NO981911D0 - Anvendelse av rhodaninderivater for fremstilling av et medikament for behandling av Alzheimer's sykdom - Google Patents
Anvendelse av rhodaninderivater for fremstilling av et medikament for behandling av Alzheimer's sykdomInfo
- Publication number
- NO981911D0 NO981911D0 NO981911A NO981911A NO981911D0 NO 981911 D0 NO981911 D0 NO 981911D0 NO 981911 A NO981911 A NO 981911A NO 981911 A NO981911 A NO 981911A NO 981911 D0 NO981911 D0 NO 981911D0
- Authority
- NO
- Norway
- Prior art keywords
- alzheimer
- medicament
- disease
- manufacture
- treatment
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/14—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/34—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/36—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
- B65H—HANDLING THIN OR FILAMENTARY MATERIAL, e.g. SHEETS, WEBS, CABLES
- B65H2511/00—Dimensions; Position; Numbers; Identification; Occurrences
- B65H2511/50—Occurence
- B65H2511/51—Presence
- B65H2511/512—Marks, e.g. invisible to the human eye; Patterns
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US94335392A | 1992-09-10 | 1992-09-10 |
Publications (2)
Publication Number | Publication Date |
---|---|
NO981911L NO981911L (no) | 1994-03-11 |
NO981911D0 true NO981911D0 (no) | 1998-04-28 |
Family
ID=25479507
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO933198A NO933198L (no) | 1992-09-10 | 1993-09-08 | Forbindelser anvendelige som hypoglycemiske midler og for behandling av Alzheimer's sykdom |
NO981911A NO981911D0 (no) | 1992-09-10 | 1998-04-28 | Anvendelse av rhodaninderivater for fremstilling av et medikament for behandling av Alzheimer's sykdom |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO933198A NO933198L (no) | 1992-09-10 | 1993-09-08 | Forbindelser anvendelige som hypoglycemiske midler og for behandling av Alzheimer's sykdom |
Country Status (20)
Country | Link |
---|---|
US (3) | US5523314A (no) |
EP (2) | EP0587377A3 (no) |
JP (1) | JPH06192091A (no) |
KR (1) | KR940006590A (no) |
CN (1) | CN1091006A (no) |
AU (1) | AU676843B2 (no) |
CA (1) | CA2105598A1 (no) |
CZ (1) | CZ181493A3 (no) |
FI (1) | FI933946A (no) |
HU (1) | HUT70184A (no) |
IL (1) | IL106877A (no) |
MX (1) | MX9305444A (no) |
MY (1) | MY131443A (no) |
NO (2) | NO933198L (no) |
NZ (1) | NZ248573A (no) |
PL (1) | PL300335A1 (no) |
RU (1) | RU2131251C1 (no) |
TW (1) | TW274546B (no) |
YU (1) | YU59593A (no) |
ZA (1) | ZA936492B (no) |
Families Citing this family (85)
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US6251928B1 (en) * | 1994-03-16 | 2001-06-26 | Eli Lilly And Company | Treatment of alzheimer's disease employing inhibitors of cathepsin D |
DE69530501D1 (de) * | 1994-10-20 | 2003-05-28 | Nippon Chemiphar Co | Chinolinderivat |
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IL117208A0 (en) * | 1995-02-23 | 1996-06-18 | Nissan Chemical Ind Ltd | Indole type thiazolidines |
US5783434A (en) * | 1995-06-06 | 1998-07-21 | Tung; Jay S. | Cathepsin and methods and compositions for inhibition thereof |
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ATE250416T1 (de) * | 1996-07-11 | 2003-10-15 | Warner Lambert Co | Verfahren zur behandlung und vorbeugung von neurodegenerativen erkrankungen durch verabreichung von einem thiazolidin |
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DE19641180A1 (de) * | 1996-09-24 | 1998-03-26 | Schering Ag | Verfahren zur Darstellung von APP-Sekretase Modulation und deren Verwendung als Mittel zur Behandlung der Alzheimer'schen Erkrankung |
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DE69825605T2 (de) | 1997-05-29 | 2005-09-15 | H. Lundbeck A/S | Behandlung der schizophrenie und der psychose |
US20040058873A1 (en) * | 1998-03-12 | 2004-03-25 | Esmond Robert W. | Method for treating or preventing Alzheimer's disease |
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WO2000018747A1 (en) * | 1998-09-30 | 2000-04-06 | Roche Diagnostics Gmbh | Rhodanine carboxylic acid derivatives for the treatment and prevention of metabolic bone disorders |
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-
1993
- 1993-09-02 ZA ZA936492A patent/ZA936492B/xx unknown
- 1993-09-02 IL IL106877A patent/IL106877A/en not_active IP Right Cessation
- 1993-09-02 EP EP19930306959 patent/EP0587377A3/en not_active Withdrawn
- 1993-09-02 NZ NZ248573A patent/NZ248573A/en unknown
- 1993-09-02 CZ CZ931814A patent/CZ181493A3/cs unknown
- 1993-09-02 EP EP98201389A patent/EP0915090A1/en not_active Withdrawn
- 1993-09-03 TW TW082107213A patent/TW274546B/zh active
- 1993-09-06 MX MX9305444A patent/MX9305444A/es unknown
- 1993-09-07 MY MYPI93001815A patent/MY131443A/en unknown
- 1993-09-07 CA CA002105598A patent/CA2105598A1/en not_active Abandoned
- 1993-09-08 HU HU9302551A patent/HUT70184A/hu unknown
- 1993-09-08 RU RU93051176A patent/RU2131251C1/ru active
- 1993-09-08 NO NO933198A patent/NO933198L/no unknown
- 1993-09-08 AU AU46218/93A patent/AU676843B2/en not_active Ceased
- 1993-09-09 CN CN93119081A patent/CN1091006A/zh active Pending
- 1993-09-09 JP JP5224434A patent/JPH06192091A/ja not_active Withdrawn
- 1993-09-09 PL PL93300335A patent/PL300335A1/xx unknown
- 1993-09-09 KR KR1019930018138A patent/KR940006590A/ko not_active Application Discontinuation
- 1993-09-09 FI FI933946A patent/FI933946A/fi unknown
- 1993-09-15 YU YU59593A patent/YU59593A/sh unknown
-
1994
- 1994-03-16 US US08/213,651 patent/US5523314A/en not_active Expired - Fee Related
-
1995
- 1995-06-06 US US08/470,822 patent/US5716975A/en not_active Expired - Fee Related
-
1996
- 1996-07-10 US US08/678,015 patent/US5661168A/en not_active Expired - Fee Related
-
1998
- 1998-04-28 NO NO981911A patent/NO981911D0/no unknown
Also Published As
Publication number | Publication date |
---|---|
RU2131251C1 (ru) | 1999-06-10 |
IL106877A0 (en) | 1993-12-28 |
AU4621893A (en) | 1994-03-17 |
TW274546B (no) | 1996-04-21 |
EP0587377A2 (en) | 1994-03-16 |
HU9302551D0 (en) | 1993-11-29 |
NO981911L (no) | 1994-03-11 |
FI933946A (fi) | 1994-03-11 |
US5661168A (en) | 1997-08-26 |
US5716975A (en) | 1998-02-10 |
KR940006590A (ko) | 1994-04-25 |
CA2105598A1 (en) | 1994-03-11 |
ZA936492B (en) | 1995-03-02 |
JPH06192091A (ja) | 1994-07-12 |
IL106877A (en) | 1998-03-10 |
US5523314A (en) | 1996-06-04 |
NO933198L (no) | 1994-03-11 |
EP0915090A1 (en) | 1999-05-12 |
EP0587377A3 (en) | 1994-09-21 |
PL300335A1 (en) | 1994-03-21 |
NZ248573A (en) | 1996-02-27 |
AU676843B2 (en) | 1997-03-27 |
MX9305444A (es) | 1994-05-31 |
YU59593A (sh) | 1997-01-08 |
HUT70184A (en) | 1995-09-28 |
CZ181493A3 (en) | 1994-03-16 |
CN1091006A (zh) | 1994-08-24 |
NO933198D0 (no) | 1993-09-08 |
FI933946A0 (fi) | 1993-09-09 |
MY131443A (en) | 2007-08-30 |
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