NO330531B1 - Pyrimidylsulfonamidderivater som kemokinreseptormodulatorer, og fremgangsmate fremstilling derav. - Google Patents

Pyrimidylsulfonamidderivater som kemokinreseptormodulatorer, og fremgangsmate fremstilling derav. Download PDF

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Publication number
NO330531B1
NO330531B1 NO20051042A NO20051042A NO330531B1 NO 330531 B1 NO330531 B1 NO 330531B1 NO 20051042 A NO20051042 A NO 20051042A NO 20051042 A NO20051042 A NO 20051042A NO 330531 B1 NO330531 B1 NO 330531B1
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Prior art keywords
amino
compound
hydroxy
pyrimidin
yield
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NO20051042A
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English (en)
Norwegian (no)
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NO20051042L (no
Inventor
Colin Bennion
Premji Meghani
Roger Victor Bonnert
Antony Ronald Cook
Mark Richard Ebden
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Astrazeneca Ab
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Publication of NO20051042L publication Critical patent/NO20051042L/no
Publication of NO330531B1 publication Critical patent/NO330531B1/no

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    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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NO20051042A 2002-07-27 2005-02-25 Pyrimidylsulfonamidderivater som kemokinreseptormodulatorer, og fremgangsmate fremstilling derav. NO330531B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0217431.6A GB0217431D0 (en) 2002-07-27 2002-07-27 Novel compounds
PCT/GB2003/003175 WO2004011443A1 (en) 2002-07-27 2003-07-23 Pyrimidyl sulphone amide derivatives as chemokine receptor modulators

Publications (2)

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NO20051042L NO20051042L (no) 2005-03-31
NO330531B1 true NO330531B1 (no) 2011-05-09

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NO20051042A NO330531B1 (no) 2002-07-27 2005-02-25 Pyrimidylsulfonamidderivater som kemokinreseptormodulatorer, og fremgangsmate fremstilling derav.

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US (2) US7582644B2 (ru)
EP (1) EP1527051B1 (ru)
JP (1) JP4619782B2 (ru)
KR (2) KR101074626B1 (ru)
CN (1) CN100345829C (ru)
AR (1) AR040700A1 (ru)
AU (1) AU2003281684B2 (ru)
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HK (1) HK1076465A1 (ru)
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NO (1) NO330531B1 (ru)
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TW (1) TWI340038B (ru)
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Families Citing this family (28)

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Publication number Priority date Publication date Assignee Title
GB0217431D0 (en) * 2002-07-27 2002-09-04 Astrazeneca Ab Novel compounds
DE60318219T2 (de) 2002-08-24 2009-01-15 Astrazeneca Ab PYRIMIDINDERIVATE ALS MODULATOREN DER AKTIVITuT VON CHEMOKINREZEPTOREN
GB0401269D0 (en) * 2004-01-21 2004-02-25 Astrazeneca Ab Compounds
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