EA015175B1 - Соединения, проявляющие активность в отношении рецептора св - Google Patents
Соединения, проявляющие активность в отношении рецептора св Download PDFInfo
- Publication number
- EA015175B1 EA015175B1 EA200970405A EA200970405A EA015175B1 EA 015175 B1 EA015175 B1 EA 015175B1 EA 200970405 A EA200970405 A EA 200970405A EA 200970405 A EA200970405 A EA 200970405A EA 015175 B1 EA015175 B1 EA 015175B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- compound
- group
- trifluoromethoxyphenyl
- cyclopropyl
- methyl
- Prior art date
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| TW200825067A (en) * | 2006-10-23 | 2008-06-16 | Lilly Co Eli | CB1 compounds |
| BRPI0910775A2 (pt) | 2008-04-22 | 2015-09-29 | Lilly Co Eli | compostos 1,5-difenil pirrolidin-2-ona como ligantes cb-1 |
| US8426448B2 (en) | 2008-04-22 | 2013-04-23 | Eli Lilly And Company | 1,5-diphenyl-pyrrolidin-2-one compounds as CB-1 ligands |
| WO2010057000A2 (en) * | 2008-11-13 | 2010-05-20 | The Trustees Of Columbia University In The City Of New York | Neuraminidase inhibitors and uses thereof |
| WO2012007847A2 (en) * | 2010-07-15 | 2012-01-19 | Oleg Iliich Epshtein | Pharmaceutical compositions and methods of treatment |
| US10154988B2 (en) | 2012-11-14 | 2018-12-18 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
| US20240158384A1 (en) * | 2020-12-14 | 2024-05-16 | The Board Of Trustees Of The Leland Stanford Junior University | Cb2 receptor agonists |
| WO2023205180A1 (en) | 2022-04-19 | 2023-10-26 | Nurix Therapeutics, Inc. | Biomarkers for cbl, and compositions and methods for their use |
| WO2023250097A1 (en) | 2022-06-22 | 2023-12-28 | Nurix Therapeutics, Inc. | Combination therapies with cbl-b inhibitor compounds and antiemetic agents |
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| WO2005077911A1 (en) * | 2004-02-17 | 2005-08-25 | Laboratorios Del Dr. Esteve S.A. | Substituted pyrazoline compounds, their preparation and use as medicaments |
| WO2005080345A2 (en) * | 2004-02-19 | 2005-09-01 | Solvay Pharmaceuticals B.V. | Imidazoline derivatives having cb1-antagonistic activity |
| WO2007020502A2 (en) * | 2005-08-16 | 2007-02-22 | Pharmacia & Upjohn Company Llc | Cannabinoid receptor ligands and uses thereof |
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Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005077911A1 (en) * | 2004-02-17 | 2005-08-25 | Laboratorios Del Dr. Esteve S.A. | Substituted pyrazoline compounds, their preparation and use as medicaments |
| WO2005080345A2 (en) * | 2004-02-19 | 2005-09-01 | Solvay Pharmaceuticals B.V. | Imidazoline derivatives having cb1-antagonistic activity |
| WO2007020502A2 (en) * | 2005-08-16 | 2007-02-22 | Pharmacia & Upjohn Company Llc | Cannabinoid receptor ligands and uses thereof |
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