PT1412332E - Derivados de quinolina e sua utilizacao como agentes antitumorais - Google Patents

Derivados de quinolina e sua utilizacao como agentes antitumorais

Info

Publication number
PT1412332E
PT1412332E PT02752656T PT02752656T PT1412332E PT 1412332 E PT1412332 E PT 1412332E PT 02752656 T PT02752656 T PT 02752656T PT 02752656 T PT02752656 T PT 02752656T PT 1412332 E PT1412332 E PT 1412332E
Authority
PT
Portugal
Prior art keywords
formula
compound
antitumor agents
quinoline derivatives
salt
Prior art date
Application number
PT02752656T
Other languages
English (en)
Inventor
Jerome P Horwitz
Stewart T Hazeldine
Thomas H Corbett
Lisa Polin
Original Assignee
Jerome P Horwitz
Stewart T Hazeldine
Thomas H Corbett
Lisa Polin
Univ Wayne State
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jerome P Horwitz, Stewart T Hazeldine, Thomas H Corbett, Lisa Polin, Univ Wayne State filed Critical Jerome P Horwitz
Publication of PT1412332E publication Critical patent/PT1412332E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
PT02752656T 2001-07-31 2002-07-31 Derivados de quinolina e sua utilizacao como agentes antitumorais PT1412332E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30914401P 2001-07-31 2001-07-31

Publications (1)

Publication Number Publication Date
PT1412332E true PT1412332E (pt) 2005-06-30

Family

ID=23196886

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02752656T PT1412332E (pt) 2001-07-31 2002-07-31 Derivados de quinolina e sua utilizacao como agentes antitumorais

Country Status (22)

Country Link
US (3) US6867219B2 (pt)
EP (1) EP1412332B1 (pt)
JP (1) JP4310185B2 (pt)
KR (1) KR20040055774A (pt)
AT (1) ATE287397T1 (pt)
AU (1) AU2002355747B2 (pt)
CA (1) CA2456173A1 (pt)
DE (1) DE60202682T2 (pt)
DK (1) DK1412332T3 (pt)
EA (1) EA007205B1 (pt)
ES (1) ES2236548T3 (pt)
GE (1) GEP20063754B (pt)
HU (1) HUP0401562A2 (pt)
IL (2) IL160082A0 (pt)
MX (1) MXPA04000968A (pt)
NO (1) NO326463B1 (pt)
NZ (1) NZ530806A (pt)
PL (1) PL367340A1 (pt)
PT (1) PT1412332E (pt)
UA (1) UA75691C2 (pt)
WO (1) WO2003011832A1 (pt)
ZA (1) ZA200401185B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001064642A2 (en) * 2000-02-29 2001-09-07 Cor Therapeutics, Inc. Benzamides and related inhibitors of factor xa
DK1412332T3 (da) * 2001-07-31 2005-05-30 Univ Wayne State Quinolinderivater og anvendelse deraf som antitumormidler
UA79293C2 (en) * 2002-07-03 2007-06-11 Univ Wayne State 4-(7'-halo-2-quino (xa-) linyloxy)phenoxy propionic acid derivatives as antineoplastic agents
RU2322236C2 (ru) * 2002-08-24 2008-04-20 Центарис Гмбх Лекарственное средство для лечения доброкачественных и злокачественных опухолевых заболеваний, содержащее производное дисоразола
US7470788B2 (en) * 2005-09-07 2008-12-30 Wayne State University Antitumor agents
US20070054938A1 (en) * 2005-09-07 2007-03-08 Horwitz Jerome P Antitumor agents
US8183379B2 (en) 2005-09-07 2012-05-22 Wayne State University Antitumor agents
EP1897542A1 (en) * 2006-09-07 2008-03-12 Sanofi-Aventis Aqueous formulation comprising an antitumor agent
JO2685B1 (en) * 2006-12-06 2013-03-03 جانسين فارماسوتيكا ان في Quinoline antibacterial derivatives
WO2009002955A1 (en) * 2007-06-27 2008-12-31 Sanofi-Aventis U.S. Llc Process for the preparation of (2r)-2-[4-(7-bromo-2-quinolyloxy)phenoxy]propanoic acid
JP2014516075A (ja) 2011-06-06 2014-07-07 シェブロン フィリップス ケミカル カンパニー エルピー 癌治療のためのメタロセン化合物の使用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6033389B2 (ja) * 1979-02-22 1985-08-02 日産化学工業株式会社 複素環エ−テル系フェノシキ脂肪酸誘導体、その製造法および該誘導体を含有する除草剤
US6197728B1 (en) * 1980-08-06 2001-03-06 Nissan Chemical Industries Ltd. Quinoxaline derivatives and herbicidal composition
US5364831A (en) * 1980-08-06 1994-11-15 Nissan Chemical Industries Ltd. Quinoxaline derivatives and herbicidal composition
US5250690A (en) * 1985-05-02 1993-10-05 Dowelanco Haloalkoxy anilide derivatives of 2-4(-heterocyclic oxyphenoxy)alkanoic or alkenoic acids and their use as herbicides
DK1412332T3 (da) * 2001-07-31 2005-05-30 Univ Wayne State Quinolinderivater og anvendelse deraf som antitumormidler
UA79293C2 (en) * 2002-07-03 2007-06-11 Univ Wayne State 4-(7'-halo-2-quino (xa-) linyloxy)phenoxy propionic acid derivatives as antineoplastic agents
US7470788B2 (en) * 2005-09-07 2008-12-30 Wayne State University Antitumor agents

Also Published As

Publication number Publication date
US7507749B2 (en) 2009-03-24
HUP0401562A2 (hu) 2004-12-28
IL160082A (en) 2009-06-15
GEP20063754B (en) 2006-02-27
EP1412332A1 (en) 2004-04-28
JP4310185B2 (ja) 2009-08-05
AU2002355747B2 (en) 2007-12-20
NZ530806A (en) 2006-05-26
UA75691C2 (en) 2006-05-15
EP1412332B1 (en) 2005-01-19
ZA200401185B (en) 2004-10-21
ES2236548T3 (es) 2005-07-16
ATE287397T1 (de) 2005-02-15
US20030144321A1 (en) 2003-07-31
US6867219B2 (en) 2005-03-15
NO326463B1 (no) 2008-12-08
DE60202682T2 (de) 2005-12-29
WO2003011832A1 (en) 2003-02-13
JP2004538314A (ja) 2004-12-24
MXPA04000968A (es) 2005-02-17
KR20040055774A (ko) 2004-06-26
NO20040382L (no) 2004-03-26
EA200400219A1 (ru) 2004-12-30
DK1412332T3 (da) 2005-05-30
IL160082A0 (en) 2004-06-20
DE60202682D1 (de) 2005-02-24
EA007205B1 (ru) 2006-08-25
CA2456173A1 (en) 2003-02-13
US20070232643A1 (en) 2007-10-04
PL367340A1 (en) 2005-02-21
US7241894B2 (en) 2007-07-10
US20050159447A1 (en) 2005-07-21

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