PT782997E - Derivados de triazolopirimidina - Google Patents

Derivados de triazolopirimidina Download PDF

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Publication number
PT782997E
PT782997E PT97105710T PT97105710T PT782997E PT 782997 E PT782997 E PT 782997E PT 97105710 T PT97105710 T PT 97105710T PT 97105710 T PT97105710 T PT 97105710T PT 782997 E PT782997 E PT 782997E
Authority
PT
Portugal
Prior art keywords
triazolo
dichloro
pyrimidine
phenyl
fluorophenyl
Prior art date
Application number
PT97105710T
Other languages
English (en)
Portuguese (pt)
Inventor
Guido Albert
Klaus-Jurgen Pees
Original Assignee
Shell Int Research
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shell Int Research filed Critical Shell Int Research
Publication of PT782997E publication Critical patent/PT782997E/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT97105710T 1991-12-30 1992-12-28 Derivados de triazolopirimidina PT782997E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP91122422 1991-12-30

Publications (1)

Publication Number Publication Date
PT782997E true PT782997E (pt) 2000-09-29

Family

ID=8207489

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97105710T PT782997E (pt) 1991-12-30 1992-12-28 Derivados de triazolopirimidina

Country Status (21)

Country Link
EP (2) EP0550113B1 (Direct)
JP (1) JP3347170B2 (Direct)
KR (1) KR100271913B1 (Direct)
CN (2) CN1033643C (Direct)
AT (2) ATE159256T1 (Direct)
AU (1) AU667204B2 (Direct)
BR (1) BR9205172A (Direct)
CA (1) CA2086404C (Direct)
DE (2) DE69222746T2 (Direct)
DK (2) DK0782997T3 (Direct)
ES (2) ES2108727T3 (Direct)
GR (2) GR3025920T3 (Direct)
HU (1) HU217349B (Direct)
IL (1) IL104244A (Direct)
NZ (1) NZ245581A (Direct)
PL (2) PL171579B1 (Direct)
PT (1) PT782997E (Direct)
RU (1) RU2089552C1 (Direct)
SG (1) SG47563A1 (Direct)
TW (1) TW224044B (Direct)
ZA (1) ZA9210043B (Direct)

Families Citing this family (72)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5593996A (en) * 1991-12-30 1997-01-14 American Cyanamid Company Triazolopyrimidine derivatives
TW258648B (Direct) * 1993-03-04 1995-10-01 Shell Internat Res Schappej Bv
IL108747A (en) * 1993-03-04 1999-03-12 Shell Int Research Mushroom-killing preparations containing a history of 6 metamorphoses of 5 - 7 Dihalo - 1, 2 - 4 Triazlo [A-1,5] Pyrimidine Certain such new compounds and their preparation
US5869486A (en) * 1995-02-24 1999-02-09 Ono Pharmaceutical Co., Ltd. Fused pyrimidines and pyriazines as pharmaceutical compounds
RU2147584C1 (ru) 1995-10-27 2000-04-20 Американ Цианамид Компани Способ получения дигалоидазолопиримидинов и способ получения дигидроксиазолопиримидинов
US5817663A (en) * 1996-10-07 1998-10-06 American Cyanamid Company Pentafluorophenylazolopyrimidines
US5750766A (en) * 1997-03-18 1998-05-12 American Cyanamid Company Process for the preparation of arylmalonates
US5756815A (en) * 1997-03-18 1998-05-26 American Cyanamid Company Process for the preparation arylamalonates
TW460476B (en) * 1997-04-14 2001-10-21 American Cyanamid Co Fungicidal trifluoromethylalkylamino-triazolopyrimidines
US6117876A (en) * 1997-04-14 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
EP1054888B1 (en) * 1998-02-11 2003-11-26 Basf Aktiengesellschaft Fungicidal 7-alkyl-triazolopyrimidines
US6124301A (en) * 1998-03-17 2000-09-26 American Cyanamid Company Enhancement of the efficacy of triazolopyrimidines
JPH11322517A (ja) * 1998-03-17 1999-11-24 American Cyanamid Co トリアゾロピリミジン類の効力の増進
US6284762B1 (en) * 1998-03-23 2001-09-04 American Cyanamid Company Fungicidal 6-(2-halo-4-alkoxyphenyl)-triazolopyrimidines
PE20001145A1 (es) * 1998-09-10 2000-10-25 American Cyanamid Co Mezclas fungicidas
US6242451B1 (en) * 1998-09-25 2001-06-05 Klaus-Juergen Pees Fungicidal trihalophenyl-triazolopyrimidines
JP2000103790A (ja) * 1998-09-25 2000-04-11 American Cyanamid Co 殺菌・殺カビ性のトリハロフェニル―トリアゾロピリミジン類
US5986135A (en) * 1998-09-25 1999-11-16 American Cyanamid Company Fungicidal trifluoromethylalkylamino-triazolopyrimidines
US6277856B1 (en) 1998-09-25 2001-08-21 American Cynamid Co. Fungicidal mixtures
TWI229674B (en) * 1998-12-04 2005-03-21 Astra Pharma Prod Novel triazolo[4,5-d]pyrimidine compounds, pharmaceutical composition containing the same, their process for preparation and uses
CN1320880C (zh) * 1998-12-23 2007-06-13 伊迪亚股份公司 改进的体内局部无创伤用制剂
US6699874B2 (en) 1999-09-24 2004-03-02 Basf Aktiengesellschaft Fungicidal mixtures
GB2355261A (en) * 1999-10-13 2001-04-18 American Cyanamid Co Triazolopyrimidine fungicides
US6559151B2 (en) 2000-05-08 2003-05-06 Basf Aktiengesellschaft 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US6747033B2 (en) 2000-06-13 2004-06-08 Basf Aktiengesellschaft Fungicidal triazolopyrimid-7-ylideneamines
JP2004503554A (ja) * 2000-06-13 2004-02-05 ビーエーエスエフ　アクチェンゲゼルシャフト 殺菌活性を有するトリアゾロピリミド−７−イリデンアミン類
ES2223932T3 (es) * 2000-08-25 2005-03-01 Basf Aktiengesellschaft Formulacion fungicida.
ES2226968T3 (es) * 2000-12-06 2005-04-01 Wyeth 6-(2-trifluorometilfenil)-triazolopirimidinas fungicidas.
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
ATE270292T1 (de) * 2001-04-09 2004-07-15 Basf Ag Fungizide 5-alkylamino-6-phenyl-7-halogen- triazolopyrimidine
DE60201089T2 (de) 2001-04-11 2004-12-30 Basf Ag 6-(2-chlor-6-fluor-phenyl)-triazolpyrimidine
ES2236509T3 (es) 2001-04-11 2005-07-16 Basf Aktiengesellschaft 5-halogen-6-fenil-7-fluoroalquilamino-triazolopirimidinas utiles como fungicidas.
DE10121101A1 (de) 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
DE10121162A1 (de) 2001-04-30 2002-10-31 Bayer Ag Triazolopyrimidine
DE10124208A1 (de) * 2001-05-18 2002-11-21 Bayer Ag Verwendung von Triazolopyrimidin-Derivaten als Mikrobizide
BR0210858A (pt) 2001-07-05 2004-06-29 Basf Ag Composto, processo para preparar o mesmo, composição adequada para o combate de fungos danosos, uso dos compostos, e, método para combater fungos danosos
EP1412356A1 (en) * 2001-07-18 2004-04-28 Basf Aktiengesellschaft Substituted 6-(2-methoxyphenyl)triazolopyrimidines as fungicides
EP1412358A1 (en) * 2001-07-18 2004-04-28 Basf Aktiengesellschaft 6-(2,6-difluorophenyl)-triazolopyrimidines as fungicides
EA006609B1 (ru) * 2001-07-18 2006-02-24 Басф Акциенгезельшафт Замещённые 6-(2-толил)триазолопиримидины
MXPA04000403A (es) 2001-07-26 2004-03-18 Basf Ag 7 - aminotriazolopirimidinas para controlar hongos nocivos.
ES2287312T3 (es) 2001-09-04 2007-12-16 Sumitomo Chemical Company, Limited Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen.
GB0126914D0 (en) * 2001-11-08 2002-01-02 Syngenta Ltd Fungicides
PL372978A1 (en) 2002-03-21 2005-08-08 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances
DE10212886A1 (de) * 2002-03-22 2003-10-02 Bayer Cropscience Ag Triazolopyrimidine
UA80304C2 (en) 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
PL376886A1 (pl) * 2002-11-15 2006-01-09 Basf Aktiengesellschaft 2-Merkapto-podstawione triazolopirymidyny, sposoby ich wytwarzania, ich zastosowanie do zwalczania szkodliwych grzybów i zawierające je środki
WO2004055018A1 (de) * 2002-12-17 2004-07-01 Basf Aktiengesellschaft Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
EA200501388A1 (ru) * 2003-03-31 2006-02-24 Басф Акциенгезельшафт 7-алкениламинотриазолопиримидины, способ их получения и их применение для борьбы с фитопатогенными грибами, а также содержащие их средства
AU2004226253A1 (en) * 2003-04-02 2004-10-14 Basf Aktiengesellschaft 7-alkinylamino-triazolopyrimidines, methods for the production and use thereof to combat harmful fungi and agents containing said compounds
CL2004000817A1 (es) * 2003-04-17 2005-04-15 Basf Ag Compuestos biciclos que contienen n; composicion que las contiene; utiles para combatir hongos fitopatogenos.
UY28506A1 (es) * 2003-09-12 2005-04-29 Basf Ag 6-halógeno-(1,2,4)triazolo(1,5-a)pirimidinas para combatir plagas animales.
US7419982B2 (en) 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
CA2539252A1 (en) 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-[(substituted)phenyl]triazolopyrimidines as anticancer agents
ATE398452T1 (de) 2003-09-24 2008-07-15 Wyeth Corp 6-aryl-7-halo-imidazoä1,2-aüpyrimidine als mittel gegen krebs
MY179926A (en) 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
EP1697367A1 (de) * 2003-12-18 2006-09-06 Basf Aktiengesellschaft 6-(2-halogenphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bek mpfung von schadpilzen sowie sie enthaltende mittel
US20070197389A1 (en) * 2004-02-25 2007-08-23 Anja Schwogler Azolopyrimidine compounds and use thereof for combating parasitic fungi
EP1751162A1 (de) * 2004-05-17 2007-02-14 Basf Aktiengesellschaft Triazolopyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen
EP1758457A1 (de) * 2004-06-09 2007-03-07 Basf Aktiengesellschaft Triazolopyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen
KR20070029257A (ko) * 2004-06-22 2007-03-13 바스프 악티엔게젤샤프트 6-(2-톨릴)-트리아졸로피리미딘의 살진균제로서의 용도,신규 6-(2-톨릴)-트리아졸로피리미딘, 이의 제조 방법,유해 진균류 방제를 위한 이의 용도, 및 이를 함유하는제제
JP2008503512A (ja) * 2004-06-22 2008-02-07 ビーエーエスエフ　アクチェンゲゼルシャフト ６−（２−フルオロフェニル）−トリアゾロピリミジン、その生産方法、有害菌類を防除するためのその使用、およびそれを含有している薬剤
MXPA06013943A (es) * 2004-06-25 2007-03-15 Basf Ag Compuestos de triazolopirimidina y su uso en el control de hongos daninos.
JP2008505151A (ja) * 2004-07-08 2008-02-21 ビーエーエスエフ　アクチェンゲゼルシャフト 置換された６−フェニル−７−アミノトリアゾロピリミジン類、それらの生産方法、病原性真菌を抑制するためのそれらの使用、およびこれらの化合物を含有する薬剤
EA200700554A1 (ru) * 2004-09-08 2007-10-26 Басф Акциенгезельшафт 6-фенил-7-амино-триазолопиримидины, способ их получения и их применение для борьбы с патогенными грибами, а также содержащее их средство
ATE400576T1 (de) * 2005-02-16 2008-07-15 Basf Se 5-alkoxyalkyl-6-alkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
AR059649A1 (es) * 2006-02-28 2008-04-16 Basf Ag 6- fenil 7-amino - amino (1,2,4) -triazolo (1,5-a) pirimidinas y su su uso para el combate de hongos daninos
RU2325390C1 (ru) * 2007-01-29 2008-05-27 Государственное образовательное учреждение высшего профессионального образования "Южно-Российский государственный технический университет (Новочеркасский политехнический институт)" СПОСОБ ПОЛУЧЕНИЯ 2-СУЛЬФОНИЛАМИНО-1,2,4,-ТРИАЗОЛО[1,5-a] ПИРИМИДИНОВ
EP1952690A3 (en) 2007-01-31 2009-04-22 Basf Se Pesticidal mixtures based on triazolopyrimidines and insecticides
EP1952691A3 (en) 2007-01-31 2008-09-17 Basf Se Method for improving plant health by application of a triazolopyrimidine derivative
RU2460298C1 (ru) * 2011-05-03 2012-09-10 Михаил Аркадьевич Ершов Стимулятор для предпосевной обработки семян зерновых культур
RU2461197C1 (ru) * 2011-05-03 2012-09-20 Михаил Аркадьевич Ершов Стимулятор для предпосевной обработки семян зерновых культур
RU2460297C1 (ru) * 2011-05-04 2012-09-10 Михаил Аркадьевич Ершов Способ стимуляции всхожести семян

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1567021A (Direct) * 1967-01-27 1969-05-16
DE3130633A1 (de) 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
HU208693B (en) * 1991-02-22 1993-12-28 Egyt Gyogyszervegyeszeti Gyar Process for producing 1,2,4-triazolo (1,5-a) pyrimidinis derivatives and their carbicycli-tetrahydro-thiofurane-tetrahydrothiopyrane-, or tetrahydropyridine- condensated derivatives or medical preparatives containing them

Also Published As

Publication number Publication date
HU9204135D0 (en) 1993-04-28
TW224044B (Direct) 1994-05-21
EP0782997A2 (en) 1997-07-09
ZA9210043B (en) 1993-07-28
SG47563A1 (en) 1998-04-17
IL104244A (en) 1997-07-13
NZ245581A (en) 1995-07-26
CN1033643C (zh) 1996-12-25
PL171579B1 (pl) 1997-05-30
RU2089552C1 (ru) 1997-09-10
PL297160A1 (en) 1993-09-06
GR3033916T3 (en) 2000-11-30
BR9205172A (pt) 1993-07-06
JPH05271234A (ja) 1993-10-19
HK1010105A1 (en) 1999-06-11
EP0550113A2 (en) 1993-07-07
KR100271913B1 (ko) 2001-02-01
DK0550113T3 (da) 1998-02-09
CN1074650C (zh) 2001-11-14
CN1141119A (zh) 1997-01-29
DE69230977T2 (de) 2000-11-09
ATE192154T1 (de) 2000-05-15
CA2086404A1 (en) 1993-07-01
ES2147411T3 (es) 2000-09-01
JP3347170B2 (ja) 2002-11-20
AU3043592A (en) 1993-07-01
ATE159256T1 (de) 1997-11-15
DE69222746D1 (de) 1997-11-20
ES2108727T3 (es) 1998-01-01
DE69222746T2 (de) 1998-02-12
CA2086404C (en) 2003-06-10
DK0782997T3 (da) 2000-08-07
DE69230977D1 (de) 2000-05-31
HUT63305A (en) 1993-08-30
AU667204B2 (en) 1996-03-14
EP0550113B1 (en) 1997-10-15
EP0550113A3 (en) 1993-08-04
IL104244A0 (en) 1993-05-13
PL174047B1 (pl) 1998-06-30
EP0782997B1 (en) 2000-04-26
GR3025920T3 (en) 1998-04-30
EP0782997A3 (en) 1998-07-22
HU217349B (hu) 2000-01-28
CN1075144A (zh) 1993-08-11

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