RS62357B1 - Dobijanje derivata 2-([1,2,3]triazol-2-il)-benzojeve kiseline - Google Patents

Dobijanje derivata 2-([1,2,3]triazol-2-il)-benzojeve kiseline

Info

Publication number
RS62357B1
RS62357B1 RS20211164A RSP20211164A RS62357B1 RS 62357 B1 RS62357 B1 RS 62357B1 RS 20211164 A RS20211164 A RS 20211164A RS P20211164 A RSP20211164 A RS P20211164A RS 62357 B1 RS62357 B1 RS 62357B1
Authority
RS
Serbia
Prior art keywords
triazol
preparation
benzoic acid
acid derivatives
derivatives
Prior art date
Application number
RS20211164A
Other languages
English (en)
Inventor
Patric Dörrwächter
Gunther Schmidt
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Publication of RS62357B1 publication Critical patent/RS62357B1/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C07D249/061,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J23/00Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
    • B01J23/70Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of the iron group metals or copper
    • B01J23/72Copper
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
RS20211164A 2017-05-03 2018-05-02 Dobijanje derivata 2-([1,2,3]triazol-2-il)-benzojeve kiseline RS62357B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP2017060451 2017-05-03
EP18722948.9A EP3619199B1 (en) 2017-05-03 2018-05-02 Preparation of 2-([1,2,3]triazol-2-yl)-benzoic acid derivatives
PCT/EP2018/061172 WO2018202689A1 (en) 2017-05-03 2018-05-02 Preparation of 2-([1,2,3]triazol-2-yl)-benzoic acid derivatives

Publications (1)

Publication Number Publication Date
RS62357B1 true RS62357B1 (sr) 2021-10-29

Family

ID=62116854

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20211164A RS62357B1 (sr) 2017-05-03 2018-05-02 Dobijanje derivata 2-([1,2,3]triazol-2-il)-benzojeve kiseline

Country Status (20)

Country Link
US (1) US11124488B2 (sr)
EP (1) EP3619199B1 (sr)
JP (1) JP7182562B2 (sr)
KR (1) KR102582197B1 (sr)
CN (1) CN110612291B (sr)
CA (1) CA3059394C (sr)
CY (1) CY1124777T1 (sr)
DK (1) DK3619199T3 (sr)
ES (1) ES2892161T3 (sr)
HR (1) HRP20211304T1 (sr)
HU (1) HUE055904T2 (sr)
IL (1) IL270274B (sr)
LT (1) LT3619199T (sr)
MX (1) MX2019012902A (sr)
PL (1) PL3619199T3 (sr)
PT (1) PT3619199T (sr)
RS (1) RS62357B1 (sr)
SI (1) SI3619199T1 (sr)
TW (1) TWI756418B (sr)
WO (1) WO2018202689A1 (sr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4138822A1 (en) 2020-04-19 2023-03-01 Idorsia Pharmaceuticals Ltd Medical use of daridorexant
TW202400149A (zh) 2022-05-13 2024-01-01 瑞士商愛杜西亞製藥有限公司 經噻唑并芳基-甲基取代之環狀肼-n-甲醯胺衍生物

Family Cites Families (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7994336B2 (en) 2006-08-15 2011-08-09 Actelion Pharmaceuticals Ltd. Azetidine compounds as orexin receptor antagonists
WO2008038251A2 (en) 2006-09-29 2008-04-03 Actelion Pharmaceuticals Ltd 3-aza-bicyclo[3.1.0]hexane derivatives
PE20081229A1 (es) * 2006-12-01 2008-08-28 Merck & Co Inc Antagonistas de receptor de orexina de diazepam sustituido
TW200833328A (en) 2006-12-28 2008-08-16 Actelion Pharmaceuticals Ltd 2-aza-bicyclo[3.1.0]hexane derivatives
JP2010526869A (ja) 2007-05-14 2010-08-05 アクテリオン ファーマシューティカルズ リミテッド 2−シクロプロピル−チアゾール誘導体
WO2008150364A1 (en) 2007-05-23 2008-12-11 Merck & Co., Inc. Cyclopropyl pyrrolidine orexin receptor antagonists
JP5759470B2 (ja) 2009-10-23 2015-08-05 ヤンセン ファーマシューティカ エヌ.ベー. オレキシン受容体調節因子としての二置換オクタヒドロピロロ[3,4−c]ピロール
JP5848251B2 (ja) 2009-10-23 2016-01-27 ヤンセン ファーマシューティカ エヌ.ベー. オレキシン受容体調節因子としての縮合複素環式化合物
US8680275B2 (en) 2009-10-23 2014-03-25 Janssen Pharmaceutica Nv Fused heterocyclic compounds as orexin receptor modulators
NZ611865A (en) 2010-12-17 2014-11-28 Taisho Pharmaceutical Co Ltd Pyrazole derivative
WO2012085857A1 (en) 2010-12-22 2012-06-28 Actelion Pharmaceuticals Ltd 3,8-diaza-bicyclo[4.2.0]oct-3-yl amides
US9108959B2 (en) 2011-03-03 2015-08-18 Merck Sharp & Dohme Corp. Process for the preparation of an orexin receptor antagonist
US9586962B2 (en) 2011-04-20 2017-03-07 Janssen Pharmaceutica Nv Disubstituted octahydropyrrolo [3,4-C] pyrroles as orexin receptor modulators
WO2013005755A1 (ja) 2011-07-05 2013-01-10 大正製薬株式会社 メチルピペリジン誘導体
WO2013050938A1 (en) * 2011-10-04 2013-04-11 Actelion Pharmaceuticals Ltd 3,7-diazabicyclo[3.3.1]nonane and 9-oxa-3,7-diazabicyclo[3.3.1]nonane derivatives
TWI565703B (zh) 2011-11-08 2017-01-11 艾克泰聯製藥有限公司 2-(1,2,3-三唑-2-基)苯甲醯胺及3-(1,2,3-三唑-2-基)吡啶醯胺衍生物
WO2013169610A1 (en) 2012-05-09 2013-11-14 Merck Sharp & Dohme Corp. Process for the preparation of an intermediate for an orexin receptor antagonist
EP2855453B1 (en) 2012-06-04 2016-12-07 Actelion Pharmaceuticals Ltd. Benzimidazole-proline derivatives
JP2014015452A (ja) 2012-06-15 2014-01-30 Taisho Pharmaceutical Co Ltd ピラゾール誘導体を含有する医薬
CN104703980B (zh) * 2012-10-10 2017-09-22 埃科特莱茵药品有限公司 属于[邻双(杂)芳基]‑[2‑(间双(杂)芳基)吡咯烷‑1‑基]甲酮衍生物的食欲素受体拮抗剂
KR20150130413A (ko) 2013-03-12 2015-11-23 액테리온 파마슈티칼 리미티드 오렉신 수용체 길항제로서의 아제티딘 아미드 유도체
TW201444849A (zh) * 2013-03-13 2014-12-01 Janssen Pharmaceutica Nv 經取代的7-氮雜雙環類及其作為食慾激素受體調節劑之用途
TW201444821A (zh) 2013-03-13 2014-12-01 Janssen Pharmaceutica Nv 經取代之哌啶化合物及其作為食慾素受體調節劑之用途
UA119151C2 (uk) 2013-12-03 2019-05-10 Ідорсія Фармасьютікалз Лтд КРИСТАЛІЧНА СОЛЬОВА ФОРМА (S)-(2-(6-ХЛОР-7-МЕТИЛ-1H-БЕНЗО[d]ІМІДАЗОЛ-2-ІЛ)-2-МЕТИЛПІРОЛІДИН-1-ІЛ)(5-МЕТОКСИ-2-(2H-1,2,3-ТРИАЗОЛ-2-ІЛ)ФЕНІЛ)МЕТАНОНУ ЯК АНТАГОНІСТ ОРЕКСИНОВОГО РЕЦЕПТОРА
PT3077389T (pt) * 2013-12-03 2017-12-15 Idorsia Pharmaceuticals Ltd Forma cristalina de (s)-(2-(6-cloro-7-metil-1hbenzo[d]imidazol-2-il)-2-metilpirrolidin-1-il)(5-metoxi-2-(2h-1,2,3-triazol-2-il)fenil)metanona e a sua utilização como como antagonistas do receptor de orexina
LT3077391T (lt) 2013-12-04 2018-10-25 Idorsia Pharmaceuticals Ltd Benzimidazolo prolino darinių panaudojimas
UY35993A (es) * 2014-02-12 2015-08-31 Eolas Therapeutics Inc Prolinas / piperidinas sustituidas como antagonistas del receptor de orexina
WO2016020403A1 (en) 2014-08-04 2016-02-11 Sandoz Ag Preparation of a benzoic acid derivative and its use for the preparation of suvorexant
CN104649983B (zh) * 2014-12-23 2018-01-23 广东东阳光药业有限公司 一种酸的制备方法
US10131653B2 (en) * 2015-04-24 2018-11-20 Takeda Pharmaceutical Company Limited Heterocyclic compound

Also Published As

Publication number Publication date
PT3619199T (pt) 2021-10-01
HUE055904T2 (hu) 2021-12-28
PL3619199T3 (pl) 2021-12-20
CA3059394C (en) 2023-09-12
WO2018202689A1 (en) 2018-11-08
IL270274B (en) 2022-08-01
JP2020518573A (ja) 2020-06-25
CA3059394A1 (en) 2018-11-08
US20210114997A1 (en) 2021-04-22
JP7182562B2 (ja) 2022-12-02
HRP20211304T1 (hr) 2021-11-12
EP3619199B1 (en) 2021-07-07
ES2892161T3 (es) 2022-02-02
TW201843144A (zh) 2018-12-16
SI3619199T1 (sl) 2021-11-30
CN110612291A (zh) 2019-12-24
CN110612291B (zh) 2024-02-13
DK3619199T3 (da) 2021-09-27
TWI756418B (zh) 2022-03-01
IL270274A (sr) 2019-12-31
MX2019012902A (es) 2019-12-16
LT3619199T (lt) 2021-09-27
KR102582197B1 (ko) 2023-09-22
CY1124777T1 (el) 2022-11-25
KR20200003097A (ko) 2020-01-08
US11124488B2 (en) 2021-09-21
EP3619199A1 (en) 2020-03-11

Similar Documents

Publication Publication Date Title
EP3402787A4 (en) PROCESSES FOR PREPARING 2,5-FURANDICARBOXYLIC ACID AND INTERMEDIATES AND DERIVATIVES THEREOF
PL3283470T3 (pl) Sposoby wytwarzania kwasu 2,5-furanodikarboksylowego i jego pochodnych
HK1254055A1 (zh) 製備奧貝膽酸及其衍生物的方法
IL260011A (en) History of 5,3-diphenyl-diazole water-soluble compounds
IL271399A (en) Methods for the preparation of heterocyclic 3,1-benzodioxole compounds
EP3384772A4 (en) AGROCHEMICAL COMPOSITION IN AQUEOUS SUSPENSION
EP3315492A4 (en) Pyrazole derivative, or pharmaceutically acceptable salt thereof
EP3490978A4 (en) SALTS OF 2, 6-DIMETHYLPYRIMIDONE DERIVATIVES AND THEIR USES
IL262405A (en) Methods for the preparation of obeticholic acid and derivatives thereof
EP3442943A4 (en) AMINOBENZOIC ACID DERIVATIVES FOR USE AS ANTI-INFLAMMATORY AGENTS, ANTI-METASTATIC AGENTS AND / OR ANTICANCER AGENTS
MX2020012771A (es) Metodos para preparar 5,6-dihidro-6-fenilbenzo[f]isoquinolin-2-ami na sustituida.
PL3619199T3 (pl) Wytwarzanie pochodnych kwasu 2-([1,2,3]triazol-2-ilo)­-benzoesowego
HK1256825A1 (zh) 取代的5,6-二氫-6-苯基苯並[f]異喹啉-2-胺化合物的固體形式
EP3530654A4 (en) CARBOXYLIC ACID COMPOUND WITH QUINOLINYL SUBSTITUTE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PHARMACEUTICAL COMPOSITION AND USE THEREOF
EP3189842A4 (en) Composition for preventing hair loss or promoting hair growth, containing oleanolic acid derivative and pharmaceutically acceptable salt thereof
HK1258757A1 (zh) 4H-吡唑並[1,5-α]苯並咪唑類化合物的鹽型、晶型及其製備方法和中間體
EP3699250A4 (en) COMPOSITION PROVIDING A FRESHNESS FEELING CONTAINING A DERIVATIVE OF 2,2,6-TRIMETHYLCYLCYCLOHEXANECARBOXYLIC ACID
IL254578A0 (en) Abscisic acid (s)-2' vinyl derivatives
EP3398946A4 (en) SALT OF MORPHOLINE DERIVATIVE AND ITS CRYSTALLINE FORM, AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF
EP3436439A4 (en) METHOD FOR PRODUCING DIPHENYLPYRAZINE DERIVATIVES
EP3166405A4 (en) 3'-substituted-abscisic acid derivatives
EP3856732C0 (en) PROCESS AND SALTS FOR THE PREPARATION OF 2,5-FURANEDICARBOXYLIC ACID
EP3177592A4 (en) Process for the preparation of 4,5,6-trichloropicolinic acid
IL257438B (en) An improved process for the preparation of tetraforsamine or its acid salt
HUP1500451A2 (en) Processes for the preparation of 1,4,7-triaza-cyclononane derivatives and intermediates