NO964348L - CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner - Google Patents

CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner

Info

Publication number
NO964348L
NO964348L NO964348A NO964348A NO964348L NO 964348 L NO964348 L NO 964348L NO 964348 A NO964348 A NO 964348A NO 964348 A NO964348 A NO 964348A NO 964348 L NO964348 L NO 964348L
Authority
NO
Norway
Prior art keywords
gastrin
cck
benzodiazepines
modulating
heterocyclic
Prior art date
Application number
NO964348A
Other languages
English (en)
Norwegian (no)
Other versions
NO964348D0 (no
Inventor
Christopher Joseph Aquino
Elisabeth Ellen Sugg
Jerzy Ryszard Szewczyk
Original Assignee
Glaxo Wellcome Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB9407433A external-priority patent/GB9407433D0/en
Priority claimed from GB9420783A external-priority patent/GB9420783D0/en
Application filed by Glaxo Wellcome Inc filed Critical Glaxo Wellcome Inc
Publication of NO964348D0 publication Critical patent/NO964348D0/no
Publication of NO964348L publication Critical patent/NO964348L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0821Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
NO964348A 1994-04-14 1996-10-11 CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner NO964348L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9407433A GB9407433D0 (en) 1994-04-14 1994-04-14 Heterocyclic derivatives
GB9420783A GB9420783D0 (en) 1994-10-14 1994-10-14 Heterocyclic derivatives
PCT/US1995/004163 WO1995028419A1 (en) 1994-04-14 1995-04-12 Cck or gastrin modulating 5-heterocyclic-1,5-benzodiazepines

Publications (2)

Publication Number Publication Date
NO964348D0 NO964348D0 (no) 1996-10-11
NO964348L true NO964348L (no) 1996-12-02

Family

ID=26304703

Family Applications (1)

Application Number Title Priority Date Filing Date
NO964348A NO964348L (no) 1994-04-14 1996-10-11 CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner

Country Status (25)

Country Link
EP (1) EP0756602B1 (is)
JP (1) JPH09511223A (is)
KR (1) KR970702274A (is)
CN (1) CN1176646A (is)
AT (1) ATE181737T1 (is)
AU (1) AU697349B2 (is)
BR (1) BR9507381A (is)
CA (1) CA2186900A1 (is)
CZ (1) CZ286764B6 (is)
DE (1) DE69510545T2 (is)
DK (1) DK0756602T3 (is)
ES (1) ES2135722T3 (is)
FI (1) FI964045A7 (is)
GR (1) GR3031335T3 (is)
HU (1) HUT76135A (is)
IL (1) IL113365A (is)
IS (1) IS4367A (is)
MX (1) MX9604765A (is)
NO (1) NO964348L (is)
NZ (1) NZ283929A (is)
PL (1) PL180026B1 (is)
RU (1) RU2152939C1 (is)
SK (1) SK281433B6 (is)
TW (1) TW369529B (is)
WO (1) WO1995028419A1 (is)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9307833D0 (en) * 1993-04-15 1993-06-02 Glaxo Inc Modulators of cholecystokinin and gastrin
PE27497A1 (es) * 1994-04-15 1997-08-07 Glaxo Inc Derivados de 1,5 benzodiazepina
EP0945445B9 (en) * 1996-12-10 2005-12-28 Zeria Pharmaceutical Co., Ltd. 1,5-benzodiazepine derivatives
US7910548B2 (en) * 1997-06-06 2011-03-22 Amylin Pharmaceuticals, Inc. Methods for treating obesity
EP1123928A4 (en) * 1998-10-20 2005-02-16 Takeda Pharmaceutical 1,5-BENZODIAZEPINE COMPOUNDS, PROCESS FOR PRODUCING THE SAME, AND MEDICAMENT
JP4535350B2 (ja) * 1998-11-17 2010-09-01 クミアイ化学工業株式会社 ピリミジニルベンズイミダゾール誘導体及び農園芸用殺菌剤
ATE402700T1 (de) * 2002-08-27 2008-08-15 Merck Patent Gmbh Glycinamid-derivate als raf-kinase-hemmer
JP4069159B2 (ja) 2004-05-25 2008-04-02 ファイザー・プロダクツ・インク テトラアザベンゾ[e]アズレン誘導体及びそれらのアナログ
RU2303597C1 (ru) * 2006-05-12 2007-07-27 Иващенко Андрей Александрович Фармацевтическая композиция, способы ее получения и применения
CN111333588A (zh) 2012-01-13 2020-06-26 日本化学药品株式会社 P2x4受体拮抗剂
CN118994191A (zh) 2016-02-05 2024-11-22 戴纳立制药公司 受体相互作用蛋白激酶1的抑制剂
HRP20220636T1 (hr) 2016-12-09 2022-07-22 Denali Therapeutics Inc. Spojevi korisni kao inhibitori ripk1
WO2021071837A1 (en) 2019-10-07 2021-04-15 Kallyope, Inc. Gpr119 agonists
BR112022017039A2 (pt) 2020-02-28 2022-11-16 Kallyope Inc Agonistas de gpr40
AU2023206890A1 (en) 2022-01-12 2024-08-22 Denali Therapeutics Inc. Crystalline forms of (s)-5-benzyl-n-(5-methyl-4-oxo-2, 3,4,5- tetrahydropyrido [3,2-b] [l,4]oxazepin-3-yl)-4h-l,2,4-triazole-3-carboxamide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2641280B1 (fr) * 1988-12-29 1994-01-21 Roussel Uclaf Nouveaux derives de la 2,4-dioxo 2,3,4,5-tetrahydro 1h-1,5-benzodiazepine, leur procede de preparation et leur application comme medicaments
GB9201180D0 (en) * 1992-01-21 1992-03-11 Glaxo Group Ltd Chemical compounds
GB9307833D0 (en) * 1993-04-15 1993-06-02 Glaxo Inc Modulators of cholecystokinin and gastrin

Also Published As

Publication number Publication date
DK0756602T3 (da) 2000-01-31
NO964348D0 (no) 1996-10-11
IS4367A (is) 1996-09-30
TW369529B (en) 1999-09-11
DE69510545T2 (de) 2000-01-13
MX9604765A (es) 1998-05-31
SK281433B6 (sk) 2001-03-12
HUT76135A (en) 1997-06-30
FI964045A0 (fi) 1996-10-09
CN1176646A (zh) 1998-03-18
DE69510545D1 (de) 1999-08-05
FI964045L (fi) 1996-10-09
BR9507381A (pt) 1997-09-23
WO1995028419A1 (en) 1995-10-26
KR970702274A (ko) 1997-05-13
PL316870A1 (en) 1997-02-17
EP0756602A1 (en) 1997-02-05
CZ297296A3 (en) 1997-09-17
AU2239095A (en) 1995-11-10
ATE181737T1 (de) 1999-07-15
EP0756602B1 (en) 1999-06-30
ES2135722T3 (es) 1999-11-01
AU697349B2 (en) 1998-10-01
HU9602835D0 (en) 1996-12-30
NZ283929A (en) 1998-02-26
JPH09511223A (ja) 1997-11-11
CZ286764B6 (en) 2000-06-14
CA2186900A1 (en) 1995-10-26
PL180026B1 (pl) 2000-12-29
FI964045A7 (fi) 1996-10-09
IL113365A (en) 1999-11-30
IL113365A0 (en) 1995-07-31
GR3031335T3 (en) 1999-12-31
RU2152939C1 (ru) 2000-07-20
SK130096A3 (en) 1997-08-06

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FC2A Withdrawal, rejection or dismissal of laid open patent application