ATE181737T1 - Cck oder gastrin modulierende 5-heterocyclicyl- 1,5-benzodiazepine - Google Patents
Cck oder gastrin modulierende 5-heterocyclicyl- 1,5-benzodiazepineInfo
- Publication number
- ATE181737T1 ATE181737T1 AT95915540T AT95915540T ATE181737T1 AT E181737 T1 ATE181737 T1 AT E181737T1 AT 95915540 T AT95915540 T AT 95915540T AT 95915540 T AT95915540 T AT 95915540T AT E181737 T1 ATE181737 T1 AT E181737T1
- Authority
- AT
- Austria
- Prior art keywords
- gastrin
- cck
- heterocyclicyl
- benzodiazepines
- modulating
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Diabetes (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Emergency Medicine (AREA)
- Molecular Biology (AREA)
- Endocrinology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9407433A GB9407433D0 (en) | 1994-04-14 | 1994-04-14 | Heterocyclic derivatives |
| GB9420783A GB9420783D0 (en) | 1994-10-14 | 1994-10-14 | Heterocyclic derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE181737T1 true ATE181737T1 (de) | 1999-07-15 |
Family
ID=26304703
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT95915540T ATE181737T1 (de) | 1994-04-14 | 1995-04-12 | Cck oder gastrin modulierende 5-heterocyclicyl- 1,5-benzodiazepine |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP0756602B1 (de) |
| JP (1) | JPH09511223A (de) |
| KR (1) | KR970702274A (de) |
| CN (1) | CN1176646A (de) |
| AT (1) | ATE181737T1 (de) |
| AU (1) | AU697349B2 (de) |
| BR (1) | BR9507381A (de) |
| CA (1) | CA2186900A1 (de) |
| CZ (1) | CZ286764B6 (de) |
| DE (1) | DE69510545T2 (de) |
| DK (1) | DK0756602T3 (de) |
| ES (1) | ES2135722T3 (de) |
| FI (1) | FI964045A7 (de) |
| GR (1) | GR3031335T3 (de) |
| HU (1) | HUT76135A (de) |
| IL (1) | IL113365A (de) |
| IS (1) | IS4367A (de) |
| MX (1) | MX9604765A (de) |
| NO (1) | NO964348L (de) |
| NZ (1) | NZ283929A (de) |
| PL (1) | PL180026B1 (de) |
| RU (1) | RU2152939C1 (de) |
| SK (1) | SK281433B6 (de) |
| TW (1) | TW369529B (de) |
| WO (1) | WO1995028419A1 (de) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9307833D0 (en) * | 1993-04-15 | 1993-06-02 | Glaxo Inc | Modulators of cholecystokinin and gastrin |
| PE27497A1 (es) * | 1994-04-15 | 1997-08-07 | Glaxo Inc | Derivados de 1,5 benzodiazepina |
| JP3999819B2 (ja) * | 1996-12-10 | 2007-10-31 | ゼリア新薬工業株式会社 | １，５―ベンゾジアセピン誘導体 |
| US7910548B2 (en) * | 1997-06-06 | 2011-03-22 | Amylin Pharmaceuticals, Inc. | Methods for treating obesity |
| EP1123928A4 (de) * | 1998-10-20 | 2005-02-16 | Takeda Pharmaceutical | 1,5-benzodiazepin-verbindungen, verfahren zu ihrer herstellung und eine medizin |
| JP4535350B2 (ja) * | 1998-11-17 | 2010-09-01 | クミアイ化学工業株式会社 | ピリミジニルベンズイミダゾール誘導体及び農園芸用殺菌剤 |
| ATE402700T1 (de) * | 2002-08-27 | 2008-08-15 | Merck Patent Gmbh | Glycinamid-derivate als raf-kinase-hemmer |
| GEP20094723B (en) | 2004-05-25 | 2009-07-10 | Pfizer Prod Inc | Tetraazabenzo [e] azulene derivatives and analogs thereof |
| RU2303597C1 (ru) * | 2006-05-12 | 2007-07-27 | Иващенко Андрей Александрович | Фармацевтическая композиция, способы ее получения и применения |
| WO2013105608A1 (ja) | 2012-01-13 | 2013-07-18 | 日本ケミファ株式会社 | Ｐ２ｘ４受容体拮抗剤 |
| US9815850B2 (en) | 2016-02-05 | 2017-11-14 | Denali Therapeutics Inc. | Compounds, compositions and methods |
| LT3552017T (lt) | 2016-12-09 | 2022-05-10 | Denali Therapeutics Inc. | Junginiai, naudotini kaip ripk1 inhibitoriai |
| JP2022552655A (ja) | 2019-10-07 | 2022-12-19 | キャリーオペ，インク． | Ｇｐｒ１１９アゴニスト |
| MX2022010548A (es) | 2020-02-28 | 2022-09-23 | Kallyope Inc | Agonistas de gpr40. |
| EP4463229A1 (de) | 2022-01-12 | 2024-11-20 | Denali Therapeutics Inc. | Kristalline formen von (s)-5-benzyl-n-(5-methyl-4-oxo-2,3,4,5-tetrahydropyrido[3,2-b! [l,4)oxazepin-3-yl)-4h-1,2,4-triazol-3-carboxamid |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2641280B1 (fr) * | 1988-12-29 | 1994-01-21 | Roussel Uclaf | Nouveaux derives de la 2,4-dioxo 2,3,4,5-tetrahydro 1h-1,5-benzodiazepine, leur procede de preparation et leur application comme medicaments |
| GB9201180D0 (en) * | 1992-01-21 | 1992-03-11 | Glaxo Group Ltd | Chemical compounds |
| GB9307833D0 (en) * | 1993-04-15 | 1993-06-02 | Glaxo Inc | Modulators of cholecystokinin and gastrin |
-
1995
- 1995-04-12 SK SK1300-96A patent/SK281433B6/sk unknown
- 1995-04-12 NZ NZ283929A patent/NZ283929A/en unknown
- 1995-04-12 CN CN95193582A patent/CN1176646A/zh active Pending
- 1995-04-12 DK DK95915540T patent/DK0756602T3/da active
- 1995-04-12 JP JP7516406A patent/JPH09511223A/ja active Pending
- 1995-04-12 ES ES95915540T patent/ES2135722T3/es not_active Expired - Lifetime
- 1995-04-12 MX MX9604765A patent/MX9604765A/es unknown
- 1995-04-12 KR KR1019960705732A patent/KR970702274A/ko not_active Ceased
- 1995-04-12 RU RU96121555/04A patent/RU2152939C1/ru active
- 1995-04-12 BR BR9507381A patent/BR9507381A/pt unknown
- 1995-04-12 CZ CZ19962972A patent/CZ286764B6/cs not_active IP Right Cessation
- 1995-04-12 AT AT95915540T patent/ATE181737T1/de not_active IP Right Cessation
- 1995-04-12 TW TW084103539A patent/TW369529B/zh active
- 1995-04-12 FI FI964045A patent/FI964045A7/fi unknown
- 1995-04-12 DE DE69510545T patent/DE69510545T2/de not_active Expired - Fee Related
- 1995-04-12 EP EP95915540A patent/EP0756602B1/de not_active Expired - Lifetime
- 1995-04-12 WO PCT/US1995/004163 patent/WO1995028419A1/en not_active Ceased
- 1995-04-12 PL PL95316870A patent/PL180026B1/pl unknown
- 1995-04-12 AU AU22390/95A patent/AU697349B2/en not_active Ceased
- 1995-04-12 CA CA002186900A patent/CA2186900A1/en not_active Abandoned
- 1995-04-12 HU HU9602835A patent/HUT76135A/hu unknown
- 1995-04-13 IL IL11336595A patent/IL113365A/xx not_active IP Right Cessation
-
1996
- 1996-09-30 IS IS4367A patent/IS4367A/is unknown
- 1996-10-11 NO NO964348A patent/NO964348L/no not_active Application Discontinuation
-
1999
- 1999-09-28 GR GR990402437T patent/GR3031335T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1176646A (zh) | 1998-03-18 |
| EP0756602A1 (de) | 1997-02-05 |
| KR970702274A (ko) | 1997-05-13 |
| NO964348D0 (no) | 1996-10-11 |
| HUT76135A (en) | 1997-06-30 |
| PL316870A1 (en) | 1997-02-17 |
| CA2186900A1 (en) | 1995-10-26 |
| HU9602835D0 (en) | 1996-12-30 |
| SK130096A3 (en) | 1997-08-06 |
| SK281433B6 (sk) | 2001-03-12 |
| GR3031335T3 (en) | 1999-12-31 |
| DK0756602T3 (da) | 2000-01-31 |
| MX9604765A (es) | 1998-05-31 |
| RU2152939C1 (ru) | 2000-07-20 |
| AU697349B2 (en) | 1998-10-01 |
| NO964348L (no) | 1996-12-02 |
| IL113365A0 (en) | 1995-07-31 |
| FI964045L (fi) | 1996-10-09 |
| FI964045A0 (fi) | 1996-10-09 |
| NZ283929A (en) | 1998-02-26 |
| TW369529B (en) | 1999-09-11 |
| BR9507381A (pt) | 1997-09-23 |
| DE69510545D1 (de) | 1999-08-05 |
| CZ286764B6 (en) | 2000-06-14 |
| FI964045A7 (fi) | 1996-10-09 |
| CZ297296A3 (en) | 1997-09-17 |
| IL113365A (en) | 1999-11-30 |
| AU2239095A (en) | 1995-11-10 |
| WO1995028419A1 (en) | 1995-10-26 |
| PL180026B1 (pl) | 2000-12-29 |
| DE69510545T2 (de) | 2000-01-13 |
| ES2135722T3 (es) | 1999-11-01 |
| IS4367A (is) | 1996-09-30 |
| EP0756602B1 (de) | 1999-06-30 |
| JPH09511223A (ja) | 1997-11-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |