OA12413A - Combination of GABA agonists and aldose reductase inhibitors. - Google Patents
Combination of GABA agonists and aldose reductase inhibitors. Download PDFInfo
- Publication number
- OA12413A OA12413A OA1200300138A OA1200300138A OA12413A OA 12413 A OA12413 A OA 12413A OA 1200300138 A OA1200300138 A OA 1200300138A OA 1200300138 A OA1200300138 A OA 1200300138A OA 12413 A OA12413 A OA 12413A
- Authority
- OA
- OAPI
- Prior art keywords
- prodrug
- gaba
- pharmaceutically acceptable
- pharmaceutical composition
- diabetic
- Prior art date
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- 239000003288 aldose reductase inhibitor Substances 0.000 title description 32
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Classifications
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- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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Landscapes
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- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| KR (1) | KR20030059287A (no) |
| CN (1) | CN1477976A (no) |
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| PT934061E (pt) | 1996-07-24 | 2003-10-31 | Warner Lambert Co | Isobutilgaba e seus derivados para o tratamento da dor |
| US6696407B1 (en) * | 1997-03-21 | 2004-02-24 | The Regents Of The University Of California | Huntington's disease treatment comprising administering aldose reductase inhibitors to increase striatal CNTF |
| US20030162754A1 (en) * | 2001-12-17 | 2003-08-28 | Tufts University | Use of GABA and GABAB agonists |
| AU2003243603A1 (en) * | 2002-06-13 | 2003-12-31 | Board Of Regents, The University Of Texas System | Methods and compositions involving aldose reductase inhibitors |
| WO2004054560A1 (en) * | 2002-12-13 | 2004-07-01 | Warner-Lambert Company Llc | Alpha-2-delta ligand to treat lower urinary tract symptoms |
| US20080318908A1 (en) * | 2002-12-17 | 2008-12-25 | Trustees Of Tufts College | Use of gaba and gabab agonists |
| MXPA05006656A (es) * | 2002-12-20 | 2006-02-22 | Dynogen Pharmaceuticals Inc | Metodos de tratamiento de desordenes de vejiga no dolorosos usando moduladores del canal de calcio subunidad (2o. |
| EP1721607A1 (en) * | 2003-03-21 | 2006-11-15 | Dynogen Pharmaceuticals, Inc. | Methods for treating lower urinary tract disorders using smooth muscle modulators and alpha-2-delta subunit calcium channel modulators |
| KR20050036195A (ko) * | 2003-10-15 | 2005-04-20 | 고재영 | 신규한 망막병증 치료제 조성물 |
| US20110092566A1 (en) * | 2004-11-19 | 2011-04-21 | Srivastava Satish K | Treatment of cancer with aldose reductase inhibitors |
| WO2007053596A1 (en) * | 2005-10-31 | 2007-05-10 | Braincells, Inc. | Gaba receptor mediated modulation of neurogenesis |
| BRPI0709961A2 (pt) | 2006-04-11 | 2011-08-02 | Novartis Ag | compostos orgánicos |
| JP2010513357A (ja) * | 2006-12-22 | 2010-04-30 | ノバルティス アーゲー | Ｄｐｐ−ｉｖ阻害剤としての１−アミノメチル−１−フェニル−シクロヘキサン誘導体 |
| EP2139330B1 (en) | 2007-03-23 | 2014-09-24 | The Board of Regents of The University of Texas System | Methods involving aldose reductase inhibitors |
| US20090270490A1 (en) * | 2008-04-24 | 2009-10-29 | The Board Of Regents Of The University Of Texas System | Methods involving aldose reductase inhibition |
| SG176464A1 (en) | 2008-05-09 | 2011-12-29 | Agency Science Tech & Res | Diagnosis and treatment of kawasaki disease |
| US9623000B2 (en) | 2008-07-31 | 2017-04-18 | Dekel Pharmaceuticals Ltd | Compositions and methods for treating inflammatory disorders |
| ES2639019T3 (es) * | 2008-09-06 | 2017-10-25 | Bionevia Pharmaceuticals Inc. | Nuevo cocristal de colina de epalrestat |
| EP2654749B1 (en) | 2010-12-23 | 2017-05-10 | The Board of Regents of The University of Texas System | Methods for treating copd |
| US8652527B1 (en) | 2013-03-13 | 2014-02-18 | Upsher-Smith Laboratories, Inc | Extended-release topiramate capsules |
| US9101545B2 (en) | 2013-03-15 | 2015-08-11 | Upsher-Smith Laboratories, Inc. | Extended-release topiramate capsules |
| CN107847548B (zh) * | 2015-05-18 | 2022-06-14 | 贝思以色列女会吏医学中心公司 | P物质、肥大细胞脱颗粒抑制剂和周围神经病 |
| WO2018195411A1 (en) * | 2017-04-21 | 2018-10-25 | Steven Hoffman | Compositions and methods for treating retinopathy |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| CA3138094A1 (en) | 2019-04-17 | 2020-10-22 | Compass Pathfinder Limited | Methods for treating anxiety disorders, headache disorders, and eating disorders with psilocybin |
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| CH449645A (de) | 1963-07-09 | 1968-01-15 | Ciba Geigy | Verfahren zur Herstellung neuer Aminosäuren |
| CH427803A (de) | 1963-12-06 | 1967-01-15 | Geigy Ag J R | Verfahren zur Herstellung eines neuen Isoxazolderivates |
| DE2460891C2 (de) * | 1974-12-21 | 1982-09-23 | Gödecke AG, 1000 Berlin | 1-Aminomethyl-1-cycloalkanessigsäuren und deren Ester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
| US3960927A (en) | 1975-03-18 | 1976-06-01 | Richardson-Merrell Inc. | Olefinic derivatives of amino acids |
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2001
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- 2001-11-19 HU HU0302555A patent/HUP0302555A3/hu unknown
- 2001-11-19 WO PCT/IB2001/002214 patent/WO2002043763A2/en not_active Application Discontinuation
- 2001-11-19 OA OA1200300138A patent/OA12413A/en unknown
- 2001-11-19 EA EA200300433A patent/EA200300433A1/ru unknown
- 2001-11-19 BR BR0115776-0A patent/BR0115776A/pt not_active IP Right Cessation
- 2001-11-19 CZ CZ20031387A patent/CZ20031387A3/cs unknown
- 2001-11-19 SK SK609-2003A patent/SK6092003A3/sk not_active Application Discontinuation
- 2001-11-19 PL PL01365378A patent/PL365378A1/xx not_active Application Discontinuation
- 2001-11-19 EP EP01983740A patent/EP1337272A2/en not_active Withdrawn
- 2001-11-19 AP APAP/P/2001/002359A patent/AP2001002359A0/en unknown
- 2001-11-19 CN CNA018195954A patent/CN1477976A/zh active Pending
- 2001-11-19 JP JP2002545733A patent/JP2004514700A/ja not_active Withdrawn
- 2001-11-19 EE EEP200300249A patent/EE200300249A/xx unknown
- 2001-11-19 AU AU2002215160A patent/AU2002215160A1/en not_active Abandoned
- 2001-11-19 CA CA002430309A patent/CA2430309A1/en not_active Abandoned
- 2001-11-19 KR KR10-2003-7007221A patent/KR20030059287A/ko not_active Application Discontinuation
- 2001-11-26 DO DO2001000294A patent/DOP2001000294A/es unknown
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- 2001-11-28 AR ARP010105542A patent/AR031432A1/es not_active Application Discontinuation
- 2001-11-29 TN TNTNSN01170A patent/TNSN01170A1/fr unknown
- 2001-11-29 US US09/997,039 patent/US6720348B2/en not_active Expired - Fee Related
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2003
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- 2003-05-22 HR HR20030419A patent/HRP20030419A2/hr not_active Application Discontinuation
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