PL2134702T5 - Krystaliczne postacie 6-[2-(metylokarbamoilo)fenylosulfanylo]-3-e-[2-(pirydyn-2-ylo)etenylo]indazolu przydatne w leczeniu nienormalnego wzrostu komórek u ssaków - Google Patents

Krystaliczne postacie 6-[2-(metylokarbamoilo)fenylosulfanylo]-3-e-[2-(pirydyn-2-ylo)etenylo]indazolu przydatne w leczeniu nienormalnego wzrostu komórek u ssaków

Info

Publication number
PL2134702T5
PL2134702T5 PL08719405.6T PL08719405T PL2134702T5 PL 2134702 T5 PL2134702 T5 PL 2134702T5 PL 08719405 T PL08719405 T PL 08719405T PL 2134702 T5 PL2134702 T5 PL 2134702T5
Authority
PL
Poland
Prior art keywords
phenylsulfanyl
methylcarbamoyl
indazole
ethenyl
pyridin
Prior art date
Application number
PL08719405.6T
Other languages
English (en)
Other versions
PL2134702T3 (pl
Inventor
Anthony Michael Campeta
Brian Patrick Chekal
Robert William Mclaughling
Robert Alan Singer
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39831473&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2134702(T5) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of PL2134702T3 publication Critical patent/PL2134702T3/pl
Publication of PL2134702T5 publication Critical patent/PL2134702T5/pl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL08719405.6T 2007-04-05 2008-03-25 Krystaliczne postacie 6-[2-(metylokarbamoilo)fenylosulfanylo]-3-e-[2-(pirydyn-2-ylo)etenylo]indazolu przydatne w leczeniu nienormalnego wzrostu komórek u ssaków PL2134702T5 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US91037907P 2007-04-05 2007-04-05
US97654607P 2007-10-01 2007-10-01
US3155408P 2008-02-26 2008-02-26
PCT/IB2008/000792 WO2008122858A2 (en) 2007-04-05 2008-03-25 Crystalline forms of 6- [2- (methylcarbamoyl) phenylsulfanyl] -3-e- [2- (pyridin-2-yl) ethenyl] indazole suitable for the treatment of abnormal cell growth in mammals
EP08719405.6A EP2134702B2 (en) 2007-04-05 2008-03-25 Crystalline forms of 6-[2-(methylcarbamoyl)phenylsulfanyl]-3-e-[2-(pyridin-2-yl)ethenyl]indazole suitable for the treatment of abnormal cell growth in mammals

Publications (2)

Publication Number Publication Date
PL2134702T3 PL2134702T3 (pl) 2017-10-31
PL2134702T5 true PL2134702T5 (pl) 2023-12-04

Family

ID=39831473

Family Applications (1)

Application Number Title Priority Date Filing Date
PL08719405.6T PL2134702T5 (pl) 2007-04-05 2008-03-25 Krystaliczne postacie 6-[2-(metylokarbamoilo)fenylosulfanylo]-3-e-[2-(pirydyn-2-ylo)etenylo]indazolu przydatne w leczeniu nienormalnego wzrostu komórek u ssaków

Country Status (23)

Country Link
US (1) US8791140B2 (pl)
EP (4) EP4074702A1 (pl)
JP (2) JP5869197B2 (pl)
KR (1) KR101237588B1 (pl)
CN (2) CN103626739B (pl)
AR (1) AR065931A1 (pl)
AU (1) AU2008236444B2 (pl)
BR (1) BRPI0809471A2 (pl)
CA (1) CA2682859C (pl)
CY (1) CY1119119T1 (pl)
DK (1) DK2134702T4 (pl)
ES (2) ES2919351T3 (pl)
FI (1) FI2134702T4 (pl)
IL (1) IL201320A (pl)
MX (1) MX2009010761A (pl)
NZ (1) NZ580126A (pl)
PL (1) PL2134702T5 (pl)
PT (1) PT2134702T (pl)
RU (1) RU2518898C2 (pl)
SG (1) SG156088A1 (pl)
SI (1) SI2134702T2 (pl)
TW (1) TWI481602B (pl)
WO (1) WO2008122858A2 (pl)

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Also Published As

Publication number Publication date
CY1119119T1 (el) 2018-02-14
CN103626739A (zh) 2014-03-12
TW200911781A (en) 2009-03-16
PL2134702T3 (pl) 2017-10-31
SI2134702T1 (sl) 2017-07-31
DK2134702T4 (da) 2023-09-25
IL201320A (en) 2016-05-31
CA2682859A1 (en) 2008-10-16
SI2134702T2 (sl) 2023-12-29
ES2634866T5 (es) 2024-03-04
AU2008236444A1 (en) 2008-10-16
EP4074702A1 (en) 2022-10-19
HK1193405A1 (zh) 2014-09-19
CN101679356A (zh) 2010-03-24
JP2014193900A (ja) 2014-10-09
EP3252047A3 (en) 2018-08-15
WO2008122858A9 (en) 2009-06-18
RU2009136593A (ru) 2011-04-10
WO2008122858A8 (en) 2009-11-26
EP2134702B1 (en) 2017-05-31
ES2919351T3 (es) 2022-07-26
FI2134702T4 (fi) 2023-09-12
KR20090127949A (ko) 2009-12-14
BRPI0809471A2 (pt) 2014-09-09
NZ580126A (en) 2012-03-30
WO2008122858A2 (en) 2008-10-16
RU2518898C2 (ru) 2014-06-10
KR101237588B1 (ko) 2013-02-27
JP5869197B2 (ja) 2016-02-24
SG156088A1 (en) 2009-11-26
CA2682859C (en) 2013-10-08
EP4249063A2 (en) 2023-09-27
IL201320A0 (en) 2010-05-31
EP3252047A2 (en) 2017-12-06
EP2134702B2 (en) 2023-08-30
US20100179329A1 (en) 2010-07-15
ES2634866T3 (es) 2017-09-29
WO2008122858A3 (en) 2009-05-07
CN103626739B (zh) 2015-12-30
DK2134702T3 (en) 2017-08-21
AU2008236444B2 (en) 2012-06-28
JP2009019030A (ja) 2009-01-29
EP2134702A2 (en) 2009-12-23
TWI481602B (zh) 2015-04-21
US8791140B2 (en) 2014-07-29
EP3252047B1 (en) 2022-05-11
PT2134702T (pt) 2017-07-31
MX2009010761A (es) 2009-10-28
EP4249063A3 (en) 2024-03-13
AR065931A1 (es) 2009-07-08

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