PL376557A1 - Postacie krystaliczne pitawastatyny wapnia - Google Patents

Postacie krystaliczne pitawastatyny wapnia

Info

Publication number
PL376557A1
PL376557A1 PL376557A PL37655704A PL376557A1 PL 376557 A1 PL376557 A1 PL 376557A1 PL 376557 A PL376557 A PL 376557A PL 37655704 A PL37655704 A PL 37655704A PL 376557 A1 PL376557 A1 PL 376557A1
Authority
PL
Poland
Prior art keywords
crystalline forms
pitavastatin calcium
pitavastatin
calcium
quinolin
Prior art date
Application number
PL376557A
Other languages
English (en)
Polish (pl)
Inventor
Der Schaaf Paul Adriaan Van
Fritz Blatter
Martin Szelagiewicz
Kai-Uwe Schöning
Original Assignee
Ciba Specialty Chemicals Holding Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32865094&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL376557(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ciba Specialty Chemicals Holding Inc. filed Critical Ciba Specialty Chemicals Holding Inc.
Publication of PL376557A1 publication Critical patent/PL376557A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14—Radicals substituted by oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
PL376557A 2003-02-12 2004-02-02 Postacie krystaliczne pitawastatyny wapnia PL376557A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP03405080 2003-02-12

Publications (1)

Publication Number Publication Date
PL376557A1 true PL376557A1 (pl) 2006-01-09

Family

ID=32865094

Family Applications (1)

Application Number Title Priority Date Filing Date
PL376557A PL376557A1 (pl) 2003-02-12 2004-02-02 Postacie krystaliczne pitawastatyny wapnia

Country Status (10)

Country Link
US (15) US20060142582A1 (https=)
EP (3) EP1592668A1 (https=)
JP (13) JP5192147B2 (https=)
CN (3) CN101219992B (https=)
AU (1) AU2004212160B2 (https=)
CA (2) CA2785954A1 (https=)
DE (1) DE202004021379U1 (https=)
PL (1) PL376557A1 (https=)
TW (4) TW201213311A (https=)
WO (1) WO2004072040A1 (https=)

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CN101219992B (zh) * 2003-02-12 2011-08-31 日产化学工业株式会社 匹伐他汀钙的晶形
AU2013204129C1 (en) * 2003-12-26 2017-03-02 Nissan Chemical Industries, Ltd. Crystal Form of Quinoline Compound and Process for its Production
TWI328006B (en) * 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production
US20070173536A1 (en) * 2004-02-06 2007-07-26 Ciba Specialty Chemicals Holding Inc. Crystalline forms of zolmitriptan
WO2006079611A1 (en) * 2005-01-31 2006-08-03 Ciba Specialty Chemicals Holding Inc. Crystalline forms of rosuvastatin calcium salt
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JP2013536219A (ja) 2010-08-25 2013-09-19 カディラ・ヘルスケア・リミテッド ピタバスタチンカルシウムおよびその調製方法
EP3178812A1 (en) 2010-11-12 2017-06-14 Hetero Research Foundation Novel polymorphs of pitavastatin calcium
WO2012106584A2 (en) * 2011-02-04 2012-08-09 Dr. Reddy's Laboratories Ltd. Pitavastatin salts
ITMI20111475A1 (it) * 2011-08-02 2013-02-03 Dipharma Francis Srl Forme cristalline di pitavastatina sale di calcio
PT2751081T (pt) 2011-09-12 2017-04-04 D O O Farma Grs Forma polimórfica de pitavastatina cálcica
EP2768805B1 (en) * 2011-10-20 2020-03-25 Oryzon Genomics, S.A. (hetero)aryl cyclopropylamine compounds as lsd1 inhibitors
WO2013098773A1 (en) * 2011-12-28 2013-07-04 Dr. Reddy's Laboratories Limited Crystalline forms of pitavastatin calcium
CN104860882A (zh) * 2015-05-15 2015-08-26 苗怡文 一种治疗高血脂症的药物匹伐他汀钙组合物
CN104844506A (zh) * 2015-05-15 2015-08-19 苗怡文 一种治疗高血脂症的药物匹伐他汀钙化合物
CN105125504A (zh) * 2015-09-17 2015-12-09 青岛华之草医药科技有限公司 一种降血脂药物匹伐他汀钙组合物颗粒剂
CN105213319A (zh) * 2015-09-17 2016-01-06 青岛华之草医药科技有限公司 一种降血脂药物匹伐他汀钙组合物干混悬剂
US10937978B2 (en) * 2016-02-25 2021-03-02 University Of Louisville Research Foundation, Inc. Methods for forming a perovskite solar cell
US10600502B2 (en) 2016-12-20 2020-03-24 Astrazeneca Uk Ltd. Systems and methods for dispensing a statin medication over the counter
CN109053568A (zh) * 2018-08-29 2018-12-21 南京卓康医药科技有限公司 一种高纯度匹伐他汀钙新晶型及其制备方法
CN113834795B (zh) * 2020-06-08 2024-12-03 上海医药集团股份有限公司 硫酸羟氯喹颗粒水分近红外光谱在线定量模型及其建立方法及检测方法
US20220008519A1 (en) 2020-07-09 2022-01-13 Costa Rican Social Security Fund / Caja Costarricense de Seguro Social (CCSS) Treatment of severe acute respiratory syndrome-related coronavirus infection with klotho
EP4405360A4 (en) 2021-09-23 2025-08-20 Erasca Inc POLYMORPHIC FORMS OF EGFR INHIBITOR
CN116969884A (zh) * 2023-07-28 2023-10-31 河北广祥制药有限公司 一种匹伐他汀钙单晶及其制备方法

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JP4281248B2 (ja) * 1998-07-23 2009-06-17 日産化学工業株式会社 キノリン誘導体の製造法及び中間体
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EP1345903A1 (en) * 2000-12-21 2003-09-24 Ciba SC Holding AG Crystalline forms of cerivastatin sodium
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CN101219992B (zh) * 2003-02-12 2011-08-31 日产化学工业株式会社 匹伐他汀钙的晶形
TWI328006B (en) 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production
CN100344422C (zh) * 2006-05-11 2007-10-24 朱能国 用人工用材林松木及其板材生产阻燃防潮装饰板材的方法
JP5353678B2 (ja) * 2009-12-17 2013-11-27 トヨタ自動車株式会社 車両の制御装置

Also Published As

Publication number Publication date
US20170022163A1 (en) 2017-01-26
JP5702494B2 (ja) 2015-04-15
EP1592668A1 (en) 2005-11-09
AU2004212160A1 (en) 2004-08-26
JP2014198743A (ja) 2014-10-23
WO2004072040A1 (en) 2004-08-26
US20120101126A1 (en) 2012-04-26
US20090182008A1 (en) 2009-07-16
JP2014205723A (ja) 2014-10-30
CN100374422C (zh) 2008-03-12
JP2018044009A (ja) 2018-03-22
TW200420541A (en) 2004-10-16
TW201345893A (zh) 2013-11-16
JP2019031574A (ja) 2019-02-28
US20060142582A1 (en) 2006-06-29
TW201213311A (en) 2012-04-01
US20140005402A1 (en) 2014-01-02
US20180346425A1 (en) 2018-12-06
TWI485135B (zh) 2015-05-21
DE202004021379U1 (de) 2008-02-21
US8853405B2 (en) 2014-10-07
EP3299359A1 (en) 2018-03-28
JP5500305B2 (ja) 2014-05-21
JP5445713B2 (ja) 2014-03-19
US20190256469A1 (en) 2019-08-22
US20160024010A1 (en) 2016-01-28
US20140364614A1 (en) 2014-12-11
JP2013177466A (ja) 2013-09-09
US20210002227A1 (en) 2021-01-07
JP2014055185A (ja) 2014-03-27
US8557993B2 (en) 2013-10-15
CN101219992A (zh) 2008-07-16
US20130053413A1 (en) 2013-02-28
JP2014024848A (ja) 2014-02-06
TW201514149A (zh) 2015-04-16
JP5192147B2 (ja) 2013-05-08
JP2016222737A (ja) 2016-12-28
CN102285916A (zh) 2011-12-21
US20180029987A1 (en) 2018-02-01
JP2020169196A (ja) 2020-10-15
CN102285916B (zh) 2015-02-25
EP2500339A1 (en) 2012-09-19
JP2011201915A (ja) 2011-10-13
US20220169614A1 (en) 2022-06-02
CN101219992B (zh) 2011-08-31
CA2785954A1 (en) 2004-08-26
JP2006518354A (ja) 2006-08-10
JP2014062115A (ja) 2014-04-10
CN1747934A (zh) 2006-03-15
CA2513837A1 (en) 2004-08-26
JP5366163B2 (ja) 2013-12-11
JP2015172086A (ja) 2015-10-01
US20200148644A1 (en) 2020-05-14
US20230322680A1 (en) 2023-10-12
AU2004212160B2 (en) 2009-05-14

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