PL103731B1 - Sposob wytwarzania kwasu 6-metoksy-alfa-karboksypenicylanowego - Google Patents

Sposob wytwarzania kwasu 6-metoksy-alfa-karboksypenicylanowego Download PDF

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Publication number
PL103731B1
PL103731B1 PL1976186599A PL18659976A PL103731B1 PL 103731 B1 PL103731 B1 PL 103731B1 PL 1976186599 A PL1976186599 A PL 1976186599A PL 18659976 A PL18659976 A PL 18659976A PL 103731 B1 PL103731 B1 PL 103731B1
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PL
Poland
Prior art keywords
acid
formula
group
proton
thienyl
Prior art date
Application number
PL1976186599A
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English (en)
Polish (pl)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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Publication of PL103731B1 publication Critical patent/PL103731B1/pl

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PL1976186599A 1975-01-17 1976-01-17 Sposob wytwarzania kwasu 6-metoksy-alfa-karboksypenicylanowego PL103731B1 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB2021/75A GB1538051A (en) 1975-01-17 1975-01-17 6-methoxy-6-(alpha-carboxyacetamido)-penicillins
GB2566975 1975-06-17
GB3418275 1975-08-16

Publications (1)

Publication Number Publication Date
PL103731B1 true PL103731B1 (pl) 1979-07-31

Family

ID=27253985

Family Applications (1)

Application Number Title Priority Date Filing Date
PL1976186599A PL103731B1 (pl) 1975-01-17 1976-01-17 Sposob wytwarzania kwasu 6-metoksy-alfa-karboksypenicylanowego

Country Status (27)

Country Link
US (1) US4048320A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (2) JPS6126548B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AR (5) AR214173A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (2) AU500339B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (2) BE837456A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (2) CA1082688A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (6) CH630921A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (2) DE2600842A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (2) DK18476A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (5) ES444344A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (2) FI65257C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (2) FR2297624A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1538051A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR58525B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HK (1) HK22882A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (2) IE42707B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (2) IL48788A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KE (1) KE3205A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX3739E (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MY (1) MY8200243A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (2) NL189299C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (2) NO153221C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
OA (2) OA05211A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PH (2) PH12702A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PL (1) PL103731B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (2) SE435715B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
YU (5) YU40131B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1538051A (en) * 1975-01-17 1979-01-10 Beecham Group Ltd 6-methoxy-6-(alpha-carboxyacetamido)-penicillins
GB1577931A (en) * 1977-02-11 1980-10-29 Beecham Group Ltd 6-methoxy -6-(2-carboxy-2-(4-hydroxyphenyl) acetamido penicillins
NZ200177A (en) * 1981-04-15 1985-09-13 Beecham Group Plc Pharmaceutical compositions containing penicillin derivatives
JO1395B1 (en) * 1981-07-10 1986-11-30 بيتشام جروب بي ال سي Method for preparing active and antibacterial sleeper derivatives
IL67672A0 (en) * 1982-01-22 1983-05-15 Beecham Group Plc Penicillin derivatives,their preparation and pharmaceutical compositions containing them
CN102268017B (zh) * 2011-06-28 2012-11-28 苏州二叶制药有限公司 广谱长效青霉素类抗生素替卡西林钠的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR205683A1 (es) * 1970-06-16 1976-05-31 Merck & Co Inc Procedimiento para la preparacion del ester de bencilo del acido 6-metoxi-6-acilamido penicilanico
YU36181B (en) * 1971-11-29 1982-02-25 Merck & Co Inc Process for obtaining 7-(2-thienylacetamido)-7-methoxy-3-carbamoyloxymethyl-3-cephem-4-carboxylates
GB1425571A (en) * 1972-03-13 1976-02-18 Astra Laekemedel Ab Penicillins and cephaosporins
GB1538051A (en) * 1975-01-17 1979-01-10 Beecham Group Ltd 6-methoxy-6-(alpha-carboxyacetamido)-penicillins

Also Published As

Publication number Publication date
CA1083142A (en) 1980-08-05
FI65257B (fi) 1983-12-30
GR58525B (en) 1977-10-31
OA05212A (fr) 1981-02-28
MY8200243A (en) 1982-12-31
SE7600397L (sv) 1976-07-19
FR2297624A1 (fr) 1976-08-13
ES458427A1 (es) 1978-08-16
JPS5195093A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-08-20
AR217070A1 (es) 1980-02-29
JPS6126548B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1986-06-20
SE435716B (sv) 1984-10-15
FI760039A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-07-18
ES458431A1 (es) 1978-12-01
JPS5195092A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-08-20
IL48791A (en) 1979-09-30
AR212327A1 (es) 1978-06-30
DE2600842A1 (de) 1976-07-22
NO760150L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-07-20
NL7600430A (nl) 1976-07-20
YU94182A (en) 1982-08-31
IE42707B1 (en) 1980-10-08
DK154888B (da) 1989-01-02
IL48788A (en) 1979-07-25
AU500339B2 (en) 1979-05-17
NO760151L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-07-20
YU40131B (en) 1985-08-31
IE42707L (en) 1976-07-17
PH12969A (en) 1979-10-19
YU93782A (en) 1982-08-31
NO153221B (no) 1985-10-28
NL7600429A (nl) 1976-07-20
CH631459A5 (de) 1982-08-13
CH631458A5 (de) 1982-08-13
CH631457A5 (de) 1982-08-13
DK18476A (da) 1976-07-18
PH12702A (en) 1979-07-20
YU94082A (en) 1982-08-31
ES458430A1 (es) 1978-08-16
YU11476A (en) 1982-08-31
AR214173A1 (es) 1979-05-15
AU1017976A (en) 1977-07-14
IE43681B1 (en) 1981-05-06
YU40621B (en) 1986-02-28
US4048320A (en) 1977-09-13
CH630921A5 (de) 1982-07-15
ES444343A1 (es) 1977-10-01
FR2297625A1 (fr) 1976-08-13
AU500354B2 (en) 1979-05-17
AR214309A1 (es) 1979-05-31
CA1082688A (en) 1980-07-29
BE837455A (fr) 1976-07-09
ES444344A1 (es) 1977-10-01
DE2600866A1 (de) 1976-07-22
FI65257C (fi) 1984-04-10
IL48788A0 (en) 1976-03-31
NL189299B (nl) 1992-10-01
OA05211A (fr) 1981-02-28
GB1538051A (en) 1979-01-10
NL189299C (nl) 1993-03-01
FI760038A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-07-18
YU11876A (en) 1982-08-31
SE7600398L (sv) 1976-07-19
JPS621955B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1987-01-16
FR2297624B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1978-11-10
AR213838A1 (es) 1979-03-30
CH630922A5 (de) 1982-07-15
DK154888C (da) 1989-05-29
FI64940B (fi) 1983-10-31
CH631456A5 (de) 1982-08-13
DE2600842C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1987-12-23
AU1018076A (en) 1977-07-14
NO153221C (no) 1986-02-05
FR2297625B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1979-09-21
MX3739E (es) 1981-06-05
DK18376A (da) 1976-07-18
BE837456A (fr) 1976-07-09
KE3205A (en) 1982-06-04
DE2600866C2 (de) 1986-03-20
FI64940C (fi) 1984-02-10
HK22882A (en) 1982-06-04
IL48791A0 (en) 1976-03-31
IE43681L (en) 1976-07-17
SE435715B (sv) 1984-10-15

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