OA12061A - Pyrazolo Ä4,3-DÜpyrimidine derivatives. - Google Patents

Pyrazolo Ä4,3-DÜpyrimidine derivatives. Download PDF

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Publication number
OA12061A
OA12061A OA1200200104A OA1200200104A OA12061A OA 12061 A OA12061 A OA 12061A OA 1200200104 A OA1200200104 A OA 1200200104A OA 1200200104 A OA1200200104 A OA 1200200104A OA 12061 A OA12061 A OA 12061A
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OA
OAPI
Prior art keywords
group
compound
alkyl
formula
ethyl
Prior art date
Application number
OA1200200104A
Other languages
English (en)
Inventor
Mark Edward Bunnage
Keith Michael Devries
Laurence James Harris
Philip Charles Levett
John Paul Mathias
Joanna Teresa Negri
Stephen Derek Albert Street
Albert Shaw Wood
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26244757&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA12061(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9924063.2A external-priority patent/GB9924063D0/en
Priority claimed from GB0018656A external-priority patent/GB0018656D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of OA12061A publication Critical patent/OA12061A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/80—Acids; Esters in position 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pregnancy & Childbirth (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Otolaryngology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
OA1200200104A 1999-10-11 2000-10-11 Pyrazolo Ä4,3-DÜpyrimidine derivatives. OA12061A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9924063.2A GB9924063D0 (en) 1999-10-11 1999-10-11 Pharmaceutically active compounds
GB0018656A GB0018656D0 (en) 2000-07-28 2000-07-28 Pharmaceutically active compounds

Publications (1)

Publication Number Publication Date
OA12061A true OA12061A (en) 2006-05-03

Family

ID=26244757

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200200104A OA12061A (en) 1999-10-11 2000-10-11 Pyrazolo Ä4,3-DÜpyrimidine derivatives.

Country Status (48)

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US (4) US6677335B1 (is")
EP (1) EP1220856B1 (is")
JP (1) JP3834236B2 (is")
KR (1) KR100549152B1 (is")
CN (3) CN100383141C (is")
AP (1) AP1238A (is")
AT (1) ATE284404T1 (is")
AU (1) AU779065B2 (is")
BG (1) BG106678A (is")
BR (1) BR0014698A (is")
CA (1) CA2387357C (is")
CO (1) CO5251477A1 (is")
CR (2) CR6617A (is")
CU (1) CU23198A3 (is")
CZ (1) CZ20021158A3 (is")
DE (1) DE60016615T2 (is")
DK (1) DK1220856T3 (is")
DZ (1) DZ3220A1 (is")
EA (1) EA004982B1 (is")
EE (1) EE05181B1 (is")
EG (1) EG24411A (is")
ES (1) ES2232502T3 (is")
GE (2) GEP20033142B (is")
GT (1) GT200000171A (is")
HR (1) HRP20020317B1 (is")
HU (1) HUP0203450A3 (is")
IL (2) IL149026A0 (is")
IN (4) IN2002MU00385A (is")
IS (1) IS2181B (is")
MA (1) MA26825A1 (is")
MX (1) MX228340B (is")
MY (1) MY130319A (is")
NO (1) NO322856B1 (is")
NZ (1) NZ518078A (is")
OA (1) OA12061A (is")
PA (1) PA8504501A1 (is")
PE (1) PE20010737A1 (is")
PH (1) PH12000002783B1 (is")
PL (1) PL357536A1 (is")
PT (1) PT1220856E (is")
RS (1) RS50476B (is")
SI (1) SI1220856T1 (is")
SK (1) SK4602002A3 (is")
SV (1) SV2002000195A (is")
TN (1) TNSN00199A1 (is")
TR (1) TR200200989T2 (is")
TW (1) TWI265925B (is")
WO (1) WO2001027113A2 (is")

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