NO331232B1 - Spontant dispergerbare N-benzoyl staurosporin-sammensetninger - Google Patents

Spontant dispergerbare N-benzoyl staurosporin-sammensetninger

Info

Publication number
NO331232B1
NO331232B1 NO20013964A NO20013964A NO331232B1 NO 331232 B1 NO331232 B1 NO 331232B1 NO 20013964 A NO20013964 A NO 20013964A NO 20013964 A NO20013964 A NO 20013964A NO 331232 B1 NO331232 B1 NO 331232B1
Authority
NO
Norway
Prior art keywords
spontaneously dispersible
benzoyl staurosporine
compositions
staurosporine compositions
benzoyl
Prior art date
Application number
NO20013964A
Other languages
English (en)
Norwegian (no)
Other versions
NO20013964L (no
NO20013964D0 (no
Inventor
Barbara Haberlin
Graham Paul Matthews
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10847896&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO331232(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20013964D0 publication Critical patent/NO20013964D0/no
Publication of NO20013964L publication Critical patent/NO20013964L/no
Publication of NO331232B1 publication Critical patent/NO331232B1/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Liposomes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dispersion Chemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Vascular Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20013964A 1999-02-16 2001-08-15 Spontant dispergerbare N-benzoyl staurosporin-sammensetninger NO331232B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9903547.9A GB9903547D0 (en) 1999-02-16 1999-02-16 Organic compounds
PCT/EP2000/001196 WO2000048571A1 (en) 1999-02-16 2000-02-14 Spontaneously dispersible n-benzoyl staurosporine compositions

Publications (3)

Publication Number Publication Date
NO20013964D0 NO20013964D0 (no) 2001-08-15
NO20013964L NO20013964L (no) 2001-10-15
NO331232B1 true NO331232B1 (no) 2011-11-07

Family

ID=10847896

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013964A NO331232B1 (no) 1999-02-16 2001-08-15 Spontant dispergerbare N-benzoyl staurosporin-sammensetninger

Country Status (34)

Country Link
US (3) US20020061873A1 (zh)
EP (1) EP1152750B1 (zh)
JP (2) JP5057610B2 (zh)
KR (2) KR100880859B1 (zh)
CN (1) CN100367930C (zh)
AR (2) AR022589A1 (zh)
AT (1) ATE430554T1 (zh)
AU (1) AU765776B2 (zh)
BR (1) BRPI0008228B8 (zh)
CA (1) CA2362277C (zh)
CL (1) CL2009001682A1 (zh)
CZ (1) CZ303979B6 (zh)
DE (1) DE60042151D1 (zh)
DK (1) DK1152750T3 (zh)
EC (1) ECSP083351A (zh)
ES (1) ES2326783T3 (zh)
GB (1) GB9903547D0 (zh)
HK (1) HK1045807B (zh)
HU (1) HUP0105364A3 (zh)
ID (1) ID30504A (zh)
IL (3) IL144512A0 (zh)
MY (1) MY128362A (zh)
NO (1) NO331232B1 (zh)
NZ (1) NZ513529A (zh)
PE (1) PE20001499A1 (zh)
PL (1) PL198330B1 (zh)
PT (1) PT1152750E (zh)
RU (1) RU2266121C2 (zh)
SI (1) SI1152750T1 (zh)
SK (1) SK286967B6 (zh)
TR (1) TR200102385T2 (zh)
TW (1) TWI240636B (zh)
WO (1) WO2000048571A1 (zh)
ZA (1) ZA200106677B (zh)

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US7795246B2 (en) 1998-08-06 2010-09-14 Cephalon, Inc. Particle-forming compositions containing fused pyrrolocarbazoles
US6200968B1 (en) * 1998-08-06 2001-03-13 Cephalon, Inc. Particle-forming compositions containing fused pyrrolocarbazoles
ES2261671T3 (es) * 2001-03-26 2006-11-16 Novartis Ag Mezcla farmaceutica que incluye una estaurosporina poco soluble en agua, un surfactante y un polimero soluble en agua.
JP4477303B2 (ja) 2001-05-16 2010-06-09 ノバルティス アーゲー Ｎ−｛５−［４−（４−メチル−ピペラジノ−メチル）−ベンゾイルアミド］−２−メチルフェニル｝−４−（３−ピリジル）−２−ピリミジン−アミンおよび化学療法剤を含んでなる併用剤
KR20090087139A (ko) * 2001-10-30 2009-08-14 노파르티스 아게 Ｆｌｔ３ 수용체 티로신 키나아제 활성의 억제제로서의 스타우로스포린 유도체
GB0206215D0 (en) 2002-03-15 2002-05-01 Novartis Ag Organic compounds
WO2004009056A1 (en) * 2002-07-23 2004-01-29 Novartis Ag Ophtalmic ointment composition comprising a drug, an ointment base and a solubiling/dispersing agent
US7842791B2 (en) * 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
TWI324604B (en) * 2003-06-18 2010-05-11 Novartis Ag New use of staurosporine derivatives
GB0512324D0 (en) 2005-06-16 2005-07-27 Novartis Ag Organic compounds
GB0419159D0 (en) * 2004-08-27 2004-09-29 Novartis Ag Organic compounds
GT200500310A (es) 2004-11-19 2006-06-19 Compuestos organicos
US20100038816A1 (en) 2006-08-16 2010-02-18 Novartis Ag Method of making solid dispersions of highly crystalline therapeutic compounds
FR2918566B1 (fr) 2007-07-11 2009-10-09 Pierre Fabre Medicament Sa Composition pharmaceutique stable d'un sel hydrosoluble de vinflunine.
US20090155352A1 (en) * 2007-11-20 2009-06-18 Cephalon, Inc. Microemulsion containing indolocarbazole compound and dosage forms containing the same
EP2229936B1 (en) * 2009-03-09 2015-05-06 PharmaSol GmbH Nanonized testosterone formulations for improved bioavailability
WO2011000811A2 (en) * 2009-06-30 2011-01-06 Novartis Ag Organic compounds
RU2560677C2 (ru) * 2009-12-22 2015-08-20 Лео Фарма А/С Кожная композиция, включающая аналог витамина d и смесь растворителя и поверхностно-активных веществ
JO3337B1 (ar) 2010-12-13 2019-03-13 Debiopharm Sa تركيبات صيدلية تشمل أليسبوريفير
US9387446B2 (en) 2011-09-22 2016-07-12 Ariel-University Research And Development Company Ltd. Emulsions and methods of making emulsions
KR20190032265A (ko) * 2015-12-09 2019-03-27 포스파제닉스 리미티드 약제학적 제형
CN108601732A (zh) 2015-12-09 2018-09-28 磷肌酸有限公司 药物制剂
MX2019006845A (es) 2016-12-21 2019-10-15 Avecho Biotechnology Ltd Proceso.
US20220395553A1 (en) 2019-11-14 2022-12-15 Cohbar, Inc. Cxcr4 antagonist peptides

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US4963367A (en) 1984-04-27 1990-10-16 Medaphore, Inc. Drug delivery compositions and methods
US4735939A (en) * 1987-02-27 1988-04-05 The Dow Chemical Company Insecticidal activity of staurosporine
US5093330A (en) * 1987-06-15 1992-03-03 Ciba-Geigy Corporation Staurosporine derivatives substituted at methylamino nitrogen
DE3824034C1 (zh) * 1988-07-15 1989-09-14 Gustav 7290 Freudenstadt De Memminger
KR0148748B1 (ko) * 1988-09-16 1998-08-17 장 크라메르, 한스 루돌프 하우스 사이클로스포린을 함유하는 약학조성물
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Also Published As

Publication number Publication date
CL2009001682A1 (es) 2010-07-23
DE60042151D1 (de) 2009-06-18
NO20013964L (no) 2001-10-15
EP1152750B1 (en) 2009-05-06
AR022589A1 (es) 2002-09-04
BRPI0008228B1 (pt) 2016-08-23
US8722664B2 (en) 2014-05-13
ECSP083351A (es) 2008-08-29
JP2002537242A (ja) 2002-11-05
ES2326783T3 (es) 2009-10-20
ID30504A (id) 2001-12-13
HUP0105364A3 (en) 2003-02-28
US8575147B2 (en) 2013-11-05
TR200102385T2 (tr) 2002-09-23
MY128362A (en) 2007-01-31
PL350556A1 (en) 2002-12-16
GB9903547D0 (en) 1999-04-07
HK1045807B (zh) 2008-12-05
CN100367930C (zh) 2008-02-13
JP5057610B2 (ja) 2012-10-24
CA2362277A1 (en) 2000-08-24
SK286967B6 (sk) 2009-08-06
PT1152750E (pt) 2009-08-07
ZA200106677B (en) 2003-01-14
SI1152750T1 (sl) 2009-10-31
PE20001499A1 (es) 2001-01-12
RU2266121C2 (ru) 2005-12-20
KR20080064914A (ko) 2008-07-09
NO20013964D0 (no) 2001-08-15
EP1152750A1 (en) 2001-11-14
IL144512A (en) 2011-03-31
HUP0105364A2 (hu) 2002-05-29
CZ20012931A3 (cs) 2001-11-14
KR20010093281A (ko) 2001-10-27
ATE430554T1 (de) 2009-05-15
BR0008228A (pt) 2001-10-30
NZ513529A (en) 2003-10-31
TWI240636B (en) 2005-10-01
AU3154200A (en) 2000-09-04
SK11722001A3 (sk) 2001-12-03
DK1152750T3 (da) 2009-08-24
CN1339963A (zh) 2002-03-13
AU765776B2 (en) 2003-10-02
IL192666A0 (en) 2009-02-11
BRPI0008228B8 (pt) 2021-05-25
US20080070897A1 (en) 2008-03-20
AR082579A2 (es) 2012-12-19
US20020061873A1 (en) 2002-05-23
IL144512A0 (en) 2002-05-23
US20140056974A1 (en) 2014-02-27
KR100880859B1 (ko) 2009-01-30
PL198330B1 (pl) 2008-06-30
CZ303979B6 (cs) 2013-07-31
JP2012111763A (ja) 2012-06-14
HK1045807A1 (en) 2002-12-13
WO2000048571A1 (en) 2000-08-24
CA2362277C (en) 2010-03-30

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