NO332370B1 - Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom - Google Patents
Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom Download PDFInfo
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- NO332370B1 NO332370B1 NO20050748A NO20050748A NO332370B1 NO 332370 B1 NO332370 B1 NO 332370B1 NO 20050748 A NO20050748 A NO 20050748A NO 20050748 A NO20050748 A NO 20050748A NO 332370 B1 NO332370 B1 NO 332370B1
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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PCT/US2003/027513 WO2004021984A2 (en) | 2002-09-04 | 2003-09-02 | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
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NO20050748L NO20050748L (no) | 2005-03-30 |
NO332370B1 true NO332370B1 (no) | 2012-09-03 |
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EP (2) | EP1551511B1 (sr) |
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KR (3) | KR101238041B1 (sr) |
CN (2) | CN101863886A (sr) |
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AU (1) | AU2003270065B2 (sr) |
BR (1) | BR0314024A (sr) |
CA (1) | CA2496842C (sr) |
CY (2) | CY1120250T1 (sr) |
DK (2) | DK1551511T5 (sr) |
ES (2) | ES2706578T3 (sr) |
GE (1) | GEP20074019B (sr) |
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HU (2) | HUE041936T2 (sr) |
IL (5) | IL166802A (sr) |
IS (1) | IS7719A (sr) |
LT (2) | LT1551511T (sr) |
MX (1) | MXPA05002301A (sr) |
MY (1) | MY139563A (sr) |
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NZ (1) | NZ538166A (sr) |
PE (1) | PE20040997A1 (sr) |
PL (1) | PL219563B1 (sr) |
PT (2) | PT2570414T (sr) |
RS (2) | RS55124B1 (sr) |
RU (1) | RU2382042C2 (sr) |
SI (2) | SI2570414T1 (sr) |
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MY139563A (en) * | 2002-09-04 | 2009-10-30 | Bristol Myers Squibb Co | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
AR043443A1 (es) * | 2003-03-07 | 2005-07-27 | Merck & Co Inc | Procedimiento de preparacion de tetrahidrotriazolopirazinas y productos intermedios |
US7318925B2 (en) * | 2003-08-08 | 2008-01-15 | Amgen Fremont, Inc. | Methods of use for antibodies against parathyroid hormone |
US7745630B2 (en) | 2003-12-22 | 2010-06-29 | Justin Stephen Bryans | Triazolyl piperidine arginine vasopressin receptor modulators |
AU2005272627A1 (en) | 2004-08-13 | 2006-02-23 | Amgen Inc. | Substituted benzofused heterocycles |
AU2005277389A1 (en) * | 2004-08-18 | 2006-03-02 | Elixir Pharmaceuticals, Inc. | Growth-hormone secretagogues |
GB0420722D0 (en) | 2004-09-17 | 2004-10-20 | Addex Pharmaceuticals Sa | Novel allosteric modulators |
WO2006036932A2 (en) * | 2004-09-27 | 2006-04-06 | Elixir Pharmaceuticals, Inc. | Sulfonamides and uses thereof |
US8143425B2 (en) * | 2004-10-12 | 2012-03-27 | Bristol-Myers Squibb Company | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
US7579360B2 (en) * | 2005-06-09 | 2009-08-25 | Bristol-Myers Squibb Company | Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors |
US20060293370A1 (en) * | 2005-06-10 | 2006-12-28 | Saunders Jeffrey O | Sulfonamide compounds and uses thereof |
US7829589B2 (en) | 2005-06-10 | 2010-11-09 | Elixir Pharmaceuticals, Inc. | Sulfonamide compounds and uses thereof |
EP1757290A1 (en) | 2005-08-16 | 2007-02-28 | Zentaris GmbH | Novel triazole derivatives as ghrelin analogue ligands of growth hormone secretagogue receptors |
NZ568807A (en) | 2005-12-21 | 2011-05-27 | Janssen Pharmaceutica Nv | Triazolopyridazines as tyrosine kinase modulators |
JP5291471B2 (ja) * | 2006-02-15 | 2013-09-18 | アボット・ラボラトリーズ | 新規なアセチル−CoAカルボキシラーゼ(ACC)阻害薬およびこれらの糖尿病、肥満および代謝症候群における使用 |
AR059898A1 (es) | 2006-03-15 | 2008-05-07 | Janssen Pharmaceutica Nv | Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2 |
CA2644963A1 (en) * | 2006-03-31 | 2007-10-11 | Novartis Ag | Organic compounds |
EP2046788A1 (en) * | 2006-07-12 | 2009-04-15 | Syngeta Participations AG | Triazolopyridine derivatives as herbicides |
EA201300152A1 (ru) | 2006-11-27 | 2013-07-30 | Х. Лундбекк А/С | Гетероариламидные производные |
EP2119719A1 (en) * | 2006-12-26 | 2009-11-18 | Daiichi Sankyo Company, Limited | Thiazepine derivative |
EP2644618B1 (en) | 2007-02-09 | 2016-08-17 | Ocera Therapeutics, Inc. | tether intermediates for the synthesis of macrocyclic ghrelin receptor modulators |
TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
BRPI0809567A2 (pt) | 2007-04-10 | 2014-09-23 | Lundbeck & Co As H | Composto, composição farmacêutica, método para modular a atividade de um receptor de p2x7, para tratar uma condição responsiva à modulação do receptor de p2x7 em um paciente, para inibir a morte de células do gânglio retinal em um paciente, e para determinar a presença ou ausência do receptor de p2x7 em uma amostra, preparação farmacêutica acondiciaonada, e, uso de um composto |
EP2142551B1 (en) | 2007-04-17 | 2015-10-14 | Bristol-Myers Squibb Company | Fused heterocyclic 11-beta-hydroxysteroid dehydrogenase type i inhibitors |
EP2152079A4 (en) * | 2007-06-04 | 2011-03-09 | Avila Therapeutics Inc | HETEROCYCLIC COMPOUNDS AND USES THEREOF |
AU2008297876B2 (en) | 2007-09-14 | 2011-07-07 | Addex Pharma S.A. | 1,3-disubstituted 4-(aryl-x-phenyl)-1h-pyridin-2-ones |
ES2409215T3 (es) | 2007-09-14 | 2013-06-25 | Janssen Pharmaceuticals, Inc. | 4-fenil-1H-piridin-2-onas 1-3-disustituidas |
CN103342695B (zh) | 2007-09-14 | 2015-04-22 | 杨森制药有限公司 | 1’,3’-二取代的-4-苯基-3,4,5,6-四氢-2h,1’h-[1,4’]二吡啶-2’-酮 |
JP5433582B2 (ja) | 2007-11-14 | 2014-03-05 | ジャンセン ファーマシューティカルズ, インコーポレイテッド. | イミダゾ[1,2−a]ピリジン誘導体およびmGluR2受容体の正のアロステリック調節因子としてのその使用 |
BRPI0918055A2 (pt) | 2008-09-02 | 2015-12-01 | Addex Pharmaceuticals Sa | derivados de 3-azabiciclo[3,1,0]hexila como moduladores de receptores metabotrópicos de glutamato. |
CN102186477B (zh) | 2008-10-16 | 2013-07-17 | 奥梅-杨森制药有限公司 | 作为代谢型谷氨酸受体调节剂的吲哚和苯并吗啉衍生物 |
EP2351743A4 (en) * | 2008-10-27 | 2012-05-09 | Takeda Pharmaceutical | BICYCLIC CONNECTION |
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