PT2094684E - 1,5-difenil-3-piridinilamino-1,5-di-hidro-pirrolidin-2-ona como modulador de receptores cb1 - Google Patents
1,5-difenil-3-piridinilamino-1,5-di-hidro-pirrolidin-2-ona como modulador de receptores cb1 Download PDFInfo
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- PT2094684E PT2094684E PT07871197T PT07871197T PT2094684E PT 2094684 E PT2094684 E PT 2094684E PT 07871197 T PT07871197 T PT 07871197T PT 07871197 T PT07871197 T PT 07871197T PT 2094684 E PT2094684 E PT 2094684E
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- phenyl
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- alkyl
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Classifications
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- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/36—Oxygen or sulfur atoms
- C07D207/38—2-Pyrrolones
Landscapes
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Applications Claiming Priority (1)
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| US86254006P | 2006-10-23 | 2006-10-23 |
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| PT78711967T PT2099784E (pt) | 2006-10-23 | 2007-10-22 | 1,5-difenil-3-piridinilamino-1,5-di-hidropirrolidin-2-ona como modulador do recetor de cbl |
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| PT78711967T PT2099784E (pt) | 2006-10-23 | 2007-10-22 | 1,5-difenil-3-piridinilamino-1,5-di-hidropirrolidin-2-ona como modulador do recetor de cbl |
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| PE20080926A1 (es) * | 2006-10-23 | 2008-07-19 | Lilly Co Eli | Compuestos cb1 |
| CN102119029B (zh) | 2008-04-22 | 2013-03-13 | 伊莱利利公司 | 作为cb-1配体的1，5-二苯基-吡咯烷-2-酮化合物 |
| JP5539323B2 (ja) * | 2008-04-22 | 2014-07-02 | イーライ リリー アンド カンパニー | Ｃｂ−１リガンドとしての１，５−ジフェニル−ピロリジン−２−オン化合物 |
| WO2010057000A2 (en) * | 2008-11-13 | 2010-05-20 | The Trustees Of Columbia University In The City Of New York | Neuraminidase inhibitors and uses thereof |
| NZ606768A (en) * | 2010-07-15 | 2015-08-28 | Oleg Iliich Epshtein | Pharmaceutical compositions and methods of treatment |
| WO2014078568A1 (en) | 2012-11-14 | 2014-05-22 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
| US20240158384A1 (en) * | 2020-12-14 | 2024-05-16 | The Board Of Trustees Of The Leland Stanford Junior University | Cb2 receptor agonists |
| WO2023205180A1 (en) | 2022-04-19 | 2023-10-26 | Nurix Therapeutics, Inc. | Biomarkers for cbl, and compositions and methods for their use |
| WO2023250097A1 (en) | 2022-06-22 | 2023-12-28 | Nurix Therapeutics, Inc. | Combination therapies with cbl-b inhibitor compounds and antiemetic agents |
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| TW200533657A (en) | 2004-02-17 | 2005-10-16 | Esteve Labor Dr | Substituted pyrazoline compounds, their preparation and use as medicaments |
| AU2005214084B2 (en) * | 2004-02-19 | 2010-06-03 | Solvay Pharmaceuticals B.V. | Imidazoline derivatives having CB1-antagonistic activity |
| US20060035245A1 (en) * | 2004-04-20 | 2006-02-16 | Ason Brandon L | Modulators of enzymatic nucleic acid elements mobilization |
| WO2007020502A2 (en) * | 2005-08-16 | 2007-02-22 | Pharmacia & Upjohn Company Llc | Cannabinoid receptor ligands and uses thereof |
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- 2007-10-22 KR KR1020097008216A patent/KR101088229B1/ko not_active Expired - Fee Related
- 2007-10-22 US US12/444,692 patent/US7998985B2/en not_active Expired - Fee Related
- 2007-10-22 CN CN2007800394514A patent/CN101528733B/zh not_active Expired - Fee Related
-
2011
- 2011-01-27 CY CY20111100093T patent/CY1111140T1/el unknown
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