PE20001489A1 - ESTEROIDE (14ß,17O)-17-(HIDROXIMETILO) CON ACTIVIDAD ANDROGENA - Google Patents
ESTEROIDE (14ß,17O)-17-(HIDROXIMETILO) CON ACTIVIDAD ANDROGENAInfo
- Publication number
- PE20001489A1 PE20001489A1 PE2000000200A PE0002002000A PE20001489A1 PE 20001489 A1 PE20001489 A1 PE 20001489A1 PE 2000000200 A PE2000000200 A PE 2000000200A PE 0002002000 A PE0002002000 A PE 0002002000A PE 20001489 A1 PE20001489 A1 PE 20001489A1
- Authority
- PE
- Peru
- Prior art keywords
- alkyl
- halogen
- cyane
- steroid
- hydroximethyl
- Prior art date
Links
- 239000003098 androgen Substances 0.000 title abstract 2
- 150000003431 steroids Chemical class 0.000 title abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 7
- 150000002367 halogens Chemical class 0.000 abstract 7
- 150000001875 compounds Chemical class 0.000 abstract 2
- LVZWSLJZHVFIQJ-UHFFFAOYSA-N Cyclopropane Chemical compound C1CC1 LVZWSLJZHVFIQJ-UHFFFAOYSA-N 0.000 abstract 1
- 229910006069 SO3H Inorganic materials 0.000 abstract 1
- -1 STEROID COMPOUND Chemical class 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical class [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 150000001721 carbon Chemical class 0.000 abstract 1
- OKTJSMMVPCPJKN-BJUDXGSMSA-N carbon-11 Chemical compound [11C] OKTJSMMVPCPJKN-BJUDXGSMSA-N 0.000 abstract 1
- 239000002583 male contraceptive agent Substances 0.000 abstract 1
- 239000003270 steroid hormone Substances 0.000 abstract 1
- 125000000020 sulfo group Chemical group O=S(=O)([*])O[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J15/00—Stereochemically pure steroids containing carbon, hydrogen, halogen or oxygen having a partially or totally inverted skeleton, e.g. retrosteroids, L-isomers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Endocrinology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP99200665 | 1999-03-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20001489A1 true PE20001489A1 (es) | 2000-12-29 |
Family
ID=8239953
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2000000200A PE20001489A1 (es) | 1999-03-08 | 2000-03-07 | ESTEROIDE (14ß,17O)-17-(HIDROXIMETILO) CON ACTIVIDAD ANDROGENA |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6881728B1 (https=) |
| EP (1) | EP1163259B1 (https=) |
| JP (1) | JP4749550B2 (https=) |
| AR (1) | AR022852A1 (https=) |
| AT (1) | ATE228143T1 (https=) |
| AU (1) | AU3162200A (https=) |
| CA (1) | CA2359218A1 (https=) |
| CO (1) | CO5150195A1 (https=) |
| DE (1) | DE60000826T2 (https=) |
| PE (1) | PE20001489A1 (https=) |
| WO (1) | WO2000053619A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU778017B2 (en) * | 1999-12-02 | 2004-11-11 | N.V. Organon | 14,15-beta-methylene substituted androgens |
| DK1343806T3 (da) * | 2000-12-11 | 2008-09-22 | Organon Nv | Methylensteroider som nye androgener |
| DE10104327A1 (de) * | 2001-01-24 | 2002-07-25 | Schering Ag | 11beta-Halogensteroide, deren Herstellung und Verwendung zur Herstellung von Arzneimitteln sowie 11beta-Halogensteroide enthaltende pharmazeutische Präparate |
| TWI221154B (en) * | 2001-09-12 | 2004-09-21 | Akzo Nobel Nv | 17alpha-hydroxy-14beta-steroids with hormonal effect |
| PE20050677A1 (es) | 2003-12-22 | 2005-10-04 | Akzo Nobel Nv | Esteroides con perfil androgenico y progestagenico mixto |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| USB337823I5 (https=) * | 1959-09-25 | 1976-03-23 | ||
| US3086027A (en) * | 1960-01-22 | 1963-04-16 | Lilly Co Eli | 19-nor-4, 9(10)-steroids and process |
| IE60780B1 (en) * | 1987-01-23 | 1994-08-10 | Akzo Nv | New 11-aryl steroid derivatives |
| US5264427A (en) * | 1992-01-29 | 1993-11-23 | Research Corporation Technologies, Inc. | 20-substituted pregnene derivatives and their use as androgen synthesis inhibitors |
| US6180682B1 (en) * | 1999-01-26 | 2001-01-30 | Virgil A. Place | Buccal drug delivery system for use in male contraception |
-
2000
- 2000-03-02 EP EP00909281A patent/EP1163259B1/en not_active Expired - Lifetime
- 2000-03-02 AT AT00909281T patent/ATE228143T1/de not_active IP Right Cessation
- 2000-03-02 AU AU31622/00A patent/AU3162200A/en not_active Abandoned
- 2000-03-02 WO PCT/EP2000/001755 patent/WO2000053619A1/en not_active Ceased
- 2000-03-02 US US09/890,845 patent/US6881728B1/en not_active Expired - Lifetime
- 2000-03-02 JP JP2000604054A patent/JP4749550B2/ja not_active Expired - Lifetime
- 2000-03-02 DE DE60000826T patent/DE60000826T2/de not_active Expired - Lifetime
- 2000-03-02 CA CA002359218A patent/CA2359218A1/en not_active Abandoned
- 2000-03-07 AR ARP000101000A patent/AR022852A1/es unknown
- 2000-03-07 PE PE2000000200A patent/PE20001489A1/es not_active Application Discontinuation
- 2000-03-08 CO CO00016933A patent/CO5150195A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP4749550B2 (ja) | 2011-08-17 |
| ATE228143T1 (de) | 2002-12-15 |
| DE60000826T2 (de) | 2003-04-10 |
| EP1163259A1 (en) | 2001-12-19 |
| CA2359218A1 (en) | 2000-09-14 |
| AU3162200A (en) | 2000-09-28 |
| US6881728B1 (en) | 2005-04-19 |
| JP2002539135A (ja) | 2002-11-19 |
| DE60000826D1 (de) | 2003-01-02 |
| CO5150195A1 (es) | 2002-04-29 |
| AR022852A1 (es) | 2002-09-04 |
| WO2000053619A1 (en) | 2000-09-14 |
| EP1163259B1 (en) | 2002-11-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Refusal |