PH12015502560B1 - Use of a thiazolo pyrimidinone for the treatment of inflammatory bowel disease - Google Patents
Use of a thiazolo pyrimidinone for the treatment of inflammatory bowel diseaseInfo
- Publication number
- PH12015502560B1 PH12015502560B1 PH12015502560A PH12015502560A PH12015502560B1 PH 12015502560 B1 PH12015502560 B1 PH 12015502560B1 PH 12015502560 A PH12015502560 A PH 12015502560A PH 12015502560 A PH12015502560 A PH 12015502560A PH 12015502560 B1 PH12015502560 B1 PH 12015502560B1
- Authority
- PH
- Philippines
- Prior art keywords
- inflammatory bowel
- bowel disease
- treatment
- thiazolo
- pyrimidinone
- Prior art date
Links
- 208000022559 Inflammatory bowel disease Diseases 0.000 title abstract 3
- AKDQOJPOLRMVMF-UHFFFAOYSA-N [1,3]thiazolo[5,4-d]pyrimidine 3-oxide Chemical compound N1=CN=C2S(=O)C=NC2=C1 AKDQOJPOLRMVMF-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 3
- 229940126062 Compound A Drugs 0.000 abstract 2
- NLDMNSXOCDLTTB-UHFFFAOYSA-N Heterophylliin A Natural products O1C2COC(=O)C3=CC(O)=C(O)C(O)=C3C3=C(O)C(O)=C(O)C=C3C(=O)OC2C(OC(=O)C=2C=C(O)C(O)=C(O)C=2)C(O)C1OC(=O)C1=CC(O)=C(O)C(O)=C1 NLDMNSXOCDLTTB-UHFFFAOYSA-N 0.000 abstract 2
- 241000124008 Mammalia Species 0.000 abstract 2
- NFGVHWUWINDVLR-UHFFFAOYSA-N 2-[(5-hydroxy-3-oxo-8-thia-2,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),4,6-triene-4-carbonyl)amino]acetic acid Chemical compound OC(=O)CNC(=O)c1c(O)nc2sc3CCCCCc3n2c1=O NFGVHWUWINDVLR-UHFFFAOYSA-N 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Inorganic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1718MU2013 | 2013-05-14 | ||
| IN2309MU2013 | 2013-07-09 | ||
| PCT/IB2014/000707 WO2014184631A1 (en) | 2013-05-14 | 2014-05-12 | Use of a thiazolo pyrimidinone for the treatment of inflammatory bowel disease |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PH12015502560A1 PH12015502560A1 (en) | 2016-02-22 |
| PH12015502560B1 true PH12015502560B1 (en) | 2016-02-22 |
Family
ID=50896342
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH12015502560A PH12015502560B1 (en) | 2013-05-14 | 2015-11-10 | Use of a thiazolo pyrimidinone for the treatment of inflammatory bowel disease |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US9610247B2 (OSRAM) |
| EP (1) | EP2996693B1 (OSRAM) |
| JP (1) | JP6407974B2 (OSRAM) |
| KR (1) | KR102239649B1 (OSRAM) |
| CN (1) | CN105209043B (OSRAM) |
| AU (1) | AU2014266968B2 (OSRAM) |
| BR (1) | BR112015028581B1 (OSRAM) |
| CA (1) | CA2912011C (OSRAM) |
| CY (1) | CY1121280T1 (OSRAM) |
| DK (1) | DK2996693T3 (OSRAM) |
| EA (1) | EA030590B1 (OSRAM) |
| ES (1) | ES2712705T3 (OSRAM) |
| HR (1) | HRP20190315T1 (OSRAM) |
| HU (1) | HUE042691T2 (OSRAM) |
| IL (1) | IL242490B (OSRAM) |
| LT (1) | LT2996693T (OSRAM) |
| MX (1) | MX358198B (OSRAM) |
| MY (1) | MY179215A (OSRAM) |
| PH (1) | PH12015502560B1 (OSRAM) |
| PL (1) | PL2996693T3 (OSRAM) |
| PT (1) | PT2996693T (OSRAM) |
| RS (1) | RS58423B1 (OSRAM) |
| SG (1) | SG11201509275PA (OSRAM) |
| SI (1) | SI2996693T1 (OSRAM) |
| SM (1) | SMT201900111T1 (OSRAM) |
| TW (1) | TWI661828B (OSRAM) |
| UA (1) | UA117244C2 (OSRAM) |
| WO (1) | WO2014184631A1 (OSRAM) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI781922B (zh) * | 2016-03-14 | 2022-11-01 | 日商參天製藥股份有限公司 | 由葡甲胺或其鹽構成之防腐劑 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009002533A1 (en) * | 2007-06-27 | 2008-12-31 | The Brigham And Women's Hospital, Inc. | Inflammatory bowel disease therapies |
| TWI500623B (zh) * | 2009-10-13 | 2015-09-21 | Torrent Pharmaceuticals Ltd | 新穎稠合噻唑及噁唑嘧啶酮 |
| US8541430B2 (en) * | 2009-11-27 | 2013-09-24 | Torrent Pharmaceuticals Limited | Fused thiazolo and oxazolo pyrimidinones |
-
2014
- 2014-05-09 TW TW103116529A patent/TWI661828B/zh not_active IP Right Cessation
- 2014-05-12 KR KR1020157033744A patent/KR102239649B1/ko not_active Expired - Fee Related
- 2014-05-12 SG SG11201509275PA patent/SG11201509275PA/en unknown
- 2014-05-12 EA EA201592159A patent/EA030590B1/ru not_active IP Right Cessation
- 2014-05-12 JP JP2016513452A patent/JP6407974B2/ja not_active Expired - Fee Related
- 2014-05-12 MX MX2015015682A patent/MX358198B/es active IP Right Grant
- 2014-05-12 MY MYPI2015704098A patent/MY179215A/en unknown
- 2014-05-12 DK DK14728622.3T patent/DK2996693T3/en active
- 2014-05-12 SM SM20190111T patent/SMT201900111T1/it unknown
- 2014-05-12 ES ES14728622T patent/ES2712705T3/es active Active
- 2014-05-12 US US14/890,131 patent/US9610247B2/en not_active Expired - Fee Related
- 2014-05-12 CA CA2912011A patent/CA2912011C/en active Active
- 2014-05-12 UA UAA201512299A patent/UA117244C2/uk unknown
- 2014-05-12 PT PT14728622T patent/PT2996693T/pt unknown
- 2014-05-12 BR BR112015028581-3A patent/BR112015028581B1/pt not_active IP Right Cessation
- 2014-05-12 PL PL14728622T patent/PL2996693T3/pl unknown
- 2014-05-12 CN CN201480028313.6A patent/CN105209043B/zh not_active Expired - Fee Related
- 2014-05-12 RS RS20190216A patent/RS58423B1/sr unknown
- 2014-05-12 LT LTEP14728622.3T patent/LT2996693T/lt unknown
- 2014-05-12 AU AU2014266968A patent/AU2014266968B2/en not_active Ceased
- 2014-05-12 SI SI201431085T patent/SI2996693T1/sl unknown
- 2014-05-12 WO PCT/IB2014/000707 patent/WO2014184631A1/en not_active Ceased
- 2014-05-12 HU HUE14728622A patent/HUE042691T2/hu unknown
- 2014-05-12 HR HRP20190315TT patent/HRP20190315T1/hr unknown
- 2014-05-12 EP EP14728622.3A patent/EP2996693B1/en active Active
-
2015
- 2015-11-08 IL IL242490A patent/IL242490B/en active IP Right Grant
- 2015-11-10 PH PH12015502560A patent/PH12015502560B1/en unknown
-
2017
- 2017-02-22 US US15/439,733 patent/US10471005B2/en not_active Expired - Fee Related
-
2019
- 2019-02-21 CY CY20191100221T patent/CY1121280T1/el unknown
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