NO983074L - Karbamoyloksyderivater av mutilin og deres anvendelse som antibakterielle midler - Google Patents

Karbamoyloksyderivater av mutilin og deres anvendelse som antibakterielle midler

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Publication number
NO983074L
NO983074L NO983074A NO983074A NO983074L NO 983074 L NO983074 L NO 983074L NO 983074 A NO983074 A NO 983074A NO 983074 A NO983074 A NO 983074A NO 983074 L NO983074 L NO 983074L
Authority
NO
Norway
Prior art keywords
mutilin
antibacterial agents
derivatives
carbamoyloxy derivatives
carbamoyloxy
Prior art date
Application number
NO983074A
Other languages
English (en)
Norwegian (no)
Other versions
NO983074D0 (no
Inventor
Jeremy David Hinks
Andrew Kenneth Takle
Eric Hunt
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9600048.4A external-priority patent/GB9600048D0/en
Priority claimed from GBGB9616305.0A external-priority patent/GB9616305D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of NO983074D0 publication Critical patent/NO983074D0/no
Publication of NO983074L publication Critical patent/NO983074L/no

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    • C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D203/08—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
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    • C07C271/36—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of rings other than six-membered aromatic rings with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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    • C07C271/62—Compounds containing any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylcarbamates
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    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
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    • C07C331/00—Derivatives of thiocyanic acid or of isothiocyanic acid
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    • C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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NO983074A 1996-01-03 1998-07-02 Karbamoyloksyderivater av mutilin og deres anvendelse som antibakterielle midler NO983074L (no)

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GBGB9600048.4A GB9600048D0 (en) 1996-01-03 1996-01-03 Novel compounds
GBGB9616305.0A GB9616305D0 (en) 1996-08-02 1996-08-02 Novel compounds
PCT/EP1996/005874 WO1997025309A1 (fr) 1996-01-03 1996-12-19 Derives carbamoyloxy de mutiline et leur utilisation en tant qu'agents antibacteriens

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MX9805416A (es) 1998-10-31
TR199801282T2 (xx) 1998-12-21
CN1214039A (zh) 1999-04-14
US6020368A (en) 2000-02-01
HUP9900973A2 (hu) 1999-08-30
AP9801283A0 (en) 1998-09-30
HUP9900973A3 (en) 2000-04-28
US6239175B1 (en) 2001-05-29
NZ325837A (en) 1999-11-29
NO983074D0 (no) 1998-07-02
PL327737A1 (en) 1998-12-21
CZ212498A3 (cs) 1998-12-16
SK91098A3 (en) 1999-02-11
EP0874809B1 (fr) 2003-08-27
KR19990076988A (ko) 1999-10-25
IL124912A0 (en) 1999-01-26
ATE248143T1 (de) 2003-09-15
JP4163254B2 (ja) 2008-10-08
AR005357A1 (es) 1999-04-28
CA2240467A1 (fr) 1997-07-17
BG102600A (en) 1999-09-30
DE69629721D1 (de) 2003-10-02
AU1307897A (en) 1997-08-01
ES2205072T3 (es) 2004-05-01
EP0874809A1 (fr) 1998-11-04
DE69629721T2 (de) 2004-06-09
BR9612426A (pt) 1999-07-13
OA10708A (en) 2002-11-28
WO1997025309A1 (fr) 1997-07-17
EA199800525A1 (ru) 1999-02-25
AU715229B2 (en) 2000-01-20

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