EA015175B1 - Соединения, проявляющие активность в отношении рецептора св - Google Patents
Соединения, проявляющие активность в отношении рецептора св Download PDFInfo
- Publication number
- EA015175B1 EA015175B1 EA200970405A EA200970405A EA015175B1 EA 015175 B1 EA015175 B1 EA 015175B1 EA 200970405 A EA200970405 A EA 200970405A EA 200970405 A EA200970405 A EA 200970405A EA 015175 B1 EA015175 B1 EA 015175B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- compound
- group
- trifluoromethoxyphenyl
- cyclopropyl
- methyl
- Prior art date
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| EA201071222A1 (ru) * | 2008-04-22 | 2011-12-30 | Эли Лилли Энд Компани | Соединения 1,5-дифенилпирролидин-2-она в качестве лигандов cb-1 |
| PL2280961T3 (pl) | 2008-04-22 | 2012-12-31 | Lilly Co Eli | Związki 1,5-difenylo-pirolidyn-2-onu jako ligandy CB-1 |
| US20110280813A1 (en) * | 2008-11-13 | 2011-11-17 | Alice Prince | Neuraminidase inhibitors and uses thereof |
| DE112011102349T5 (de) * | 2010-07-15 | 2013-04-18 | Oleg Iliich Epshtein | Pharmazeutische Zusammensetzung und Behandlungsverfahren |
| EP3610890A1 (en) | 2012-11-14 | 2020-02-19 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
| WO2022132803A1 (en) * | 2020-12-14 | 2022-06-23 | The Board Of Trustees Of The Leland Stanford Junior University | Cb2 receptor agonists |
| WO2023205180A1 (en) | 2022-04-19 | 2023-10-26 | Nurix Therapeutics, Inc. | Biomarkers for cbl, and compositions and methods for their use |
| US20230414598A1 (en) | 2022-06-22 | 2023-12-28 | Nurix Therapeutics, Inc. | Combination therapies with cbl-b inhibitor compounds and antiemetic agents |
Citations (3)
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| WO2005077911A1 (en) * | 2004-02-17 | 2005-08-25 | Laboratorios Del Dr. Esteve S.A. | Substituted pyrazoline compounds, their preparation and use as medicaments |
| WO2005080345A2 (en) * | 2004-02-19 | 2005-09-01 | Solvay Pharmaceuticals B.V. | Imidazoline derivatives having cb1-antagonistic activity |
| WO2007020502A2 (en) * | 2005-08-16 | 2007-02-22 | Pharmacia & Upjohn Company Llc | Cannabinoid receptor ligands and uses thereof |
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Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005077911A1 (en) * | 2004-02-17 | 2005-08-25 | Laboratorios Del Dr. Esteve S.A. | Substituted pyrazoline compounds, their preparation and use as medicaments |
| WO2005080345A2 (en) * | 2004-02-19 | 2005-09-01 | Solvay Pharmaceuticals B.V. | Imidazoline derivatives having cb1-antagonistic activity |
| WO2007020502A2 (en) * | 2005-08-16 | 2007-02-22 | Pharmacia & Upjohn Company Llc | Cannabinoid receptor ligands and uses thereof |
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