NO328211B1 - Intraokulaere trykksenkende preparater for topisk administrering omfattende en angiotensin II-antagonist, en borsyre og en etylendiamintetraeddiksyre. - Google Patents
Intraokulaere trykksenkende preparater for topisk administrering omfattende en angiotensin II-antagonist, en borsyre og en etylendiamintetraeddiksyre. Download PDFInfo
- Publication number
- NO328211B1 NO328211B1 NO20016023A NO20016023A NO328211B1 NO 328211 B1 NO328211 B1 NO 328211B1 NO 20016023 A NO20016023 A NO 20016023A NO 20016023 A NO20016023 A NO 20016023A NO 328211 B1 NO328211 B1 NO 328211B1
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- Prior art keywords
- groups
- salts
- intraocular pressure
- methyl
- acid
- Prior art date
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- 239000004327 boric acid Substances 0.000 title claims abstract description 16
- 229940123413 Angiotensin II antagonist Drugs 0.000 title claims abstract description 14
- 239000002333 angiotensin II receptor antagonist Substances 0.000 title claims abstract description 14
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- 238000002360 preparation method Methods 0.000 claims description 49
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- 102400000344 Angiotensin-1 Human genes 0.000 claims 1
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/0012—Galenical forms characterised by the site of application
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- A61P27/00—Drugs for disorders of the senses
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
Landscapes
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- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Materials For Medical Uses (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP16494599 | 1999-06-11 | ||
| PCT/JP2000/003779 WO2000076543A1 (fr) | 1999-06-11 | 2000-06-09 | Composition permettant de reduire la tension oculaire et destinee a l'administration topique |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20016023D0 NO20016023D0 (no) | 2001-12-10 |
| NO20016023L NO20016023L (no) | 2002-01-29 |
| NO328211B1 true NO328211B1 (no) | 2010-01-11 |
Family
ID=15802847
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20016023A NO328211B1 (no) | 1999-06-11 | 2001-12-10 | Intraokulaere trykksenkende preparater for topisk administrering omfattende en angiotensin II-antagonist, en borsyre og en etylendiamintetraeddiksyre. |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6777436B2 (tr) |
| EP (1) | EP1186302B1 (tr) |
| KR (1) | KR100611543B1 (tr) |
| CN (1) | CN1198650C (tr) |
| AT (1) | ATE295721T1 (tr) |
| AU (1) | AU759513B2 (tr) |
| BR (1) | BR0011477A (tr) |
| CA (1) | CA2376780C (tr) |
| CZ (1) | CZ300553B6 (tr) |
| DE (1) | DE60020230T2 (tr) |
| ES (1) | ES2242619T3 (tr) |
| HK (1) | HK1042050A1 (tr) |
| HU (1) | HUP0201466A3 (tr) |
| IL (2) | IL146917A0 (tr) |
| MX (1) | MXPA01012752A (tr) |
| NO (1) | NO328211B1 (tr) |
| NZ (1) | NZ516033A (tr) |
| PL (1) | PL200009B1 (tr) |
| PT (1) | PT1186302E (tr) |
| RU (1) | RU2227740C2 (tr) |
| TR (1) | TR200103603T2 (tr) |
| TW (1) | TWI245639B (tr) |
| WO (1) | WO2000076543A1 (tr) |
| ZA (1) | ZA200109943B (tr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4000505B2 (ja) * | 1999-12-01 | 2007-10-31 | 第一三共株式会社 | 緑内障を治療するための併用剤 |
| TW200304812A (en) * | 2002-03-08 | 2003-10-16 | Sankyo Co | An eye drop containing a tetrazole derivative |
| US20050119299A1 (en) * | 2002-03-08 | 2005-06-02 | Sankyo Company, Limited | Ophthalmic solutions containing tetrazole derivatives |
| PL1872783T3 (pl) * | 2005-04-21 | 2012-05-31 | Santen Pharmaceutical Co Ltd | Środek leczniczy w schorzeniach rogówkowo-spojówkowych |
| ES2394130T3 (es) | 2007-11-30 | 2013-01-22 | Toltec Pharmaceuticals, Llc | Composiciones y métodos para tratar infecciones vaginales y biopelículas vaginales patógenas |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1991015206A1 (en) * | 1990-04-05 | 1991-10-17 | E.I. Du Pont De Nemours And Company | Treatment of glaucoma and ocular hypertension with imidazole angiotensin-ii receptor antagonists |
| CZ154994A3 (en) * | 1993-07-02 | 1995-09-13 | Senju Pharma Co | Visual hypotensive agent |
| CN1140409A (zh) * | 1994-02-08 | 1997-01-15 | 希巴-盖吉股份公司 | 血管紧张素ii拮抗剂对正常眼压性青光眼的治疗 |
| DK0795326T3 (da) * | 1994-03-16 | 2001-11-26 | Sankyo Co | Okulærtensionssænkende middel |
| JPH07324034A (ja) * | 1994-05-30 | 1995-12-12 | Toa Yakuhin Kk | フマル酸ケトチフェン含有の点眼剤 |
-
2000
- 2000-06-09 TW TW089111297A patent/TWI245639B/zh not_active IP Right Cessation
- 2000-06-09 ES ES00935630T patent/ES2242619T3/es not_active Expired - Lifetime
- 2000-06-09 AU AU51086/00A patent/AU759513B2/en not_active Ceased
- 2000-06-09 NZ NZ516033A patent/NZ516033A/en not_active IP Right Cessation
- 2000-06-09 HU HU0201466A patent/HUP0201466A3/hu unknown
- 2000-06-09 CA CA002376780A patent/CA2376780C/en not_active Expired - Fee Related
- 2000-06-09 PL PL352161A patent/PL200009B1/pl not_active IP Right Cessation
- 2000-06-09 IL IL14691700A patent/IL146917A0/xx active IP Right Grant
- 2000-06-09 PT PT00935630T patent/PT1186302E/pt unknown
- 2000-06-09 EP EP00935630A patent/EP1186302B1/en not_active Expired - Lifetime
- 2000-06-09 BR BR0011477-4A patent/BR0011477A/pt not_active Application Discontinuation
- 2000-06-09 WO PCT/JP2000/003779 patent/WO2000076543A1/ja not_active Application Discontinuation
- 2000-06-09 AT AT00935630T patent/ATE295721T1/de not_active IP Right Cessation
- 2000-06-09 MX MXPA01012752A patent/MXPA01012752A/es active IP Right Grant
- 2000-06-09 TR TR2001/03603T patent/TR200103603T2/tr unknown
- 2000-06-09 RU RU2001133273/15A patent/RU2227740C2/ru not_active IP Right Cessation
- 2000-06-09 DE DE60020230T patent/DE60020230T2/de not_active Expired - Lifetime
- 2000-06-09 CN CNB008113513A patent/CN1198650C/zh not_active Expired - Fee Related
- 2000-06-09 KR KR1020017015901A patent/KR100611543B1/ko not_active IP Right Cessation
- 2000-06-09 CZ CZ20014415A patent/CZ300553B6/cs not_active IP Right Cessation
-
2001
- 2001-12-03 ZA ZA200109943A patent/ZA200109943B/en unknown
- 2001-12-04 IL IL146917A patent/IL146917A/en not_active IP Right Cessation
- 2001-12-10 NO NO20016023A patent/NO328211B1/no not_active IP Right Cessation
- 2001-12-10 US US10/016,535 patent/US6777436B2/en not_active Expired - Fee Related
-
2002
- 2002-05-23 HK HK02103878A patent/HK1042050A1/xx not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |