PT2833864T - Formulações farmacêuticas que compreendem antagonistas de ccr3 - Google Patents

Formulações farmacêuticas que compreendem antagonistas de ccr3

Info

Publication number
PT2833864T
PT2833864T PT13714618T PT13714618T PT2833864T PT 2833864 T PT2833864 T PT 2833864T PT 13714618 T PT13714618 T PT 13714618T PT 13714618 T PT13714618 T PT 13714618T PT 2833864 T PT2833864 T PT 2833864T
Authority
PT
Portugal
Prior art keywords
pharmaceutical formulations
ccr3 antagonists
ccr3
antagonists
formulations
Prior art date
Application number
PT13714618T
Other languages
English (en)
Portuguese (pt)
Inventor
Fetscher Alfred
Matthias Scher Jochen
Original Assignee
Alkahest Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2833864(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alkahest Inc filed Critical Alkahest Inc
Publication of PT2833864T publication Critical patent/PT2833864T/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • A61K9/2022—Organic macromolecular compounds
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Transplantation (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT13714618T 2012-04-04 2013-04-02 Formulações farmacêuticas que compreendem antagonistas de ccr3 PT2833864T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04

Publications (1)

Publication Number Publication Date
PT2833864T true PT2833864T (pt) 2019-03-28

Family

ID=49292482

Family Applications (2)

Application Number Title Priority Date Filing Date
PT13714618T PT2833864T (pt) 2012-04-04 2013-04-02 Formulações farmacêuticas que compreendem antagonistas de ccr3
PT182134585T PT3524230T (pt) 2012-04-04 2013-04-02 Formulações farmacêuticas que compreendem antagonistas de ccr3

Family Applications After (1)

Application Number Title Priority Date Filing Date
PT182134585T PT3524230T (pt) 2012-04-04 2013-04-02 Formulações farmacêuticas que compreendem antagonistas de ccr3

Country Status (31)

Country Link
US (3) US10213421B2 (instruction)
EP (3) EP3970693B1 (instruction)
JP (4) JP6320990B2 (instruction)
KR (2) KR102138709B1 (instruction)
CN (1) CN104203213A (instruction)
AR (1) AR090596A1 (instruction)
AU (1) AU2013245028B2 (instruction)
BR (1) BR112014024479A8 (instruction)
CA (1) CA2869058C (instruction)
CL (1) CL2014002524A1 (instruction)
CY (1) CY1121137T1 (instruction)
DK (2) DK2833864T3 (instruction)
EA (1) EA027627B1 (instruction)
ES (2) ES2898179T3 (instruction)
HR (1) HRP20190069T1 (instruction)
HU (2) HUE056943T2 (instruction)
IL (1) IL234299A (instruction)
IN (1) IN2014DN07082A (instruction)
LT (1) LT2833864T (instruction)
MX (1) MX358307B (instruction)
NZ (1) NZ628993A (instruction)
PH (1) PH12014502241A1 (instruction)
PL (2) PL2833864T3 (instruction)
PT (2) PT2833864T (instruction)
RS (1) RS58360B1 (instruction)
SI (1) SI2833864T1 (instruction)
SM (1) SMT201900121T1 (instruction)
TR (1) TR201821285T4 (instruction)
TW (1) TW201400115A (instruction)
UY (1) UY34730A (instruction)
WO (1) WO2013149987A1 (instruction)

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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
MY199462A (en) 2017-04-05 2023-10-30 Alkahest Inc Methods and compositions for treating retina-associated disease using ccr3-inhibitors
JP2020513005A (ja) 2017-04-05 2020-04-30 アルカヘスト，インコーポレイテッド Ｃｃｒ３阻害剤を用いて、加齢性機能障害を治療するための方法及び組成物
US20190111042A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. Methods and Compositions for Treating Pruritus, Xerosis, and Associated Disease Using CCR-Inhibitors
MX2020011114A (es) 2018-05-15 2021-01-29 Alkahest Inc Tratamiento de enfermedades asociadas con el envejecimiento con moduladores de la leucotrieno a4 hidrolasa.
WO2020069008A1 (en) * 2018-09-26 2020-04-02 Alkahest, Inc. Methods and compositions for treating aging-associated impairments using ccr3-inhibitors
EP4206153A4 (en) 2020-08-27 2024-05-15 Agc Inc. ALKALI-FREE GLASS AND PLATE GLASS
US11957671B2 (en) 2021-11-01 2024-04-16 Alkahest, Inc. Benzodioxane modulators of leukotriene A4 hydrolase (LTA4H) for prevention and treatment of aging-associated diseases

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JP2002501898A (ja) 1998-02-02 2002-01-22 メルク エンド カムパニー インコーポレーテッド ケモカイン受容体活性の環状アミン調節剤
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