS 67304A
Authority
RS
Serbia
Prior art keywords
solid amorphous
dried solid
pressure nozzles
amorphous drug
homogeneous spray
Prior art date
Application number
YU67304A
Other languages
English (en)
Inventor
Ronald Arthur Beyerinck
Roderick Jack Ray
Daniel Elmont Dobry
Dana Marie Settell
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27663274&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS67304(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of RS67304A publication Critical patent/RS67304A/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
  • Vaporization, Distillation, Condensation, Sublimation, And Cold Traps (AREA)
  • Glanulating (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)
  • Disintegrating Or Milling (AREA)

Abstract

Homogene čvrste amorfne disperzije leka u polimerima koji povećavaju rastvorljivost su stvorene u željenim većim veličinama čestica sa minimumom sitnozrnih čestica upotrebom raspršivača i uslova sposobnih da proizvedu kapljice koje imaju srednji prečnik od najmanje 50 mikrona i D10 od najmanje 10 mikrona.
YU67304A 2002-02-01 2003-01-20 Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles RS67304A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35398602P 2002-02-01 2002-02-01
PCT/IB2003/000120 WO2003063821A2 (en) 2002-02-01 2003-01-20 Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles

Publications (1)

Publication Number Publication Date
RS67304A true RS67304A (en) 2006-10-27

Family

ID=27663274

Family Applications (1)

Application Number Title Priority Date Filing Date
YU67304A RS67304A (en) 2002-02-01 2003-01-20 Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles

Country Status (20)

Country Link
US (1) US7780988B2 (sr)
EP (1) EP1469830A2 (sr)
JP (1) JP2005523260A (sr)
KR (1) KR100758045B1 (sr)
CN (1) CN1787808A (sr)
AR (1) AR038369A1 (sr)
AU (1) AU2003239463B2 (sr)
BR (1) BR0307515A (sr)
CA (1) CA2474958A1 (sr)
GT (1) GT200300024A (sr)
MX (1) MXPA04007435A (sr)
PA (1) PA8565401A1 (sr)
PE (1) PE20030804A1 (sr)
PL (1) PL371593A1 (sr)
RS (1) RS67304A (sr)
RU (1) RU2288703C2 (sr)
TW (1) TW200404576A (sr)
UY (1) UY27645A1 (sr)
WO (1) WO2003063821A2 (sr)
ZA (1) ZA200405971B (sr)

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Also Published As

Publication number Publication date
PL371593A1 (en) 2005-06-27
PA8565401A1 (es) 2003-12-10
US7780988B2 (en) 2010-08-24
EP1469830A2 (en) 2004-10-27
RU2004123639A (ru) 2005-04-20
ZA200405971B (en) 2006-05-31
AU2003239463B2 (en) 2007-10-18
US20030185893A1 (en) 2003-10-02
TW200404576A (en) 2004-04-01
RU2288703C2 (ru) 2006-12-10
KR20040083491A (ko) 2004-10-02
AR038369A1 (es) 2005-01-12
WO2003063821A2 (en) 2003-08-07
WO2003063821A3 (en) 2003-11-13
CN1787808A (zh) 2006-06-14
KR100758045B1 (ko) 2007-09-11
JP2005523260A (ja) 2005-08-04
BR0307515A (pt) 2004-12-07
GT200300024A (es) 2003-09-22
PE20030804A1 (es) 2003-09-19
CA2474958A1 (en) 2003-08-07
MXPA04007435A (es) 2004-10-11
UY27645A1 (es) 2003-09-30

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