EA200600022A1 - Применение производных бицикло [2.2.1] гептана для приготовления нейропротекторных фармацевтических композиций - Google Patents
Применение производных бицикло [2.2.1] гептана для приготовления нейропротекторных фармацевтических композицийInfo
- Publication number
- EA200600022A1 EA200600022A1 EA200600022A EA200600022A EA200600022A1 EA 200600022 A1 EA200600022 A1 EA 200600022A1 EA 200600022 A EA200600022 A EA 200600022A EA 200600022 A EA200600022 A EA 200600022A EA 200600022 A1 EA200600022 A1 EA 200600022A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- pharmaceutical compositions
- heptana
- bicyclo
- derivative
- prepare
- Prior art date
Links
- 230000000324 neuroprotective effect Effects 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Abstract
Изобретение относится к применению соединений общей формулы I (где Rозначает водород или гидроксил; Rозначает водород или алкил и Rозначает алкил) и их фармацевтически приемлемых кислотно-аддитивных солей для приготовления фармацевтических композиций, обладающих нейропротекторным действием.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU0301906A HUP0301906A3 (en) | 2003-06-23 | 2003-06-23 | Use of bicyclo[2.2.1]heptane derivatives for producing of pharmaceutical compositions having neuroprotectiv activity |
PCT/HU2004/000062 WO2004112769A1 (en) | 2003-06-23 | 2004-06-22 | Use of bicyclo[2.2.1]heptane derivatives for the preparation of neuroprotective pharmaceutical compositions |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200600022A1 true EA200600022A1 (ru) | 2006-08-25 |
EA010868B1 EA010868B1 (ru) | 2008-12-30 |
Family
ID=90001689
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200600022A EA010868B1 (ru) | 2003-06-23 | 2004-06-22 | Применение производных бицикло[2.2.1]гептана для приготовления нейропротекторных фармацевтических композиций |
Country Status (23)
Country | Link |
---|---|
US (1) | US20060258750A1 (ru) |
EP (1) | EP1660063A1 (ru) |
JP (1) | JP2007516165A (ru) |
KR (1) | KR20060023997A (ru) |
CN (1) | CN1812778A (ru) |
AU (1) | AU2004248982A1 (ru) |
BG (1) | BG109414A (ru) |
BR (1) | BRPI0411772A (ru) |
CA (1) | CA2529254A1 (ru) |
CZ (1) | CZ200631A3 (ru) |
EA (1) | EA010868B1 (ru) |
HR (1) | HRP20060023A2 (ru) |
HU (1) | HUP0301906A3 (ru) |
IL (1) | IL172408A0 (ru) |
IS (1) | IS8239A (ru) |
MX (1) | MXPA05014127A (ru) |
NO (1) | NO20060277L (ru) |
PL (1) | PL378630A1 (ru) |
RS (1) | RS20050954A (ru) |
SK (1) | SK50082006A3 (ru) |
UA (1) | UA81052C2 (ru) |
WO (1) | WO2004112769A1 (ru) |
ZA (1) | ZA200510138B (ru) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5173190B2 (ja) | 2004-08-25 | 2013-03-27 | 武田薬品工業株式会社 | 腹圧性尿失禁の予防・治療剤及びそのスクリーニング方法 |
EP2018863B9 (en) | 2006-05-16 | 2015-02-18 | Takeda Pharmaceutical Company Limited | Fused heterocyclic compound and use thereof |
US20100266504A1 (en) | 2007-11-15 | 2010-10-21 | Takahiro Matsumoto | Condensed pyridine derivative and use thereof |
CZ2008602A3 (cs) * | 2008-10-09 | 2009-11-25 | Ústav chemických procesu Akademie ved Ceské republiky | Zpusob a zarízení pro izolaci kyseliny tereftalové |
EP2510949A4 (en) | 2009-12-11 | 2013-11-13 | Astellas Pharma Inc | THERAPEUTICS FOR FIBROMYALGIA |
US11478467B2 (en) | 2017-05-04 | 2022-10-25 | Sreenivasarao Vepachedu | Targeted drug rescue with novel compositions, combinations, and methods thereof |
US20210052600A1 (en) | 2017-12-27 | 2021-02-25 | Takeda Pharmaceutical Company Limited | Therapeutic agents for stress urinary incontinence and incotinence of feces |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HU227114B1 (en) * | 1999-05-11 | 2010-07-28 | Egis Gyogyszergyar Nyilvanosan | (1r, 2s, 4r)-(-)-2-[n,n-(dimethylamino-ethoxy)]-2-phenyl-1,7,7-trimethyl-bicyclo[2.2.1]heptane of high purity and pharmaceutically acceptable acid addition salts thereof, process for preparation of them and medicaments containing the same |
US6335371B1 (en) * | 2000-11-28 | 2002-01-01 | Orion Corporation | Method for inducing cognition enhancement |
HUP0103017A3 (en) * | 2001-07-18 | 2004-05-28 | Egis Gyogyszergyar Nyilvanosan | Pharmaceutical composition for the treatment of diseases caused by impairment of cognitive functions and its use |
-
2003
- 2003-06-23 HU HU0301906A patent/HUP0301906A3/hu unknown
-
2004
- 2004-06-22 EA EA200600022A patent/EA010868B1/ru not_active IP Right Cessation
- 2004-06-22 CN CNA2004800177453A patent/CN1812778A/zh active Pending
- 2004-06-22 CA CA002529254A patent/CA2529254A1/en not_active Abandoned
- 2004-06-22 KR KR1020057024601A patent/KR20060023997A/ko not_active Application Discontinuation
- 2004-06-22 SK SK5008-2006A patent/SK50082006A3/sk not_active Application Discontinuation
- 2004-06-22 PL PL378630A patent/PL378630A1/pl not_active Application Discontinuation
- 2004-06-22 JP JP2006516495A patent/JP2007516165A/ja active Pending
- 2004-06-22 AU AU2004248982A patent/AU2004248982A1/en not_active Abandoned
- 2004-06-22 WO PCT/HU2004/000062 patent/WO2004112769A1/en active Application Filing
- 2004-06-22 EP EP04743721A patent/EP1660063A1/en not_active Withdrawn
- 2004-06-22 UA UAA200600574A patent/UA81052C2/uk unknown
- 2004-06-22 RS YUP-2005/0954A patent/RS20050954A/sr unknown
- 2004-06-22 BR BRPI0411772-7A patent/BRPI0411772A/pt not_active IP Right Cessation
- 2004-06-22 ZA ZA200510138A patent/ZA200510138B/xx unknown
- 2004-06-22 MX MXPA05014127A patent/MXPA05014127A/es not_active Application Discontinuation
- 2004-06-22 US US10/562,393 patent/US20060258750A1/en not_active Abandoned
-
2005
- 2005-12-06 IL IL172408A patent/IL172408A0/en unknown
-
2006
- 2006-01-16 CZ CZ20060031A patent/CZ200631A3/cs unknown
- 2006-01-17 HR HR20060023A patent/HRP20060023A2/xx not_active Application Discontinuation
- 2006-01-18 IS IS8239A patent/IS8239A/is unknown
- 2006-01-19 NO NO20060277A patent/NO20060277L/no not_active Application Discontinuation
- 2006-01-23 BG BG109414A patent/BG109414A/bg unknown
Also Published As
Publication number | Publication date |
---|---|
JP2007516165A (ja) | 2007-06-21 |
AU2004248982A1 (en) | 2004-12-29 |
IL172408A0 (en) | 2006-04-10 |
UA81052C2 (en) | 2007-11-26 |
EP1660063A1 (en) | 2006-05-31 |
MXPA05014127A (es) | 2006-02-24 |
HUP0301906D0 (en) | 2003-08-28 |
EA010868B1 (ru) | 2008-12-30 |
HRP20060023A2 (en) | 2006-05-31 |
RS20050954A (en) | 2007-08-03 |
BRPI0411772A (pt) | 2006-08-08 |
HUP0301906A3 (en) | 2006-03-28 |
WO2004112769A1 (en) | 2004-12-29 |
CZ200631A3 (cs) | 2006-05-17 |
US20060258750A1 (en) | 2006-11-16 |
BG109414A (bg) | 2006-11-30 |
HUP0301906A2 (en) | 2006-02-28 |
KR20060023997A (ko) | 2006-03-15 |
CA2529254A1 (en) | 2004-12-29 |
SK50082006A3 (sk) | 2006-05-04 |
IS8239A (is) | 2006-01-18 |
PL378630A1 (pl) | 2006-05-15 |
ZA200510138B (en) | 2007-03-28 |
NO20060277L (no) | 2006-01-19 |
CN1812778A (zh) | 2006-08-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |