NO330521B1 - Substituerte etynylfenyl-1,8-naftyridin-4(1H)-on-forbindelser som er fosfodiesterase-4-inhibitorer, farmasoytiske preparater som omfatter forbindelsene, samt anvendelse av forbindelsene ved fremstilling av medikamenter - Google Patents

Substituerte etynylfenyl-1,8-naftyridin-4(1H)-on-forbindelser som er fosfodiesterase-4-inhibitorer, farmasoytiske preparater som omfatter forbindelsene, samt anvendelse av forbindelsene ved fremstilling av medikamenter Download PDF

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Publication number
NO330521B1
NO330521B1 NO20041293A NO20041293A NO330521B1 NO 330521 B1 NO330521 B1 NO 330521B1 NO 20041293 A NO20041293 A NO 20041293A NO 20041293 A NO20041293 A NO 20041293A NO 330521 B1 NO330521 B1 NO 330521B1
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NO
Norway
Prior art keywords
dihydro
carboxamide
phenyl
naphthyridin
isopropyl
Prior art date
Application number
NO20041293A
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English (en)
Norwegian (no)
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NO20041293D0 (no
NO20041293L (no
Inventor
Mario Girard
Daniel Guay
Richard Friesen
Pierre Hamel
Sebastien Laliberte
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Merck Frosst Canada Ltd
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Publication of NO20041293D0 publication Critical patent/NO20041293D0/no
Publication of NO20041293L publication Critical patent/NO20041293L/no
Publication of NO330521B1 publication Critical patent/NO330521B1/no

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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NO20041293A 2001-08-29 2004-03-26 Substituerte etynylfenyl-1,8-naftyridin-4(1H)-on-forbindelser som er fosfodiesterase-4-inhibitorer, farmasoytiske preparater som omfatter forbindelsene, samt anvendelse av forbindelsene ved fremstilling av medikamenter NO330521B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31609301P 2001-08-29 2001-08-29
PCT/CA2002/001324 WO2003018579A1 (en) 2001-08-29 2002-08-27 Alkyne-aryl phosphodiesterase-4 inhibitors

Publications (3)

Publication Number Publication Date
NO20041293D0 NO20041293D0 (no) 2004-03-26
NO20041293L NO20041293L (no) 2004-05-27
NO330521B1 true NO330521B1 (no) 2011-05-09

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NO20041293A NO330521B1 (no) 2001-08-29 2004-03-26 Substituerte etynylfenyl-1,8-naftyridin-4(1H)-on-forbindelser som er fosfodiesterase-4-inhibitorer, farmasoytiske preparater som omfatter forbindelsene, samt anvendelse av forbindelsene ved fremstilling av medikamenter

Country Status (28)

Country Link
US (2) US6743802B2 (ja)
EP (2) EP2305677A1 (ja)
JP (1) JP4157035B2 (ja)
KR (1) KR100928849B1 (ja)
CN (1) CN100338061C (ja)
AR (1) AR036365A1 (ja)
AU (1) AU2002322940B2 (ja)
BR (1) BR0212042A (ja)
CA (1) CA2456817C (ja)
DO (1) DOP2002000456A (ja)
EA (1) EA006800B1 (ja)
EC (1) ECSP044992A (ja)
GE (1) GEP20063805B (ja)
HK (1) HK1080073B (ja)
HR (1) HRP20040151A2 (ja)
HU (1) HUP0401729A3 (ja)
IL (1) IL160213A0 (ja)
IS (1) IS7138A (ja)
JO (1) JO2311B1 (ja)
MX (1) MXPA04001889A (ja)
NO (1) NO330521B1 (ja)
NZ (1) NZ530931A (ja)
PE (1) PE20030416A1 (ja)
PL (1) PL367716A1 (ja)
RS (1) RS17004A (ja)
UA (1) UA75957C2 (ja)
WO (1) WO2003018579A1 (ja)
ZA (1) ZA200400952B (ja)

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