NO332370B1 - Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom - Google Patents
Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom Download PDFInfo
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- NO332370B1 NO332370B1 NO20050748A NO20050748A NO332370B1 NO 332370 B1 NO332370 B1 NO 332370B1 NO 20050748 A NO20050748 A NO 20050748A NO 20050748 A NO20050748 A NO 20050748A NO 332370 B1 NO332370 B1 NO 332370B1
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Classifications
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- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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PCT/US2003/027513 WO2004021984A2 (en) | 2002-09-04 | 2003-09-02 | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
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NO20050748L NO20050748L (no) | 2005-03-30 |
NO332370B1 true NO332370B1 (no) | 2012-09-03 |
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NO20050748A NO332370B1 (no) | 2002-09-04 | 2005-02-11 | Heterocykliske aromatiske forbindelser, farmasoytisk preparat inneholdende slike samt anvendelse av slike for fremstilling av farmasoytisk preparat forbehandling av sykdom |
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EP (2) | EP1551511B1 (pt) |
JP (1) | JP4658600B2 (pt) |
KR (3) | KR101238041B1 (pt) |
CN (2) | CN101863886A (pt) |
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AU (1) | AU2003270065B2 (pt) |
BR (1) | BR0314024A (pt) |
CA (1) | CA2496842C (pt) |
CY (2) | CY1120250T1 (pt) |
DK (2) | DK1551511T5 (pt) |
ES (2) | ES2706578T3 (pt) |
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HR (1) | HRP20050188B1 (pt) |
HU (2) | HUE041936T2 (pt) |
IL (5) | IL166802A (pt) |
IS (1) | IS7719A (pt) |
LT (2) | LT1551511T (pt) |
MX (1) | MXPA05002301A (pt) |
MY (1) | MY139563A (pt) |
NO (1) | NO332370B1 (pt) |
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PE (1) | PE20040997A1 (pt) |
PL (1) | PL219563B1 (pt) |
PT (2) | PT1551511T (pt) |
RS (2) | RS55124B1 (pt) |
RU (1) | RU2382042C2 (pt) |
SI (2) | SI2570414T1 (pt) |
TW (2) | TWI330185B (pt) |
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MY139563A (en) * | 2002-09-04 | 2009-10-30 | Bristol Myers Squibb Co | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
AR043443A1 (es) * | 2003-03-07 | 2005-07-27 | Merck & Co Inc | Procedimiento de preparacion de tetrahidrotriazolopirazinas y productos intermedios |
US7318925B2 (en) * | 2003-08-08 | 2008-01-15 | Amgen Fremont, Inc. | Methods of use for antibodies against parathyroid hormone |
US7745630B2 (en) | 2003-12-22 | 2010-06-29 | Justin Stephen Bryans | Triazolyl piperidine arginine vasopressin receptor modulators |
US7572783B2 (en) | 2004-08-13 | 2009-08-11 | Amgen Inc. | Substituted benzofused heterocycles |
US20080261873A1 (en) * | 2004-08-18 | 2008-10-23 | Elixir Pharmaceuticals, Inc. | Growth-Hormone Secretagogues |
GB0420722D0 (en) | 2004-09-17 | 2004-10-20 | Addex Pharmaceuticals Sa | Novel allosteric modulators |
MX2007003398A (es) * | 2004-09-27 | 2007-05-21 | Elixir Pharmaceuticals Inc | Sulfonamidas y sus usos. |
US8143425B2 (en) * | 2004-10-12 | 2012-03-27 | Bristol-Myers Squibb Company | Heterocyclic aromatic compounds useful as growth hormone secretagogues |
US7579360B2 (en) * | 2005-06-09 | 2009-08-25 | Bristol-Myers Squibb Company | Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors |
MX2007015617A (es) * | 2005-06-10 | 2008-03-06 | Elixir Pharmaceuticals Inc | Compuestos de sulfonamida y usos de los mismos. |
US7829589B2 (en) | 2005-06-10 | 2010-11-09 | Elixir Pharmaceuticals, Inc. | Sulfonamide compounds and uses thereof |
EP1757290A1 (en) | 2005-08-16 | 2007-02-28 | Zentaris GmbH | Novel triazole derivatives as ghrelin analogue ligands of growth hormone secretagogue receptors |
US8030305B2 (en) * | 2005-12-21 | 2011-10-04 | Janssen Pharmaceutica N.V. | Triazolopyridazines as kinase modulators |
CN101421255A (zh) * | 2006-02-15 | 2009-04-29 | 艾博特公司 | 新的乙酰辅助a羧化酶(acc)抑制剂及其在糖尿病、肥胖症和代谢综合症中的应用 |
AR059898A1 (es) | 2006-03-15 | 2008-05-07 | Janssen Pharmaceutica Nv | Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2 |
JP2009531390A (ja) * | 2006-03-31 | 2009-09-03 | ノバルティス アクチエンゲゼルシャフト | 有機化合物 |
EP2046788A1 (en) * | 2006-07-12 | 2009-04-15 | Syngeta Participations AG | Triazolopyridine derivatives as herbicides |
EA201300152A1 (ru) | 2006-11-27 | 2013-07-30 | Х. Лундбекк А/С | Гетероариламидные производные |
JPWO2008078725A1 (ja) * | 2006-12-26 | 2010-04-30 | 第一三共株式会社 | チアゼピン誘導体 |
ES2602789T3 (es) | 2007-02-09 | 2017-02-22 | Ocera Therapeutics, Inc. | Productos intermedios conectores para la síntesis de moduladores macrocíclicos del receptor de la grelina |
TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
JP2010523668A (ja) | 2007-04-10 | 2010-07-15 | ハー・ルンドベック・アクチエゼルスカベット | P2x7拮抗薬としてのヘテロアリールアミド類似体 |
WO2008130951A1 (en) * | 2007-04-17 | 2008-10-30 | Bristol-Myers Squibb Company | Fused heterocyclic 11-beta-hydroxysteroid dehydrogenase type i inhibitors |
EP2152079A4 (en) * | 2007-06-04 | 2011-03-09 | Avila Therapeutics Inc | HETEROCYCLIC COMPOUNDS AND USES THEREOF |
ATE516272T1 (de) | 2007-09-14 | 2011-07-15 | Ortho Mcneil Janssen Pharm | 1,3-disubstituierte 4-(aryl-x-phenyl)-1h-pyridin- 2-one |
JP5133416B2 (ja) | 2007-09-14 | 2013-01-30 | オルソー−マクニール−ジャンセン ファーマシューティカルズ, インコーポレイテッド. | 1’,3’−二置換−4−フェニル−3,4,5,6−テトラヒドロ−2h,1’h−[1,4’]ビピリジニル−2’−オン |
EP2205565B1 (en) | 2007-09-14 | 2013-04-17 | Janssen Pharmaceuticals, Inc. | 1,3-disubstituted-4-phenyl-1 h-pyridin-2-ones |
EP2220083B1 (en) | 2007-11-14 | 2017-07-19 | Janssen Pharmaceuticals, Inc. | Imidazo[1,2-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
US8691849B2 (en) | 2008-09-02 | 2014-04-08 | Janssen Pharmaceuticals, Inc. | 3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors |
CA2738849C (en) | 2008-10-16 | 2016-06-28 | Addex Pharma S.A. | Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors |
EP2351743A4 (en) * | 2008-10-27 | 2012-05-09 | Takeda Pharmaceutical | BICYCLIC CONNECTION |
CN102232074B (zh) | 2008-11-28 | 2014-12-03 | 奥梅-杨森制药有限公司 | 作为代谢性谷氨酸盐受体调节剂的吲哚和苯并噁嗪衍生物 |
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