NZ741907A - 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof - Google Patents

1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof

Info

Publication number
NZ741907A
NZ741907A NZ741907A NZ74190713A NZ741907A NZ 741907 A NZ741907 A NZ 741907A NZ 741907 A NZ741907 A NZ 741907A NZ 74190713 A NZ74190713 A NZ 74190713A NZ 741907 A NZ741907 A NZ 741907A
Authority
NZ
New Zealand
Prior art keywords
pyridin
pyrazolo
compound
disclosed
pyridines
Prior art date
Application number
NZ741907A
Other languages
English (en)
Inventor
John Hood
Sunil Kumar Kc
David Mark Wallace
Original Assignee
Samumed Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Samumed Llc filed Critical Samumed Llc
Publication of NZ741907A publication Critical patent/NZ741907A/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dispersion Chemistry (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
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NZ741907A 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof NZ741907A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261642915P 2012-05-04 2012-05-04
NZ724837A NZ724837A (en) 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof

Publications (1)

Publication Number Publication Date
NZ741907A true NZ741907A (en) 2020-02-28

Family

ID=49513001

Family Applications (3)

Application Number Title Priority Date Filing Date
NZ741907A NZ741907A (en) 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
NZ629282A NZ629282A (en) 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
NZ724837A NZ724837A (en) 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof

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NZ629282A NZ629282A (en) 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
NZ724837A NZ724837A (en) 2012-05-04 2013-05-03 1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof

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Country Link
US (8) US8883822B2 (enExample)
EP (2) EP3593800A1 (enExample)
JP (3) JP6209593B2 (enExample)
KR (1) KR102223301B1 (enExample)
CN (2) CN107417707A (enExample)
AU (2) AU2013256141B2 (enExample)
BR (1) BR112014024284B1 (enExample)
CA (1) CA2854229C (enExample)
CL (1) CL2014002983A1 (enExample)
CO (1) CO7170178A2 (enExample)
CY (1) CY1122703T1 (enExample)
DK (1) DK2770994T3 (enExample)
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MA (1) MA37577B1 (enExample)
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MX (1) MX362466B (enExample)
MY (1) MY173049A (enExample)
NZ (3) NZ741907A (enExample)
PE (1) PE20142365A1 (enExample)
PH (3) PH12014502369B1 (enExample)
PL (1) PL2770994T3 (enExample)
PT (1) PT2770994T (enExample)
RS (1) RS59668B1 (enExample)
RU (1) RU2689141C2 (enExample)
SG (2) SG11201407148XA (enExample)
SI (1) SI2770994T1 (enExample)
SM (1) SMT201900618T1 (enExample)
WO (1) WO2013166396A2 (enExample)
ZA (2) ZA201406274B (enExample)

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BR112012002854B1 (pt) 2009-08-10 2020-02-18 Samumed, Llc Composto ou sal farmaceuticamente aceitável, composição farmacêutica e uso dos mesmos
US8450340B2 (en) 2009-12-21 2013-05-28 Samumed, Llc 1H-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
US9442092B2 (en) 2011-06-20 2016-09-13 Kerry Lane Methods for treatment of autism
ES2711777T3 (es) 2011-09-14 2019-05-07 Samumed Llc Indazol-3-carboxamidas y su uso como inhibidores de la ruta de señalización de Wnt/b-catenina
PH12017500997A1 (en) 2012-04-04 2018-02-19 Samumed Llc Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof
SI2770994T1 (sl) 2012-05-04 2020-02-28 Samumed, Llc 1H-pirazolo(3,4-B)piridini in njihove terapevtske uporabe
WO2014110086A2 (en) 2013-01-08 2014-07-17 Samumed, Llc 3-(benzoimidazol-2-yl)-indazole inhibitors of the wnt signaling pathway and therapeutic uses thereof
SI3080100T1 (sl) 2013-12-11 2023-04-28 Celgene Quanticel Research, Inc. Inhibitorji lizin specifične demetilaze-1
AU2015236855B2 (en) * 2014-03-27 2018-11-01 Cancer Research Technology Limited Pyridyl piperidines
WO2016040180A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-benzo[d]imidazol-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
WO2016040190A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
WO2016040182A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 2-(1h-indazol-3-yl)-1h-imidazo[4,5-c]pyridine and therapeutic uses thereof
WO2016040184A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
WO2016040181A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
WO2016040185A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 2-(1h-indazol-3-yl)-3h-imidazo[4,5-b]pyridine and therapeutic uses thereof
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JP7630905B2 (ja) 2016-11-07 2025-02-18 バイオスプライス セラピューティクス インコーポレイテッド 単回用量の調整済み注射用製剤

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