RS50868B - Stereoselektivni postupak za dobijanje nukleozidnih analoga - Google Patents

Stereoselektivni postupak za dobijanje nukleozidnih analoga

Info

Publication number
RS50868B
RS50868B YUP-975/03A YUP97503A RS50868B RS 50868 B RS50868 B RS 50868B YU P97503 A YUP97503 A YU P97503A RS 50868 B RS50868 B RS 50868B
Authority
RS
Serbia
Prior art keywords
alkyl
optionally substituted
formula
fluoro
bromo
Prior art date
Application number
YUP-975/03A
Other languages
English (en)
Serbian (sr)
Inventor
Qing Yu
Original Assignee
Shire Canada Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shire Canada Inc. filed Critical Shire Canada Inc.
Publication of YU97503A publication Critical patent/YU97503A/sh
Publication of RS50868B publication Critical patent/RS50868B/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D327/00Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/04Five-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D411/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
YUP-975/03A 2001-06-15 2002-06-14 Stereoselektivni postupak za dobijanje nukleozidnih analoga RS50868B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29807901P 2001-06-15 2001-06-15

Publications (2)

Publication Number Publication Date
YU97503A YU97503A (sh) 2006-05-25
RS50868B true RS50868B (sr) 2010-08-31

Family

ID=23148927

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-975/03A RS50868B (sr) 2001-06-15 2002-06-14 Stereoselektivni postupak za dobijanje nukleozidnih analoga

Country Status (28)

Country Link
US (2) US7109334B2 (enExample)
EP (2) EP1632490B1 (enExample)
JP (1) JP4542776B2 (enExample)
KR (1) KR100832617B1 (enExample)
CN (1) CN1297553C (enExample)
AP (1) AP1559A (enExample)
AT (2) ATE313542T1 (enExample)
AU (2) AU2002344862C1 (enExample)
BR (2) BR0210444A (enExample)
CA (1) CA2449338C (enExample)
CO (1) CO5550497A2 (enExample)
CY (1) CY1107805T1 (enExample)
DE (2) DE60222031T2 (enExample)
DK (2) DK1632490T3 (enExample)
EA (1) EA006372B1 (enExample)
ES (2) ES2293445T3 (enExample)
HR (1) HRP20031021B1 (enExample)
IL (2) IL159139A0 (enExample)
MX (1) MXPA03011627A (enExample)
NO (1) NO326135B1 (enExample)
NZ (1) NZ529906A (enExample)
OA (1) OA12628A (enExample)
PL (2) PL215267B1 (enExample)
PT (1) PT1632490E (enExample)
RS (1) RS50868B (enExample)
SI (2) SI1406896T1 (enExample)
WO (1) WO2002102796A1 (enExample)
ZA (1) ZA200309307B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7501514B1 (en) 2003-10-15 2009-03-10 Shire Biochem, Inc. Enantiomeric resolution of 2-substituted 4-substituted 1,3-oxathiolanes nucleosides
JP4653966B2 (ja) * 2004-04-19 2011-03-16 ダイセル化学工業株式会社 2−ベンゾイルオキシアセトアルデヒド誘導体の製造法
WO2009039582A1 (en) * 2007-09-28 2009-04-02 Avexa Limited A process for chiral resolution of 2-substituted 4-substituted 1,3-oxathiolanes
US20130165350A1 (en) * 2011-12-22 2013-06-27 Affymetrix, Inc. Surface linkers for array synthesis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR840001591A (ko) * 1981-09-29 1984-05-07 구라바야시 이꾸시로 당케탈류의 제조방법
US5587480A (en) * 1990-11-13 1996-12-24 Biochem Pharma, Inc. Substituted 1,3-oxathiolanes and substituted 1,3-dithiolanes with antiviral properties
ATE143016T1 (de) * 1990-11-13 1996-10-15 Iaf Biochem Int Substituierte 1,3-oxathiolane mit antiviralen eigenschaften
US5532349A (en) * 1993-07-20 1996-07-02 Mitsui Toatsu Chemicals, Inc. Process for producing 1-(2'-deoxy-β-D-erythro-pentofuranosyl)-5-trifluoromethyluracil derivatives
ES2232169T3 (es) * 1998-08-12 2005-05-16 Gilead Sciences, Inc. Procedimiento de fabricacion de nucleosidos de 1,3-oxatiolano.

Also Published As

Publication number Publication date
NZ529906A (en) 2006-03-31
DE60208202T2 (de) 2006-08-17
DK1632490T3 (da) 2008-01-28
DE60222031D1 (de) 2007-10-04
SI1406896T1 (sl) 2006-04-30
AU2002344862B2 (en) 2008-05-01
EA200400042A1 (ru) 2004-06-24
KR100832617B1 (ko) 2008-05-27
HK1070652A1 (en) 2005-06-24
KR20040017233A (ko) 2004-02-26
CO5550497A2 (es) 2005-08-31
ATE370945T1 (de) 2007-09-15
JP2004535428A (ja) 2004-11-25
HRP20031021A2 (en) 2004-06-30
WO2002102796A8 (en) 2003-09-18
PL218777B1 (pl) 2015-01-30
WO2002102796A1 (en) 2002-12-27
PL366907A1 (en) 2005-02-07
US20060183899A1 (en) 2006-08-17
HRP20031021B1 (hr) 2007-09-30
IL159139A (en) 2010-04-15
BR0210444A (pt) 2004-08-17
NO20035556D0 (no) 2003-12-12
BRPI0210444B1 (pt) 2017-06-20
NO326135B1 (no) 2008-10-06
JP4542776B2 (ja) 2010-09-15
CN1297553C (zh) 2007-01-31
AP1559A (en) 2006-01-24
YU97503A (sh) 2006-05-25
CA2449338A1 (en) 2002-12-27
SI1632490T1 (sl) 2008-02-29
PT1632490E (pt) 2007-11-07
DE60208202D1 (de) 2006-01-26
EP1632490B1 (en) 2007-08-22
EP1406896A1 (en) 2004-04-14
ZA200309307B (en) 2005-02-23
EP1406896B1 (en) 2005-12-21
PL215267B1 (pl) 2013-11-29
US7109334B2 (en) 2006-09-19
US7230100B2 (en) 2007-06-12
ES2293445T3 (es) 2008-03-16
ATE313542T1 (de) 2006-01-15
DK1406896T3 (da) 2006-05-08
US20030135048A1 (en) 2003-07-17
CA2449338C (en) 2012-02-07
OA12628A (en) 2006-06-13
CN1543463A (zh) 2004-11-03
EP1406896B8 (en) 2006-11-15
MXPA03011627A (es) 2005-03-07
IL159139A0 (en) 2004-06-01
AU2008203443B2 (en) 2011-06-16
EP1632490A1 (en) 2006-03-08
DE60222031T2 (de) 2008-05-21
EA006372B1 (ru) 2005-12-29
PL401835A1 (pl) 2013-02-18
CY1107805T1 (el) 2013-06-19
AU2002344862C1 (en) 2009-02-19
AU2008203443A1 (en) 2008-08-21
ES2254695T3 (es) 2006-06-16

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