NO811731L - Fremgangsmaate for fremstilling av imidazo-rifamycin-derivater - Google Patents

Fremgangsmaate for fremstilling av imidazo-rifamycin-derivater

Info

Publication number
NO811731L
NO811731L NO811731A NO811731A NO811731L NO 811731 L NO811731 L NO 811731L NO 811731 A NO811731 A NO 811731A NO 811731 A NO811731 A NO 811731A NO 811731 L NO811731 L NO 811731L
Authority
NO
Norway
Prior art keywords
imidazo
procedure
preparation
rifamycin derivatives
rifamycin
Prior art date
Application number
NO811731A
Other languages
English (en)
Other versions
NO155622C (no
NO155622B (no
Inventor
Egido Marchi
Lauretta Montecchi
Original Assignee
Alfa Farmaceutici Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfa Farmaceutici Spa filed Critical Alfa Farmaceutici Spa
Publication of NO811731L publication Critical patent/NO811731L/no
Publication of NO155622B publication Critical patent/NO155622B/no
Publication of NO155622C publication Critical patent/NO155622C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
NO811731A 1980-05-22 1981-05-21 Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrido- og isokinolin (1[,2[:1,2) imidazo (5,4-c) rifamycin sv og s derivater. NO155622C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT03429/80A IT1154655B (it) 1980-05-22 1980-05-22 Derivati imidazo-rifamicinici metodi per la loro preparazione e loro uso come sostanza ad azione antibatterica

Publications (3)

Publication Number Publication Date
NO811731L true NO811731L (no) 1981-11-23
NO155622B NO155622B (no) 1987-01-19
NO155622C NO155622C (no) 1987-04-29

Family

ID=11107198

Family Applications (1)

Application Number Title Priority Date Filing Date
NO811731A NO155622C (no) 1980-05-22 1981-05-21 Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrido- og isokinolin (1[,2[:1,2) imidazo (5,4-c) rifamycin sv og s derivater.

Country Status (25)

Country Link
US (1) US4341785A (no)
JP (1) JPS5711987A (no)
AR (1) AR226212A1 (no)
AT (1) AT373599B (no)
AU (1) AU537093B2 (no)
BE (1) BE888895A (no)
CA (1) CA1142518A (no)
CH (1) CH648037A5 (no)
DE (1) DE3120460A1 (no)
DK (1) DK157876C (no)
EG (1) EG14891A (no)
ES (1) ES502906A0 (no)
FI (1) FI69467C (no)
FR (1) FR2482967A1 (no)
GB (1) GB2079270B (no)
GR (1) GR75640B (no)
IE (1) IE51204B1 (no)
IT (1) IT1154655B (no)
LU (1) LU83376A1 (no)
NL (1) NL187022C (no)
NO (1) NO155622C (no)
PH (2) PH17207A (no)
PT (1) PT73064B (no)
SE (1) SE453089B (no)
ZA (1) ZA813430B (no)

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US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics
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US7256187B2 (en) * 2004-03-10 2007-08-14 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime derivatives effective against drug-resistant microbes
US7265107B2 (en) * 2004-03-10 2007-09-04 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime cyclo derivatives effective against drug-resistant microbes
US7202246B2 (en) * 2004-06-09 2007-04-10 Cumbre Pharmaceuticals Inc. Spiro-rifamycin derivatives targeting RNA polymerase
US20060210492A1 (en) * 2005-03-02 2006-09-21 Kodsi Robert E Use of rifaximin for treatment and prevention of periodontal conditions
US8003118B2 (en) * 2005-03-02 2011-08-23 Kodsi Robert E Use of rifaximin for the prevention of aspiration pneumonia and/or sepsis
US20060210483A1 (en) * 2005-03-02 2006-09-21 Kodsi Robert E Non-systemic antibiotic formulations and related method of use and treatment of upper respiratory infections
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ITBO20050123A1 (it) 2005-03-07 2005-06-06 Alfa Wassermann Spa Formulazioni farmaceutiche gastroresistenti contenenti rifaximina
EP1928890B1 (en) 2005-08-11 2013-04-03 Targanta Therapeutics Inc. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
ES2747259T3 (es) 2006-03-09 2020-03-10 Salix Pharmaceuticals Inc Preparación anti-disfunción rectal de rifaximina
ES2538478T3 (es) 2006-08-02 2015-06-22 Salix Pharmaceuticals, Inc. Métodos para el tratamiento de enteritis por radiación
ITMI20061692A1 (it) 2006-09-05 2008-03-06 Alfa Wassermann Spa Uso di polioli per ottenere forme polimorfe stabili di rifaximina
KR101667534B1 (ko) * 2006-09-22 2016-10-19 씨아이피엘에이 엘티디. 리팍시민
US20080159987A1 (en) * 2007-01-03 2008-07-03 Leonard Weinstock Use of Rifaximin for the Treatment of Restless Legs Syndrome
US20080161337A1 (en) * 2007-01-03 2008-07-03 Leonard Weinstock Use of Rifaximin for the Treatment of Chronic Prostatitis
ITMI20071241A1 (it) * 2007-06-20 2008-12-21 Solmag S P A Processo per la preparazione di rifaximina amorfa e rifaximina amorfa cosi' ottenuta
WO2009008005A1 (en) 2007-07-06 2009-01-15 Lupin Limited Pharmaceutical compositions of rifaximin
ES2798253T3 (es) 2007-07-06 2020-12-10 Lupin Ltd Composiciones farmacéuticas de rifaximina
US7709634B2 (en) * 2007-09-20 2010-05-04 Apotex Pharmachem Inc. Amorphous form of rifaximin and processes for its preparation
US8486956B2 (en) 2008-02-25 2013-07-16 Salix Pharmaceuticals, Ltd Forms of rifaximin and uses thereof
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US11779571B2 (en) 2008-02-26 2023-10-10 Salix Pharmaceuticals, Inc. Methods for treating irritable bowel syndrome (IBS)
PL2294012T3 (pl) 2008-05-07 2014-12-31 Salix Pharmaceuticals Inc Podawanie środka czyszczącego jelito i antybiotyku w leczeniu choroby jelit
WO2010019511A2 (en) 2008-08-13 2010-02-18 Targanta Therapeutics Corp. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
AU2009297562B2 (en) 2008-09-26 2015-04-23 Alfasigma S.P.A. Agent for preventing and/or treating functional gastrointestinal disorder
JP6037615B2 (ja) 2008-10-02 2016-12-07 サリックス ファーマシューティカルズ リミテッド 肝性脳症を治療する方法
EP2355805B1 (en) 2008-12-10 2019-02-13 Cipla Limited Rifaximin complexes
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BR112012005627A2 (pt) 2009-09-13 2017-02-21 Salix Pharmaceuticals Ltd "uso de rifaximina para preparação de um medicamento para tratar síndrome do intestino irritável (ibs)"
UA110199C2 (en) 2009-10-27 2015-12-10 Lupin Ltd Solid rifaximin dispersion
NZ600362A (en) 2009-11-23 2014-08-29 Cipla Ltd Topical foam composition
EP2401282B2 (en) 2009-12-28 2017-01-04 Silvio Massimo Lavagna Method for the production of amorphous rifaximin
EP2536282A4 (en) 2010-02-18 2013-07-03 Salix Pharmaceuticals Ltd METHOD FOR THE TREATMENT OF INFECTIONS
IT1398550B1 (it) 2010-03-05 2013-03-01 Alfa Wassermann Spa Formulazioni comprendenti rifaximina utili per ottenere un effetto prolungato nel tempo
EP2544660B1 (en) 2010-03-10 2018-06-13 Lupin Limited Rifaximin ready-to-use suspension
PT2593463T (pt) 2010-07-12 2020-09-17 Salix Pharmaceuticals Ltd Formulações de rifaximina e usos das mesmas
US8759513B2 (en) 2010-09-13 2014-06-24 Sequent Scientific Limited Polymorphic form of rifaximin and process for its preparation
CN103827122B (zh) 2011-02-11 2016-08-31 萨利克斯药品有限公司 利福昔明的形式及其用途
AU2012251385A1 (en) 2011-05-02 2013-11-21 Ranbaxy Laboratories Limited Rifaximin dimethylformamide solvate
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ITBO20110461A1 (it) 2011-07-29 2013-01-30 Alfa Wassermann Spa Composizioni farmaceutiche comprendenti rifaximina, processi per la loro preparazione e loro uso nel trattamento di infezioni vaginali.
RU2496475C2 (ru) 2011-10-26 2013-10-27 Александр Васильевич Иващенко Фармацевтическая композиция и набор для лечения бактериальных инфекций
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WO2014091432A1 (en) 2012-12-12 2014-06-19 Ranbaxy Laboratories Limited Pharmaceutical compositions of rifaximin
AU2014229467A1 (en) 2013-03-15 2015-08-06 Alfa Wassermann S.P.A. Rifaximin for use in the treating of vaginal infections.
JP2016516988A (ja) 2013-03-15 2016-06-09 アルファ ワッセルマン ソシエタ ペル アチオニAlfa Wassermann S.P.A. 膣感染症を診断するための方法
ES2829285T3 (es) 2013-04-12 2021-05-31 Alfasigma Spa Administración de AINE y composiciones, métodos y sistemas relacionados
US9018225B1 (en) 2013-07-26 2015-04-28 Novel Laboratories Rifaximin crystalline forms and methods of preparation thereof
ES2621557T3 (es) 2014-03-31 2017-07-04 Euticals S.P.A. Mezcla polimórfica de rifaximina y su uso para la preparación de formulaciones sólidas
JP6693946B2 (ja) 2014-05-04 2020-05-13 サリックス ファーマスーティカルズ,インコーポレーテッド Ibs微生物叢及びその使用
AU2015260837B2 (en) 2014-05-12 2019-02-28 Alfasigma S.P.A. New solvated crystal form of rifaximin, production, compositions and uses thereof
EP2982764A1 (en) 2014-08-05 2016-02-10 ALFA WASSERMANN S.p.A. Identification of vaginal bacteria
US9988398B2 (en) 2016-06-07 2018-06-05 Cadila Healthcare Limited Crystalline form of rifaximin and process for its preparation
PT3518924T (pt) 2016-09-30 2022-10-27 Salix Pharmaceuticals Inc Formas de dispersão sólidas de rifaximina
IT201700091912A1 (it) * 2017-08-08 2019-02-08 Biofer Spa Nuove pirido-imidazo rifamicine
PL3645539T3 (pl) 2017-06-26 2021-10-25 Biofer S.P.A. Pochodne pirydoimidazoryfamycyny jako środek przeciwbakteryjny

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE273377C (no) *
AT273377B (de) * 1967-03-01 1969-08-11 Lepetit Spa Verfahren zur Herstellung von neuen Rifamycinen
AT344898B (de) * 1975-06-13 1978-08-10 Archifar Ind Chim Trentino Verfahren zur herstellung neuer rifamycin-verbindungen
DK345977A (da) * 1976-09-30 1978-03-31 Archifar Ind Chim Trentino G rifamycinforbindelser og fremgangsmaade til deres fremstillin
CH629212A5 (it) * 1976-10-18 1982-04-15 Erba Farmitalia Procedimento per la preparazione di composti di rifamicina.
CH633014A5 (en) * 1978-06-09 1982-11-15 Erba Farmitalia Rifamycin compounds

Also Published As

Publication number Publication date
IT1154655B (it) 1987-01-21
PH17207A (en) 1984-06-19
SE8103216L (sv) 1981-11-23
FI69467C (fi) 1986-02-10
DK157876B (da) 1990-02-26
NO155622C (no) 1987-04-29
NL187022C (nl) 1991-05-01
BE888895A (fr) 1981-09-16
AU7065581A (en) 1981-11-26
ATA222781A (de) 1983-06-15
DK224781A (da) 1981-11-23
AT373599B (de) 1984-02-10
ES8203388A1 (es) 1982-04-01
DE3120460A1 (de) 1982-03-11
FR2482967A1 (fr) 1981-11-27
IT8003429A0 (it) 1980-05-22
AR226212A1 (es) 1982-06-15
FI69467B (fi) 1985-10-31
US4341785A (en) 1982-07-27
EG14891A (en) 1985-12-31
GR75640B (no) 1984-08-02
FR2482967B1 (no) 1985-03-29
GB2079270A (en) 1982-01-20
GB2079270B (en) 1984-01-18
PT73064B (en) 1982-07-05
FI811565L (fi) 1981-11-23
IE811139L (en) 1981-11-22
NL187022B (nl) 1990-12-03
NL8102290A (nl) 1981-12-16
JPS5711987A (en) 1982-01-21
LU83376A1 (fr) 1981-09-11
IE51204B1 (en) 1986-10-29
NO155622B (no) 1987-01-19
PT73064A (en) 1981-06-01
AU537093B2 (en) 1984-06-07
DK157876C (da) 1990-07-30
SE453089B (sv) 1988-01-11
ZA813430B (en) 1982-06-30
PH18704A (en) 1985-09-05
CH648037A5 (de) 1985-02-28
ES502906A0 (es) 1982-04-01
JPS6123192B2 (no) 1986-06-04
CA1142518A (en) 1983-03-08
DE3120460C2 (no) 1990-12-13

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