NO312463B1 - Pyrimid [4,5-b] indoler og forbindelser - Google Patents
Pyrimid [4,5-b] indoler og forbindelser Download PDFInfo
- Publication number
- NO312463B1 NO312463B1 NO19993359A NO993359A NO312463B1 NO 312463 B1 NO312463 B1 NO 312463B1 NO 19993359 A NO19993359 A NO 19993359A NO 993359 A NO993359 A NO 993359A NO 312463 B1 NO312463 B1 NO 312463B1
- Authority
- NO
- Norway
- Prior art keywords
- pyrrolidinyl
- pyrimido
- acetic acid
- indol
- indoles
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/12—Mucolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Ophthalmology & Optometry (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3522397P | 1997-01-08 | 1997-01-08 | |
| US4374997P | 1997-04-09 | 1997-04-09 | |
| PCT/US1997/024300 WO1998042708A2 (en) | 1997-01-08 | 1997-12-19 | Pharmaceutically active tricyclic amines |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO993359D0 NO993359D0 (no) | 1999-07-07 |
| NO993359L NO993359L (no) | 1999-09-07 |
| NO312463B1 true NO312463B1 (no) | 2002-05-13 |
Family
ID=26711898
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19993359A NO312463B1 (no) | 1997-01-08 | 1999-07-07 | Pyrimid [4,5-b] indoler og forbindelser |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US5932728A (cs) |
| EP (1) | EP0964865B1 (cs) |
| JP (1) | JP2002511061A (cs) |
| KR (1) | KR20000069940A (cs) |
| CN (1) | CN1128798C (cs) |
| AT (1) | ATE233763T1 (cs) |
| AU (1) | AU723709B2 (cs) |
| CA (1) | CA2275389A1 (cs) |
| CZ (1) | CZ288076B6 (cs) |
| DE (1) | DE69719563T2 (cs) |
| DK (1) | DK0964865T3 (cs) |
| ES (1) | ES2193424T3 (cs) |
| FI (1) | FI991568A7 (cs) |
| HU (1) | HUP0003692A3 (cs) |
| NO (1) | NO312463B1 (cs) |
| NZ (1) | NZ336659A (cs) |
| PL (1) | PL334451A1 (cs) |
| PT (1) | PT964865E (cs) |
| RU (1) | RU2200737C2 (cs) |
| SI (1) | SI0964865T1 (cs) |
| SK (1) | SK283378B6 (cs) |
| WO (1) | WO1998042708A2 (cs) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020147216A1 (en) * | 2000-01-31 | 2002-10-10 | Yuhong Zhou | Mucin synthesis inhibitors |
| US7345051B2 (en) | 2000-01-31 | 2008-03-18 | Genaera Corporation | Mucin synthesis inhibitors |
| US6737427B2 (en) * | 2000-01-31 | 2004-05-18 | Genaera Corporation | Mucin synthesis inhibitors |
| JP2005515173A (ja) * | 2001-10-31 | 2005-05-26 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | ピリミド[4,5−b]インドール誘導体 |
| WO2004058764A1 (en) * | 2002-12-27 | 2004-07-15 | Bayer Healthcare Ag | 4-phenyl-pyrimido [4,5-b] indole derivatives |
| WO2011011186A2 (en) * | 2009-07-22 | 2011-01-27 | The Board Of Trustees Of The University Of Illinois | Hdac inhibitors and therapeutic methods using the same |
| BR112013023266B8 (pt) | 2011-03-15 | 2021-04-06 | L Livermore Nat Security Llc | inibidores da girase tricíclicos |
| SG11201404241SA (en) | 2012-01-27 | 2014-08-28 | Univ Montreal | Pyrimido[4,5-b]indole derivatives and use thereof in the expansion of hematopoietic stem cells |
| JP6954844B2 (ja) | 2015-06-05 | 2021-10-27 | エマ−ケベック | 造血幹細胞を培養するため及び/又は造血幹細胞を前駆体へ分化させるための方法及びその使用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK0633886T3 (da) * | 1992-04-03 | 2000-12-18 | Upjohn Co | Farmaceutisk aktive bicyclisk-heterocycliske aminer |
| US5502187A (en) * | 1992-04-03 | 1996-03-26 | The Upjohn Company | Pharmaceutically active bicyclic-heterocyclic amines |
| US5795986A (en) * | 1995-03-02 | 1998-08-18 | Pharmacia & Upjohn Company | Pyrimido 4,5-B!indoles |
-
1997
- 1997-12-19 NZ NZ336659A patent/NZ336659A/xx unknown
- 1997-12-19 RU RU99117141/04A patent/RU2200737C2/ru not_active IP Right Cessation
- 1997-12-19 HU HU0003692A patent/HUP0003692A3/hu unknown
- 1997-12-19 CN CN97180464A patent/CN1128798C/zh not_active Expired - Fee Related
- 1997-12-19 SK SK901-99A patent/SK283378B6/sk unknown
- 1997-12-19 DK DK97955063T patent/DK0964865T3/da active
- 1997-12-19 CA CA002275389A patent/CA2275389A1/en not_active Abandoned
- 1997-12-19 FI FI991568A patent/FI991568A7/fi unknown
- 1997-12-19 WO PCT/US1997/024300 patent/WO1998042708A2/en not_active Application Discontinuation
- 1997-12-19 CZ CZ19992388A patent/CZ288076B6/cs not_active IP Right Cessation
- 1997-12-19 KR KR1019997006153A patent/KR20000069940A/ko not_active Ceased
- 1997-12-19 DE DE69719563T patent/DE69719563T2/de not_active Expired - Fee Related
- 1997-12-19 PT PT97955063T patent/PT964865E/pt unknown
- 1997-12-19 PL PL97334451A patent/PL334451A1/xx unknown
- 1997-12-19 AT AT97955063T patent/ATE233763T1/de not_active IP Right Cessation
- 1997-12-19 AU AU86554/98A patent/AU723709B2/en not_active Ceased
- 1997-12-19 JP JP54567998A patent/JP2002511061A/ja not_active Withdrawn
- 1997-12-19 ES ES97955063T patent/ES2193424T3/es not_active Expired - Lifetime
- 1997-12-19 EP EP97955063A patent/EP0964865B1/en not_active Expired - Lifetime
- 1997-12-19 US US08/994,901 patent/US5932728A/en not_active Expired - Fee Related
- 1997-12-19 SI SI9730521T patent/SI0964865T1/xx unknown
-
1999
- 1999-07-07 NO NO19993359A patent/NO312463B1/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO1998042708A2 (en) | 1998-10-01 |
| DK0964865T3 (da) | 2003-05-05 |
| RU2200737C2 (ru) | 2003-03-20 |
| EP0964865B1 (en) | 2003-03-05 |
| CA2275389A1 (en) | 1998-10-01 |
| HUP0003692A2 (hu) | 2001-04-28 |
| CN1239961A (zh) | 1999-12-29 |
| PT964865E (pt) | 2003-06-30 |
| AU8655498A (en) | 1998-10-20 |
| SI0964865T1 (en) | 2003-08-31 |
| DE69719563D1 (de) | 2003-04-10 |
| AU723709B2 (en) | 2000-09-07 |
| DE69719563T2 (de) | 2003-11-27 |
| CN1128798C (zh) | 2003-11-26 |
| KR20000069940A (ko) | 2000-11-25 |
| JP2002511061A (ja) | 2002-04-09 |
| US5932728A (en) | 1999-08-03 |
| NZ336659A (en) | 2001-01-26 |
| FI991568L (fi) | 1999-07-08 |
| HUP0003692A3 (en) | 2002-10-28 |
| NO993359D0 (no) | 1999-07-07 |
| SK90199A3 (en) | 2000-05-16 |
| EP0964865A2 (en) | 1999-12-22 |
| ES2193424T3 (es) | 2003-11-01 |
| PL334451A1 (en) | 2000-02-28 |
| CZ288076B6 (cs) | 2001-04-11 |
| SK283378B6 (sk) | 2003-06-03 |
| NO993359L (no) | 1999-09-07 |
| FI991568A7 (fi) | 1999-07-08 |
| HK1023344A1 (en) | 2000-09-08 |
| WO1998042708A3 (en) | 1998-12-17 |
| ATE233763T1 (de) | 2003-03-15 |
| CZ238899A3 (cs) | 1999-10-13 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| KR100341190B1 (ko) | 피페리딘및피페라진 | |
| DK174161B1 (da) | Anellerede indolderivater, fremgangsmåde til deres fremstilling og fremgangsmåde til fremstilling af farmaceutisk præparat indeholdende dem | |
| AU2009253978B2 (en) | 3,4-dihydropyrimidine TRPA1 antagonists | |
| EP2081572A1 (en) | Benzimidazole cannabinoid agonists bearing a substituted heterocyclic group | |
| JP2002542245A (ja) | 置換イミダゾール、それらの製造および使用 | |
| SK67699A3 (en) | Novel substituted pyrazole derivatives for the treatment of cardiocirculatory diseases | |
| JPH04235974A (ja) | 新規なイミダゾール誘導体、それらの製造法、得られる新規な中間体、それらの薬剤としての使用及びそれらを含有する製薬組成物 | |
| TW201111374A (en) | Compounds which selectively modulate the CB2 receptor | |
| AU2019272383B2 (en) | P-Phenylenediamine Derivative As Potassium Channel Regulator And Preparation Method And Medical Application Thereof | |
| NO175978B (no) | Analogifremgangsmåte for fremstilling av terapeutisk aktive bis-aza-bicykliske forbindelser | |
| KR20190033538A (ko) | 이미다조피리딘아민 페닐 유도체 및 그의 용도 | |
| JP2024540080A (ja) | Irak4分解剤およびその合成 | |
| NO312463B1 (no) | Pyrimid [4,5-b] indoler og forbindelser | |
| EP3418277B1 (en) | Substituted amino six-membered nitric heterocyclic ring compound and preparation and use thereof | |
| DK163581B (da) | Kondenserede pyrazol-3-oxo-propannitrilderivater og fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende forbindelserne | |
| NO172490B (no) | Analogifremgangsmaate for fremstilling av terapeutisk aktive 1,4-disubstituerte piperazinderivater | |
| NO873108L (no) | Fremgangsmaate for fremstilling av terapeutisk aktive 1,4-benzodiazepiner. | |
| KR20060010839A (ko) | 세로토닌 재흡수 저해제로서의 인돌 유도체 | |
| IE56839B1 (en) | New 1h,3h-pyrrolo(1,2-c)thiazole derivatives,their preparation and compositions containing them | |
| DK142321B (da) | Analogifremgangsmåde til fremstilling af D-6-methyl-8-(2-methylsulfinylethyl)-ergolin og syreadditionssalte deraf. | |
| WO2000006575A2 (en) | Azabicyclic compounds | |
| NO830758L (no) | Analogifremgangsmaate for fremstilling av terapeutisk aktive 4-fenyl-4,5,6,7-tetrahydro tieno (2,3-c) pyridin-derivater | |
| AU651171B2 (en) | Oxazinobenzazole compounds | |
| DK143752B (da) | Analogifremgangsmaade til fremstilling af pyridobenzodiazepinoner eller farmakologisk acceptable salte deraf | |
| DK165878B (da) | 3-substituerede-5-aminoalkyl-beta-carbolinderivater og fremgangsmaade til deres fremstilling |