OA06263A - Dérivés acylés. - Google Patents

Dérivés acylés.

Info

Publication number
OA06263A
OA06263A OA56816A OA56816A OA06263A OA 06263 A OA06263 A OA 06263A OA 56816 A OA56816 A OA 56816A OA 56816 A OA56816 A OA 56816A OA 06263 A OA06263 A OA 06263A
Authority
OA
OAPI
Prior art keywords
triazin
methyl
group
acylated derivatives
dioxo
Prior art date
Application number
OA56816A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH588278A external-priority patent/CH641468A5/de
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of OA06263A publication Critical patent/OA06263A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Mutual Connection Of Rods And Tubes (AREA)
  • Reinforcement Elements For Buildings (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
OA56816A 1978-05-30 1979-05-29 Dérivés acylés. OA06263A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH588278A CH641468A5 (de) 1978-05-30 1978-05-30 Cephemderivate.
CH224879 1979-03-08

Publications (1)

Publication Number Publication Date
OA06263A true OA06263A (fr) 1981-06-30

Family

ID=25689901

Family Applications (1)

Application Number Title Priority Date Filing Date
OA56816A OA06263A (fr) 1978-05-30 1979-05-29 Dérivés acylés.

Country Status (40)

Country Link
EP (2) EP0045525B1 (fr)
JP (2) JPS54157596A (fr)
AT (3) AT367764B (fr)
BG (1) BG50163A3 (fr)
BR (1) BR7903368A (fr)
CA (1) CA1141373A (fr)
CS (1) CS219254B2 (fr)
CU (1) CU35088A (fr)
CY (1) CY1182A (fr)
DD (1) DD143911A5 (fr)
DE (4) DE2966946D1 (fr)
DK (1) DK149282C (fr)
EG (1) EG14153A (fr)
ES (2) ES480990A1 (fr)
FI (1) FI65434C (fr)
FR (2) FR2427337A1 (fr)
GB (2) GB2099418B (fr)
GR (1) GR72242B (fr)
HK (1) HK31383A (fr)
HU (1) HU183089B (fr)
IE (1) IE49047B1 (fr)
IL (1) IL57392A (fr)
IS (1) IS1203B6 (fr)
IT (1) IT1121517B (fr)
KE (1) KE3268A (fr)
LU (1) LU81325A1 (fr)
MC (1) MC1259A1 (fr)
MT (1) MTP845B (fr)
MY (1) MY8400127A (fr)
NL (1) NL7904083A (fr)
NO (1) NO159797C (fr)
NZ (1) NZ190532A (fr)
OA (1) OA06263A (fr)
PH (1) PH15148A (fr)
PL (1) PL122458B1 (fr)
PT (1) PT69698A (fr)
RO (1) RO77560A (fr)
SE (1) SE437522B (fr)
SG (1) SG10483G (fr)
YU (3) YU42485B (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI67385C (fi) * 1979-11-21 1985-03-11 Hoffmann La Roche Foerfarande foer framstaellning av (6r 7r)-7-(2-(2-amino-4-tiazolyl)-2-(z-metoxiimino)acetamido)-3-cefem-4-karboxylsyraderivat
US4349672A (en) * 1979-11-29 1982-09-14 Hoffmann-La Roche Inc. Cephalosporin derivatives
NZ196552A (en) * 1980-03-25 1984-07-06 Hoffmann La Roche Cephalosporin derivatives and pharmaceutical compositions;intermediate cephalosporins
CA1154009A (fr) * 1980-03-25 1983-09-20 Roland Reiner Derives de cephalosporine
GR75706B (fr) * 1980-06-30 1984-08-02 Sanofi Sa
US4308267A (en) 1980-07-03 1981-12-29 Smithkline Corporation 7-[2-Alkoxyimino-2-(amino-thiazole)acetamido]-3-[1-(sulfaminoalkly)tetrazolthiomethyl]cephalosporins
DK379581A (da) * 1980-10-06 1982-04-07 Hoffmann La Roche Fremgangsmaade til fremstilling af acylderivater
FR2494278A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de la cephalosporine, leurs preparations et les medicaments qui les contiennent
EP0058250A3 (fr) * 1981-02-17 1983-08-17 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Dérivés de céphalosporine, leur préparation et compositions pharmaceutiques les contenant
EP0185220A3 (fr) * 1984-12-19 1987-09-02 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Intermédiaires pour la préparation de céphalosporines
CA1296012C (fr) 1986-03-19 1992-02-18 Susumu Nakagawa Derives de 6,7-dihydroxy-isoquinaline
RU2021274C1 (ru) 1991-05-17 1994-10-15 Польска Акадэмия Наук Институт Хэмии Органичнэй Способ получения аминотиазолильных производных цефалоспорина
KR950014571B1 (ko) * 1991-11-18 1995-12-08 제일제당주식회사 세펨 유도체의 제조방법
AT398764B (de) * 1992-01-28 1995-01-25 Lek Tovarna Farmacevtskih Verfahren zur herstellung von ceftriaxondinatrium-salzhemiheptahydrat
AT399877B (de) * 1992-02-20 1995-08-25 Biochemie Gmbh Neues verfahren zur herstellung von ceftriaxon
KR100197788B1 (ko) * 1995-06-30 1999-06-15 김충환 세펨 유도체의 제조방법
DE102011117421A1 (de) 2011-11-02 2013-05-02 Hans-Peter Gabel Pharmazeutische Zusammensetzung zur Behandlung von Borreliose
RU2504548C1 (ru) * 2012-09-28 2014-01-20 Федеральное Государственное Автономное Образовательное Учреждение Высшего Профессионального Образования "Сибирский Федеральный Университет" (Сфу) ПРОИЗВОДНОЕ β-ЛАКТАМНОГО АНТИБИОТИКА ЦЕФТРИАКСОНА

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH609989A5 (en) * 1974-06-21 1979-03-30 Hoffmann La Roche Process for the preparation of acyl derivatives
CA1100129A (fr) * 1974-08-02 1981-04-28 William H.W. Lunn Traduction non-disponible
FR2345153A1 (fr) * 1976-03-25 1977-10-21 Roussel Uclaf Nouvelles alcoyloximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
DK162391C (da) * 1976-04-12 1992-03-09 Fujisawa Pharmaceutical Co Analogifremgangsmaade til fremstilling af syn-isomerer af 3,7-disubstituerede 3-cephem-4-carboxylsyreforbindelser
GR63088B (en) * 1976-04-14 1979-08-09 Takeda Chemical Industries Ltd Preparation process of novel cephalosporins
JPS5329936A (en) * 1976-08-31 1978-03-20 Takeda Chem Ind Ltd Antibiotic composition
NL7805715A (nl) * 1977-06-03 1978-12-05 Hoffmann La Roche Werkwijze voor het bereiden van acylderivaten.
US4200745A (en) * 1977-12-20 1980-04-29 Eli Lilly And Company 7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins

Also Published As

Publication number Publication date
MC1259A1 (fr) 1980-01-14
JPS54157596A (en) 1979-12-12
LU81325A1 (de) 1980-12-16
JPS6016994A (ja) 1985-01-28
YU42485B (en) 1988-10-31
GB2022090B (en) 1982-12-15
AT367764B (de) 1982-07-26
IL57392A0 (en) 1979-09-30
ATE7229T1 (de) 1984-05-15
DK149282C (da) 1986-09-01
AU4736679A (en) 1979-12-06
FR2509312B1 (fr) 1984-06-29
IS1203B6 (is) 1986-03-24
DD143911A5 (de) 1980-09-17
ES480990A1 (es) 1980-08-16
EP0045525A2 (fr) 1982-02-10
DK222679A (da) 1979-12-01
SE7904682L (sv) 1979-12-01
YU123379A (en) 1983-04-30
GR72242B (fr) 1983-10-04
NO159797B (no) 1988-10-31
FR2509312A1 (fr) 1983-01-14
GB2022090A (en) 1979-12-12
DK149282B (da) 1986-04-21
CA1141373A (fr) 1983-02-15
NL7904083A (nl) 1979-12-04
JPS613795B2 (fr) 1986-02-04
KE3268A (en) 1983-05-13
EP0005830A1 (fr) 1979-12-12
ATA390479A (de) 1981-12-15
DE2922036C2 (de) 1983-02-17
FR2427337A1 (fr) 1979-12-28
SG10483G (en) 1983-12-16
HK31383A (en) 1983-09-02
BR7903368A (pt) 1979-12-11
JPS613355B2 (fr) 1986-01-31
NZ190532A (en) 1983-03-15
IT7923049A0 (it) 1979-05-28
PL122458B1 (en) 1982-07-31
YU45257B (en) 1992-05-28
EG14153A (en) 1983-03-31
IS2490A7 (is) 1979-12-01
DE2963720D1 (en) 1982-11-04
DE2954159C2 (de) 1983-10-06
FI65434C (fi) 1984-05-10
ES488687A0 (es) 1980-12-16
FI791703A (fi) 1979-12-01
PL215972A1 (fr) 1980-02-11
ES8101606A1 (es) 1980-12-16
DE2922036A1 (de) 1979-12-06
CU35088A (en) 1982-08-24
ATE1586T1 (de) 1982-10-15
NO791776L (no) 1979-12-03
EP0005830B1 (fr) 1982-09-22
EP0045525A3 (en) 1982-02-17
CY1182A (en) 1983-10-07
HU183089B (en) 1984-04-28
PT69698A (en) 1979-06-01
MY8400127A (en) 1984-12-31
FI65434B (fi) 1984-01-31
IL57392A (en) 1982-05-31
GB2099418B (en) 1983-06-02
YU45256B (en) 1992-05-28
AU524230B2 (en) 1982-09-09
PH15148A (en) 1982-08-24
RO77560A (fr) 1982-04-12
SE437522B (sv) 1985-03-04
CS219254B2 (en) 1983-03-25
IT1121517B (it) 1986-04-02
NO159797C (no) 1989-02-08
GB2099418A (en) 1982-12-08
MTP845B (en) 1980-07-21
DE2966946D1 (en) 1984-05-30
EP0045525B1 (fr) 1984-04-25
BG50163A3 (en) 1992-05-15
IE791041L (en) 1979-11-30
YU74585A (en) 1987-12-31
YU74485A (en) 1987-12-31
IE49047B1 (en) 1985-07-24

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Publication Publication Date Title
OA06263A (fr) Dérivés acylés.